ATE183993T1 - Zwischenprodukte für die herstellung einer substituierten 2,5-diamino-3-hydroxyhexan. - Google Patents

Zwischenprodukte für die herstellung einer substituierten 2,5-diamino-3-hydroxyhexan.

Info

Publication number
ATE183993T1
ATE183993T1 AT94929340T AT94929340T ATE183993T1 AT E183993 T1 ATE183993 T1 AT E183993T1 AT 94929340 T AT94929340 T AT 94929340T AT 94929340 T AT94929340 T AT 94929340T AT E183993 T1 ATE183993 T1 AT E183993T1
Authority
AT
Austria
Prior art keywords
loweralkyl
independently selected
alkoxy
hydrogen
substituted
Prior art date
Application number
AT94929340T
Other languages
English (en)
Inventor
Timothy L Stuk
Francis A J Kerdesky
Linda M Lijewski
Daniel W Norbeck
David Scarpetti
Jien-Heh J Tien
Michael S Allen
Denton C Langridge
Laura Melcher
Daniel S Reno
Hing Leung Sham
Chen Zhao
Anthony R Haight
M Robert Leanna
Howard E Morton
Timothy A Robbins
Thomas J Sowin
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Application granted granted Critical
Publication of ATE183993T1 publication Critical patent/ATE183993T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04Ortho- or peri-condensed ring systems
    • C07D221/06Ring systems of three rings
    • C07D221/14Aza-phenalenes, e.g. 1,8-naphthalimide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/22Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C225/00Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
    • C07C225/02Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C225/14Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
    • C07C225/16Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32Oximes
    • C07C251/34Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/36Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atoms of the oxyimino groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C251/40Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atoms of the oxyimino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/01Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/42Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/20Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by nitrogen atoms not being part of nitro or nitroso groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT94929340T 1993-10-22 1994-09-26 Zwischenprodukte für die herstellung einer substituierten 2,5-diamino-3-hydroxyhexan. ATE183993T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14179593A 1993-10-22 1993-10-22
US08/281,502 US5491253A (en) 1993-10-22 1994-07-27 Process for the preparation of a substituted 2,5-diamino-3-hydroxyhexane

Publications (1)

Publication Number Publication Date
ATE183993T1 true ATE183993T1 (de) 1999-09-15

Family

ID=26839452

Family Applications (2)

Application Number Title Priority Date Filing Date
AT94929340T ATE183993T1 (de) 1993-10-22 1994-09-26 Zwischenprodukte für die herstellung einer substituierten 2,5-diamino-3-hydroxyhexan.
AT99101692T ATE238983T1 (de) 1993-10-22 1994-09-26 Herstellung einer substituierten 2,5-diamino-3- hydroxyhexan

Family Applications After (1)

Application Number Title Priority Date Filing Date
AT99101692T ATE238983T1 (de) 1993-10-22 1994-09-26 Herstellung einer substituierten 2,5-diamino-3- hydroxyhexan

Country Status (11)

