ATE127126T1 - Verfahren zur herstellung von 1-alpha,3-beta,24- trihydroxy-delta-5-steroidderivaten. - Google Patents
Verfahren zur herstellung von 1-alpha,3-beta,24- trihydroxy-delta-5-steroidderivaten.Info
- Publication number
- ATE127126T1 ATE127126T1 AT89111561T AT89111561T ATE127126T1 AT E127126 T1 ATE127126 T1 AT E127126T1 AT 89111561 T AT89111561 T AT 89111561T AT 89111561 T AT89111561 T AT 89111561T AT E127126 T1 ATE127126 T1 AT E127126T1
- Authority
- AT
- Austria
- Prior art keywords
- alpha
- delta
- formula
- trihydroxy
- beta
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 150000003431 steroids Chemical class 0.000 title 1
- QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 abstract 2
- 229910052784 alkaline earth metal Inorganic materials 0.000 abstract 2
- 150000001342 alkaline earth metals Chemical class 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 229910052751 metal Inorganic materials 0.000 abstract 2
- 239000002184 metal Substances 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 229910021529 ammonia Inorganic materials 0.000 abstract 1
- 239000013067 intermediate product Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP63165148A JPH0749435B2 (ja) | 1988-07-04 | 1988-07-04 | １α，３β，２４−トリヒドロキシ−△▲上５▼−ステロイド類の製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE127126T1 true ATE127126T1 (de) | 1995-09-15 |
Family
ID=15806795
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT89111561T ATE127126T1 (de) | 1988-07-04 | 1989-06-24 | Verfahren zur herstellung von 1-alpha,3-beta,24- trihydroxy-delta-5-steroidderivaten. |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US5117015A (de) |
| EP (1) | EP0349869B1 (de) |
| JP (1) | JPH0749435B2 (de) |
| AT (1) | ATE127126T1 (de) |
| DE (1) | DE68924010T2 (de) |
| DK (1) | DK174183B1 (de) |
| ES (1) | ES2076175T3 (de) |
| PT (1) | PT91011B (de) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0946584B1 (de) | 1996-12-20 | 2003-04-23 | Novo Nordisk A/S | Verbindungen zur Regulierung der Meiose |
| JP2007517878A (ja) * | 2004-01-15 | 2007-07-05 | ワーナー・チルコット・カンパニー・インコーポレーテッド | エチニルエストラジオールのジ−ステロイド型プロドラッグ |
| JP2007517877A (ja) * | 2004-01-15 | 2007-07-05 | ワーナー・チルコット・カンパニー・インコーポレーテッド | エストラジオールのジ−ステロイド型プロドラッグ |
| ES2523045T3 (es) * | 2005-07-12 | 2014-11-20 | Warner Chilcott Company, Llc | Derivado éster de etinil estradiol |
| CN101228177A (zh) * | 2005-07-12 | 2008-07-23 | 沃纳奇尔科特公司 | 雌二醇的3-酯前药 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1081424A (fr) * | 1953-05-26 | 1954-12-20 | Ile De Rech S Tech Soc Civ | Procédé de préparation de dérivés du cholestane et des cholestènes di-oxygénés en position 3 et 24 |
| US3901928A (en) * | 1973-01-10 | 1975-08-26 | Robert Henry Hesse | 1' ,3' -dihydroxy steroid-5-enes method of preparing same and their use for preparing 1' -hydroxy-25-hydrogen vitamin d compounds |
| US4670190A (en) * | 1973-01-10 | 1987-06-02 | Hesse Robert H | 1-α-hydroxy vitamin D compounds and process for preparing same |
| DE2400189A1 (de) * | 1974-01-03 | 1975-07-17 | Basf Ag | Verfahren zur herstellung von 1 alphahydroxy-cholesterinen |
| US3907843A (en) * | 1974-06-14 | 1975-09-23 | Wisconsin Alumni Res Found | 1{60 -Hydroxyergocalciferol and processes for preparing same |
| US4022891A (en) * | 1974-06-18 | 1977-05-10 | Teijin Limited | Novel 1α,24-dihydroxycholecalciferol compositions, novel precursors thereof, and processes for preparing them |
| IL45897A (en) * | 1974-10-22 | 1978-12-17 | Yeda Res & Dev | Process for the preparation of 1 hydroxy-provitamin d3 |
| LU80545A1 (de) * | 1978-11-17 | 1980-06-05 | Hoffmann La Roche | Verfahren zur herstellung von 1a,3s-dihydroxy->5-steroiden |
| JPS5854160A (ja) * | 1981-09-28 | 1983-03-31 | 旭化成株式会社 | 床下収納庫 |
| JPH0681758B2 (ja) * | 1988-04-28 | 1994-10-19 | 帝人株式会社 | １α，３β−ジヒドロキシ−△▲上５▼−ステロイドの製造方法 |
-
1988
- 1988-07-04 JP JP63165148A patent/JPH0749435B2/ja not_active Expired - Lifetime
-
1989
- 1989-06-24 AT AT89111561T patent/ATE127126T1/de not_active IP Right Cessation
- 1989-06-24 ES ES89111561T patent/ES2076175T3/es not_active Expired - Lifetime
- 1989-06-24 EP EP89111561A patent/EP0349869B1/de not_active Expired - Lifetime
- 1989-06-24 DE DE68924010T patent/DE68924010T2/de not_active Expired - Lifetime
- 1989-06-26 DK DK198903166A patent/DK174183B1/da not_active IP Right Cessation
- 1989-06-29 PT PT91011A patent/PT91011B/pt not_active IP Right Cessation
-
1991
- 1991-04-30 US US07/696,255 patent/US5117015A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP0349869A2 (de) | 1990-01-10 |
| PT91011A (pt) | 1990-02-08 |
| ES2076175T3 (es) | 1995-11-01 |
| DK316689D0 (da) | 1989-06-26 |
| EP0349869B1 (de) | 1995-08-30 |
| JPH0215093A (ja) | 1990-01-18 |
| US5117015A (en) | 1992-05-26 |
| DK316689A (da) | 1990-01-05 |
| JPH0749435B2 (ja) | 1995-05-31 |
| DE68924010T2 (de) | 1996-01-25 |
| DK174183B1 (da) | 2002-08-19 |
| EP0349869A3 (en) | 1990-04-25 |
| PT91011B (pt) | 1995-01-31 |
| DE68924010D1 (de) | 1995-10-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| EELA | Cancelled due to lapse of time |