ATE278665T1 - Verfahren zur herstellung von n-acyl-3,4- dehydroprolin und n-acyl-3,4-dehydropiperidin-2- carbonsäure derivaten - Google Patents
Verfahren zur herstellung von n-acyl-3,4- dehydroprolin und n-acyl-3,4-dehydropiperidin-2- carbonsäure derivatenInfo
- Publication number
- ATE278665T1 ATE278665T1 AT00918809T AT00918809T ATE278665T1 AT E278665 T1 ATE278665 T1 AT E278665T1 AT 00918809 T AT00918809 T AT 00918809T AT 00918809 T AT00918809 T AT 00918809T AT E278665 T1 ATE278665 T1 AT E278665T1
- Authority
- AT
- Austria
- Prior art keywords
- acyl
- dehydropiperidine
- dehydroproline
- producing
- carboxylic acid
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000006823 (C1-C6) acyl group Chemical group 0.000 abstract 1
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004170 methylsulfonyl group Chemical group [H]C([H])([H])S(*)(=O)=O 0.000 abstract 1
- 125000003170 phenylsulfonyl group Chemical group C1(=CC=CC=C1)S(=O)(=O)* 0.000 abstract 1
- 125000002088 tosyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1C([H])([H])[H])S(*)(=O)=O 0.000 abstract 1
- 125000004044 trifluoroacetyl group Chemical group FC(C(=O)*)(F)F 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/20—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pyrrole Compounds (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19913699A DE19913699A1 (de) | 1999-03-26 | 1999-03-26 | Verfahren zur Herstellung von 3,4-Dihydroprolinen und 3,4-Dehydropiperidinen |
| PCT/EP2000/002377 WO2000058284A1 (de) | 1999-03-26 | 2000-03-17 | Verfahren zur herstellung von n-acyl-3,4 - dehydroprolin und n-acyl-3,4 - dehydropiperidin-2-carbonsäure derivaten |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE278665T1 true ATE278665T1 (de) | 2004-10-15 |
Family
ID=7902464
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00918809T ATE278665T1 (de) | 1999-03-26 | 2000-03-17 | Verfahren zur herstellung von n-acyl-3,4- dehydroprolin und n-acyl-3,4-dehydropiperidin-2- carbonsäure derivaten |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US6579971B1 (enExample) |
| EP (1) | EP1165509B1 (enExample) |
| JP (1) | JP3868210B2 (enExample) |
| KR (1) | KR20010104730A (enExample) |
| CN (1) | CN1345310A (enExample) |
| AT (1) | ATE278665T1 (enExample) |
| AU (1) | AU3962500A (enExample) |
| BR (1) | BR0009330A (enExample) |
| CA (1) | CA2368479C (enExample) |
| CZ (1) | CZ20013456A3 (enExample) |
| DE (2) | DE19913699A1 (enExample) |
| ES (1) | ES2230088T3 (enExample) |
| HK (1) | HK1045156A1 (enExample) |
| HU (1) | HUP0200420A2 (enExample) |
| IL (1) | IL145525A0 (enExample) |
| MX (1) | MXPA01009679A (enExample) |
| NO (1) | NO20014645L (enExample) |
| RU (1) | RU2001129097A (enExample) |
| TR (1) | TR200102747T2 (enExample) |
| TW (1) | TWI276626B (enExample) |
| WO (1) | WO2000058284A1 (enExample) |
| ZA (1) | ZA200107629B (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN100396666C (zh) * | 2005-12-14 | 2008-06-25 | 郑州大学 | （4s）-1-叔丁氧羰基-4-氨基-l-脯氨酸乙酯及其合成工艺 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4291040A (en) * | 1979-10-22 | 1981-09-22 | E. R. Squibb & Sons, Inc. | Mercaptoacyl derivatives of 4-disubstituted prolines and 4-substituted dehydroprolines |
| US5580575A (en) | 1989-12-22 | 1996-12-03 | Imarx Pharmaceutical Corp. | Therapeutic drug delivery systems |