Country Link
US (11) US5491253A (de)
EP (2) EP0724563B1 (de)
JP (2) JP3822233B2 (de)
AT (2) ATE183993T1 (de)
CA (1) CA2174000C (de)
DE (2) DE69420421T2 (de)
DK (2) DK0916646T3 (de)
ES (2) ES2138667T3 (de)
GR (1) GR3031939T3 (de)
PT (1) PT916646E (de)
WO (1) WO1995011224A1 (de)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995023793A1 (en) * 1994-03-02 1995-09-08 Daicel Chemical Industries, Ltd. 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same
JP3338227B2 (ja) * 1995-02-28 2002-10-28 高砂香料工業株式会社 ケトニトリル誘導体及びヘキセノン誘導体の製造方法
US6037157A (en) 1995-06-29 2000-03-14 Abbott Laboratories Method for improving pharmacokinetics
US5932766A (en) * 1997-05-30 1999-08-03 Abbott Laboratories Process for the preparation of substituted keto-enamines
MY121765A (en) 1998-07-20 2006-02-28 Abbott Lab Polymorph of ritonavir
US6307090B1 (en) 1999-01-22 2001-10-23 The United States Of America As Represented By The Department Of Health And Human Services Acylated oligopeptide derivatives having cell signal inhibiting activity
ATE509026T1 (de) * 1999-03-23 2011-05-15 Us Gov Health & Human Serv Phenylalanin- derivate
US7226991B1 (en) * 1999-03-23 2007-06-05 United States Of America, Represented By The Secretary, Department Of Health And Human Services Phenylalanine derivatives
US6765019B1 (en) 1999-05-06 2004-07-20 University Of Kentucky Research Foundation Permeable, water soluble, non-irritating prodrugs of chemotherapeutic agents with oxaalkanoic acids
US6573409B1 (en) * 1999-07-02 2003-06-03 The Nutrasweet Company Process for the preparation of 3,3-dimethylbutanal
CN102584799A (zh) * 1999-09-16 2012-07-18 田边三菱制药株式会社 含氮的6-员芳香环化合物
IT1313624B1 (it) 1999-09-21 2002-09-09 Archimica Spa Ora Clariant Lif Procedimento per la sintesi del ritonavir
ES2287048T3 (es) 1999-10-22 2007-12-16 The Government Of The Usa, As Represented By The Secretary, Department Of Health And Human Services Inhbicion de la motilidad celular y la angiognesis mediante nhibidores del dominio gbr2sh2.
US7871981B2 (en) * 1999-10-22 2011-01-18 The United States Of America As Represented By The Department Of Health And Human Services Inhibition of cell motility, angiogenesis, and metastasis
SI1248600T1 (sl) 2000-01-19 2008-08-31 Abbott Lab Izboljšane farmacevtske formulacije inhibitorjev proteaze HIV
US7425537B2 (en) * 2000-08-22 2008-09-16 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services SH2 domain binding inhibitors
AU2001285133A1 (en) * 2000-08-22 2002-03-04 The Government Of The United States Of America, Represented By The Secretary, Department Of Health And Human Services SH2 domain binding inhibitors
US7060165B2 (en) * 2002-02-14 2006-06-13 Pcbu Services, Inc. Processes for purification and production of fluorocarbons
ATE384038T1 (de) * 2002-10-18 2008-02-15 Tohru Yokozawa Verfahren zur herstellung optisch aktiver aminoalkohole
US20040138104A1 (en) * 2003-01-14 2004-07-15 The Government Of The United States Of America Represented By The Secretary, Peptides
US6933504B2 (en) * 2003-03-12 2005-08-23 General Electric Company CT detector having a segmented optical coupler and method of manufacturing same
US20050119163A1 (en) * 2003-09-18 2005-06-02 The Government Of The United States Of America, As Represented By The Secretary, SH2 domain binding inhibitors
WO2006090264A1 (en) * 2005-02-28 2006-08-31 Ranbaxy Laboratories Limited A process for the synthesis of 2-amino-5-protected amino-3-hydroxy-1, 6-diphenylhexane or a salt thereof - an intermediate for antiviral drugs
CA2620469C (en) 2005-09-02 2014-04-01 Amgen Inc. Methods of modulating intestinal fluid balance
US20080160204A1 (en) * 2006-12-28 2008-07-03 Lavoie Adrien R Spontaneous copper seed deposition process for metal interconnects
WO2008149228A1 (en) * 2007-06-08 2008-12-11 Aurobindo Pharma Limited An improved process for the preparation of substantially pure (2s,3s,5s)-5-amino-2-n,n-dibenzylamino-3-hydroxy-1,6-diphenylhexane
JP5204438B2 (ja) * 2007-07-31 2013-06-05 東ソ−・エフテック株式会社 含フッ素アミン化合物の製造方法
CN101967130B (zh) * 2010-07-02 2012-12-26 厦门市亨瑞生化有限公司 利托那韦中间体的合成方法
CN107602454B (zh) * 2017-09-19 2020-12-01 佛山科学技术学院 磺酰胺类化合物及其制备方法和用途
US10529439B2 (en) 2017-10-24 2020-01-07 Spin Memory, Inc. On-the-fly bit failure detection and bit redundancy remapping techniques to correct for fixed bit defects
US10438995B2 (en) 2018-01-08 2019-10-08 Spin Memory, Inc. Devices including magnetic tunnel junctions integrated with selectors

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2784228A (en) * 1953-08-26 1957-03-05 North Carolina Pharmacentical Alkaline hydrogenation of oximinoketones
GB1383186A (en) * 1972-07-26 1975-02-05 Luso Farmaco Inst Beta-aminoketone derivatives
US5142056A (en) * 1989-05-23 1992-08-25 Abbott Laboratories Retroviral protease inhibiting compounds
US5177259A (en) * 1986-04-11 1993-01-05 Warner-Lambert Company Diarylalkanoids having activity as lipoxygenase inhibitors
WO1988002374A2 (en) * 1986-09-30 1988-04-07 The Upjohn Company Renin inhibitory peptides having novel c-terminal moieties
NO169837C (no) * 1987-12-21 1992-08-12 Astra Ab Analogifremgangsmaate for fremstilling av nye terapeutisk aktive forbindelser
DE3829594A1 (de) * 1988-09-01 1990-03-15 Bayer Ag Neue renininhibitoren, verfahren zur herstellung und ihre verwendung in arzneimitteln
US5354866A (en) * 1989-05-23 1994-10-11 Abbott Laboratories Retroviral protease inhibiting compounds
IE913840A1 (en) * 1990-11-20 1992-05-20 Abbott Lab Retroviral protease inhibiting compounds
JPH06184069A (ja) * 1991-11-19 1994-07-05 Lonza Ag α−ヒドロキシ−β−アミノカルボン酸の製造方法
KR100187613B1 (ko) * 1992-12-29 1999-06-01 스티븐 에프. 웨인스톡 레트로바이러스성 프로테이제 억제 화합물, 이의 제조방법 및 이를 함유하는 약제학적 조성물
IL110752A (en) * 1993-09-13 2000-07-26 Abbott Lab Liquid semi-solid or solid pharmaceutical composition for an HIV protease inhibitor

