ATE204281T1 - Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungen - Google Patents
Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungenInfo
- Publication number
- ATE204281T1 ATE204281T1 AT95922295T AT95922295T ATE204281T1 AT E204281 T1 ATE204281 T1 AT E204281T1 AT 95922295 T AT95922295 T AT 95922295T AT 95922295 T AT95922295 T AT 95922295T AT E204281 T1 ATE204281 T1 AT E204281T1
- Authority
- AT
- Austria
- Prior art keywords
- hydrogen
- rapamycinamidinocarbamates
- alkynyl
- alkenyl
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Transplantation (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/259,763 US5463048A (en) | 1994-06-14 | 1994-06-14 | Rapamycin amidino carbamates |
PCT/US1995/007412 WO1995034565A1 (en) | 1994-06-14 | 1995-06-09 | Rapamycin amidino carbamates and pharmaceutical compositions containing them |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE204281T1 true ATE204281T1 (de) | 2001-09-15 |
Family
ID=22986267
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT95922295T ATE204281T1 (de) | 1994-06-14 | 1995-06-09 | Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungen |
Country Status (13)
Country | Link |
---|---|
US (5) | US5463048A (de) |
EP (1) | EP0765329B1 (de) |
JP (1) | JPH10501268A (de) |
AT (1) | ATE204281T1 (de) |
AU (1) | AU2703295A (de) |
CA (1) | CA2192972A1 (de) |
DE (1) | DE69522225T2 (de) |
DK (1) | DK0765329T3 (de) |
ES (1) | ES2159641T3 (de) |
GR (1) | GR3036940T3 (de) |
HK (1) | HK1011030A1 (de) |
PT (1) | PT765329E (de) |
WO (1) | WO1995034565A1 (de) |
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US6331537B1 (en) | 1998-06-03 | 2001-12-18 | Gpi Nil Holdings, Inc. | Carboxylic acids and carboxylic acid isosteres of N-heterocyclic compounds |
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1994
- 1994-06-14 US US08/259,763 patent/US5463048A/en not_active Expired - Lifetime
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1995
- 1995-05-24 US US08/448,902 patent/US5541192A/en not_active Expired - Lifetime
- 1995-05-24 US US08/450,772 patent/US5637590A/en not_active Expired - Lifetime
- 1995-05-24 US US08/450,771 patent/US5508286A/en not_active Expired - Lifetime
- 1995-05-24 US US08/448,866 patent/US5541191A/en not_active Expired - Lifetime
- 1995-06-09 JP JP8502371A patent/JPH10501268A/ja not_active Withdrawn
- 1995-06-09 CA CA002192972A patent/CA2192972A1/en not_active Abandoned
- 1995-06-09 AT AT95922295T patent/ATE204281T1/de not_active IP Right Cessation
- 1995-06-09 PT PT95922295T patent/PT765329E/pt unknown
- 1995-06-09 WO PCT/US1995/007412 patent/WO1995034565A1/en active IP Right Grant
- 1995-06-09 DK DK95922295T patent/DK0765329T3/da active
- 1995-06-09 ES ES95922295T patent/ES2159641T3/es not_active Expired - Lifetime
- 1995-06-09 AU AU27032/95A patent/AU2703295A/en not_active Abandoned
- 1995-06-09 DE DE69522225T patent/DE69522225T2/de not_active Expired - Fee Related
- 1995-06-09 EP EP95922295A patent/EP0765329B1/de not_active Expired - Lifetime
-
1998
- 1998-11-24 HK HK98112280A patent/HK1011030A1/xx not_active IP Right Cessation
-
2001
- 2001-10-18 GR GR20010401809T patent/GR3036940T3/el not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP0765329B1 (de) | 2001-08-16 |
US5541192A (en) | 1996-07-30 |
CA2192972A1 (en) | 1995-12-21 |
EP0765329A1 (de) | 1997-04-02 |
WO1995034565A1 (en) | 1995-12-21 |
DK0765329T3 (da) | 2001-10-08 |
ES2159641T3 (es) | 2001-10-16 |
US5541191A (en) | 1996-07-30 |
AU2703295A (en) | 1996-01-05 |
JPH10501268A (ja) | 1998-02-03 |
HK1011030A1 (en) | 1999-07-02 |
DE69522225D1 (de) | 2001-09-20 |
GR3036940T3 (en) | 2002-01-31 |
US5463048A (en) | 1995-10-31 |
DE69522225T2 (de) | 2002-03-21 |
US5637590A (en) | 1997-06-10 |
PT765329E (pt) | 2001-12-28 |
US5508286A (en) | 1996-04-16 |
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