| JPH09502191A (ja) | 1993-09-09 | 1997-03-04 | シエーリング アクチエンゲゼルシヤフト | 作用物質およびガスを含有する微粒子 |
| DE19630082A1 (de) * | 1996-07-26 | 1998-01-29 | Basf Ag | Verfahren zur Herstellung von 3-Pyrrolin-2-carbonsäure-Derivaten |
| US6090800A (en) | 1997-05-06 | 2000-07-18 | Imarx Pharmaceutical Corp. | Lipid soluble steroid prodrugs |
| DE19723473A1 (de) * | 1997-06-04 | 1998-12-10 | Basf Ag | Verfahren zur Herstellung von chiralen 3,4-Didehydroprolinen |
| CA2319433C (en) | 1998-02-09 | 2008-04-22 | Bracco Research S.A. | Targeted delivery of biologically active media |
-
1999
- 1999-03-26 DE DE19913699A patent/DE19913699A1/de not_active Withdrawn
-
2000
- 2000-03-09 TW TW089104251A patent/TWI276626B/zh not_active IP Right Cessation
- 2000-03-17 US US09/937,312 patent/US6579971B1/en not_active Expired - Lifetime
- 2000-03-17 BR BR0009330-0A patent/BR0009330A/pt not_active IP Right Cessation
- 2000-03-17 CN CN00805579A patent/CN1345310A/zh active Pending
- 2000-03-17 CA CA002368479A patent/CA2368479C/en not_active Expired - Fee Related
- 2000-03-17 DE DE50008117T patent/DE50008117D1/de not_active Expired - Fee Related
- 2000-03-17 RU RU2001129097/04A patent/RU2001129097A/ru unknown
- 2000-03-17 EP EP00918809A patent/EP1165509B1/de not_active Expired - Lifetime
- 2000-03-17 HU HU0200420A patent/HUP0200420A2/hu unknown
- 2000-03-17 ES ES00918809T patent/ES2230088T3/es not_active Expired - Lifetime
- 2000-03-17 AT AT00918809T patent/ATE278665T1/de not_active IP Right Cessation
- 2000-03-17 CZ CZ20013456A patent/CZ20013456A3/cs unknown
- 2000-03-17 HK HK02106153.8A patent/HK1045156A1/zh unknown
- 2000-03-17 JP JP2000607987A patent/JP3868210B2/ja not_active Expired - Fee Related
- 2000-03-17 TR TR2001/02747T patent/TR200102747T2/xx unknown
- 2000-03-17 MX MXPA01009679A patent/MXPA01009679A/es unknown
- 2000-03-17 KR KR1020017012187A patent/KR20010104730A/ko not_active Abandoned
- 2000-03-17 AU AU39625/00A patent/AU3962500A/en not_active Abandoned
- 2000-03-17 WO PCT/EP2000/002377 patent/WO2000058284A1/de not_active Ceased
- 2000-03-17 IL IL14552599A patent/IL145525A0/xx unknown
-
2001
- 2001-09-17 ZA ZA200107629A patent/ZA200107629B/en unknown
- 2001-09-25 NO NO20014645A patent/NO20014645L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2001129097A (ru) | 2004-03-20 |
| CZ20013456A3 (cs) | 2002-05-15 |
| AU3962500A (en) | 2000-10-16 |
| NO20014645D0 (no) | 2001-09-25 |
| MXPA01009679A (es) | 2002-03-14 |
| EP1165509B1 (de) | 2004-10-06 |
| KR20010104730A (ko) | 2001-11-26 |
| CA2368479C (en) | 2005-03-01 |
| WO2000058284A1 (de) | 2000-10-05 |
| TWI276626B (en) | 2007-03-21 |
| CN1345310A (zh) | 2002-04-17 |
| NO20014645L (no) | 2001-09-25 |
| HUP0200420A2 (hu) | 2002-05-29 |
| CA2368479A1 (en) | 2000-10-05 |
| TR200102747T2 (tr) | 2002-02-21 |
| ES2230088T3 (es) | 2005-05-01 |
| BR0009330A (pt) | 2002-01-08 |
| IL145525A0 (en) | 2002-06-30 |
| ZA200107629B (en) | 2002-09-17 |
| DE50008117D1 (de) | 2004-11-11 |
| EP1165509A1 (de) | 2002-01-02 |
| JP2002540190A (ja) | 2002-11-26 |
| US6579971B1 (en) | 2003-06-17 |
| HK1045156A1 (zh) | 2002-11-15 |
| JP3868210B2 (ja) | 2007-01-17 |
| DE19913699A1 (de) | 2000-09-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| REN | Ceased due to non-payment of the annual fee |