Also Published As

Publication number Publication date
JP2006206597A (ja) 2006-08-10
EP0916646A3 (de) 1999-08-18
US5616776A (en) 1997-04-01
DK0916646T3 (da) 2003-08-25
DK0724563T3 (da) 2000-03-20
EP0724563A1 (de) 1996-08-07
EP0916646A2 (de) 1999-05-19
US5625092A (en) 1997-04-29
JPH09504024A (ja) 1997-04-22
EP0916646B1 (de) 2003-05-02
US5491253A (en) 1996-02-13
CA2174000A1 (en) 1995-04-27
US5543552A (en) 1996-08-06
DE69420421D1 (de) 1999-10-07
US5543549A (en) 1996-08-06
US5654466A (en) 1997-08-05
EP0724563B1 (de) 1999-09-01
JP4172717B2 (ja) 2008-10-29
ES2138667T3 (es) 2000-01-16
DE69420421T2 (de) 2000-05-04
PT916646E (pt) 2003-09-30
US5569777A (en) 1996-10-29
JP3822233B2 (ja) 2006-09-13
DE69432611T2 (de) 2004-03-18
US5565604A (en) 1996-10-15
US5541328A (en) 1996-07-30
WO1995011224A1 (en) 1995-04-27
DE69432611D1 (de) 2003-06-05
ATE238983T1 (de) 2003-05-15
HK1011677A1 (en) 1999-07-16
CA2174000C (en) 2005-05-24
US5543551A (en) 1996-08-06
US5508409A (en) 1996-04-16
ES2198094T3 (es) 2004-01-16
GR3031939T3 (en) 2000-03-31

Similar Documents

Publication Publication Date Title
ATE183993T1 (de) Zwischenprodukte für die herstellung einer substituierten 2,5-diamino-3-hydroxyhexan.
ATE210635T1 (de) Aromatische hydroxamsäure-verbindungen, ihre herstellung und verwendung
DE68929330D1 (de) Zwischenprodukte für die Herstellung von Derivaten der 4-Oxochinolin-3-carbonsäure
ES2070660A1 (es) Un procedimiento para la preparacion de 2,5-damino-3-hidroxihexanos sustituidos, utiles como inhibidores de proteasas retrovirales.
DE69532634D1 (de) Zwischenprodukte für die herstellung von pharmazeutischem camptothecin
DE69915004D1 (de) 5-Oxo-pyrrolidine-2-Carbonsäure-Hydroxamidderivate
IL72100A (en) 6-fluoro-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid derivatives,their preparation and pharmaceutical compositions comprising them
CA2109482A1 (en) Process for producing alanylglutamine
CA2011087A1 (en) Use of trifluoromethylphenylazolylmethyloxiranes as crop protection agents
DK519985A (da) Quinoloncarboxylsyrederivater, fremgangsmaade til fremstilling deraf og antibakterielt middel indeholdende saadanne derivater
NO902555D0 (no) N-heteroaryl-purin-6-aminer og fremgangsmaate for fremstilling derav.
NO894349D0 (no) Tienopyridin-type mevalonolaktoner.
DE69121259D1 (de) Beta-Lactam-Verbindungen und ihre Herstellung
AU3551884A (en) Quinazoline and isoquinoline derivatives
HUT53886A (en) Fungicide preparations containing propencarboxylic acid derivatives as agents and process for producing the agents
NO910904D0 (no) Fremgangsmaate for fremstilling av en substituert aminforbindelse.
ATE73768T1 (de) 2,5,6,7-tetranor-18,18,19,19-tetradehydro-4,8inter-m-phenylene-pgi2-derivate.
ATE245147T1 (de) Substituierte aminochinazolinon (thion) derivate
CA2231633A1 (en) Process for the preparation of anti-malarial drugs
ATE226585T1 (de) Thiazolobenzoheterocyclen, ihre herstellung und diese enthaltende phatrmazeutische zubereitungen
AU1586588A (en) Fungicidal derivatives of propenoic acid and processes for their preparation
ATE192141T1 (de) Aromatische hydroxamsäure-verbindungen, ihre herstellung und verwendung
DE69511449D1 (de) Octahydro-2-Naphthalincarbonsäure-Derivate, ihre Herstellung und Verwendung
DE69008130D1 (de) Glutarsäurederivate und ihre Herstellung.
MX9700720A (es) Procedimiento para la preparacion de un 2,5-diamino-3-hidroxihexano.

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee