NO168767C - Cyklopenta(d)pyrimidinderivater og fremgangsmaate til fremstilling derav - Google Patents
Cyklopenta(d)pyrimidinderivater og fremgangsmaate til fremstilling deravInfo
- Publication number
- NO168767C NO168767C NO860852A NO860852A NO168767C NO 168767 C NO168767 C NO 168767C NO 860852 A NO860852 A NO 860852A NO 860852 A NO860852 A NO 860852A NO 168767 C NO168767 C NO 168767C
- Authority
- NO
- Norway
- Prior art keywords
- sup
- cyclopenta
- procedures
- preparing
- pyrimidine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Dental Preparations (AREA)
- Saccharide Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Luminescent Compositions (AREA)
- Soil Working Implements (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Eyeglasses (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP4362685 | 1985-03-07 |
Publications (3)
Publication Number | Publication Date |
---|---|
NO860852L NO860852L (no) | 1986-09-08 |
NO168767B NO168767B (no) | 1991-12-23 |
NO168767C true NO168767C (no) | 1992-04-01 |
Family
ID=12669058
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO860852A NO168767C (no) | 1985-03-07 | 1986-03-07 | Cyklopenta(d)pyrimidinderivater og fremgangsmaate til fremstilling derav |
Country Status (15)
Country | Link |
---|---|
US (1) | US4749704A (no) |
EP (1) | EP0194161B1 (no) |
JP (1) | JPS6270A (no) |
KR (1) | KR890003839B1 (no) |
AT (1) | ATE106077T1 (no) |
AU (1) | AU580391B2 (no) |
CA (1) | CA1273632A (no) |
DE (1) | DE3689848T2 (no) |
DK (1) | DK165109C (no) |
ES (3) | ES8704905A1 (no) |
FI (1) | FI88717C (no) |
HK (1) | HK1005450A1 (no) |
IE (1) | IE64504B1 (no) |
NO (1) | NO168767C (no) |
ZA (1) | ZA861708B (no) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5037980A (en) * | 1988-04-18 | 1991-08-06 | American Cyanamid Company | Phenyl imidazo[1,2-a]pyrimidines |
US5877178A (en) * | 1991-04-08 | 1999-03-02 | Duquesne University Of The Holy Ghost | Pyrimidine derivatives and methods of making and using these derivatives |
US5234936A (en) * | 1991-10-24 | 1993-08-10 | American Home Products Corporation | Pyrimidocycloalkanes as a ii antagonists |
ATE374190T1 (de) * | 2003-08-12 | 2007-10-15 | Hoffmann La Roche | Tetrahydrochinazolinderivate als cfr-antagonisten |
JPWO2007049342A1 (ja) | 2005-10-26 | 2009-04-30 | 三菱電機株式会社 | エレベーター群管理制御装置 |
CN103288753A (zh) | 2006-07-06 | 2013-09-11 | 阵列生物制药公司 | 作为akt蛋白激酶抑制剂的环戊二烯并[d]嘧啶 |
CA2656566C (en) | 2006-07-06 | 2014-06-17 | Array Biopharma Inc. | Dihydrofuro pyrimidines as akt protein kinase inhibitors |
SI2054418T1 (sl) | 2006-07-06 | 2012-02-29 | Array Biopharma Inc | Dihidrotieno pirimidini kot AKT protein kinazni inhibitorji |
US8063050B2 (en) | 2006-07-06 | 2011-11-22 | Array Biopharma Inc. | Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors |
WO2008021456A2 (en) * | 2006-08-16 | 2008-02-21 | Cytovia, Inc. | N-aryl-5,7-dihydrofuro[3,4-d]pyrimidin-4-amines and analogs as activators of caspases and inducers of apoptosis and the use thereof |
US8846683B2 (en) | 2007-07-05 | 2014-09-30 | Array Biopharma, Inc. | Pyrimidyl cyclopentanes as Akt protein kinase inhibitors |
TWI450720B (zh) | 2007-07-05 | 2014-09-01 | Array Biopharma Inc | 作為akt蛋白質激酶抑制劑之嘧啶環戊烷 |
KR20150091196A (ko) | 2007-07-05 | 2015-08-07 | 어레이 바이오파마 인크. | Akt 단백질 키나제 억제제로서의 피리미딜 시클로펜탄 |
US9409886B2 (en) | 2007-07-05 | 2016-08-09 | Array Biopharma Inc. | Pyrimidyl cyclopentanes as AKT protein kinase inhibitors |
ES2422733T3 (es) | 2008-01-09 | 2013-09-13 | Array Biopharma Inc | Pirimidilciclopentanos hidroxilados como inhibidores de proteínas cinasas AKT |
EP2240455B1 (en) | 2008-01-09 | 2012-12-26 | Array Biopharma, Inc. | Hydroxylated pyrimidyl cyclopentane as akt protein kinase inhibitor |
DE112009002588B4 (de) | 2008-10-20 | 2019-08-14 | Mitsubishi Electric Corporation | Aufzuggruppenverwaltungssystem |
CA2831932A1 (en) | 2011-04-01 | 2012-10-04 | Genentech, Inc. | Combinations of akt and mek inhibitor compounds, and methods of use |
AU2012236166A1 (en) | 2011-04-01 | 2013-11-14 | Genentech, Inc. | Combinations of AKT inhibitor compounds and chemotherapeutic agents, and methods of use |
GB201121127D0 (en) | 2011-12-08 | 2012-01-18 | Dow Corning | Treatment of filler with silane |
CN111303053B (zh) * | 2020-03-16 | 2023-01-17 | 中国海洋大学 | 环戊并[d]嘧啶类化合物及其药学上可接受的盐、溶剂合物或者前药以及应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3470182A (en) * | 1967-02-09 | 1969-09-30 | Sandoz Ag | 4-amino-substituted quinazolines |
US3980650A (en) * | 1972-05-05 | 1976-09-14 | N.V. Koninklijke Pharmaceutische Fabrieken V/H Brocades-Stheeman En Pharmacia | 4-Amino-pyrimidine derivatives |
US3915976A (en) * | 1972-09-01 | 1975-10-28 | Sandoz Ag | Substituted-4-phenyl-5h-cycloalkano(d)pyrimidines |
PH20344A (en) * | 1981-01-29 | 1986-12-04 | Sankyo Co | Aminopyrimidine derivatives, processes for their preparation, and fungicidal, insecticidal and acaricidal compositions containing them |
JPS57203072A (en) * | 1981-06-05 | 1982-12-13 | Sankyo Co Ltd | 4-anilinopyrimidine derivative, its preparation, antidepressant comprising it as active ingredient |
-
1986
- 1986-03-06 US US06/837,079 patent/US4749704A/en not_active Expired - Lifetime
- 1986-03-06 JP JP61049238A patent/JPS6270A/ja not_active Withdrawn
- 1986-03-07 IE IE59786A patent/IE64504B1/en not_active IP Right Cessation
- 1986-03-07 ES ES552796A patent/ES8704905A1/es not_active Expired
- 1986-03-07 AU AU54481/86A patent/AU580391B2/en not_active Ceased
- 1986-03-07 CA CA000503571A patent/CA1273632A/en not_active Expired - Lifetime
- 1986-03-07 EP EP86301660A patent/EP0194161B1/en not_active Expired - Lifetime
- 1986-03-07 ZA ZA861708A patent/ZA861708B/xx unknown
- 1986-03-07 FI FI860969A patent/FI88717C/fi not_active IP Right Cessation
- 1986-03-07 KR KR1019860001624A patent/KR890003839B1/ko not_active IP Right Cessation
- 1986-03-07 DE DE3689848T patent/DE3689848T2/de not_active Expired - Fee Related
- 1986-03-07 DK DK106586A patent/DK165109C/da not_active IP Right Cessation
- 1986-03-07 AT AT86301660T patent/ATE106077T1/de not_active IP Right Cessation
- 1986-03-07 NO NO860852A patent/NO168767C/no unknown
- 1986-11-14 ES ES557199A patent/ES8801222A1/es not_active Expired
- 1986-11-14 ES ES557198A patent/ES8801221A1/es not_active Expired
-
1998
- 1998-05-27 HK HK98104569A patent/HK1005450A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
HK1005450A1 (en) | 1999-01-08 |
FI860969A0 (fi) | 1986-03-07 |
NO168767B (no) | 1991-12-23 |
ATE106077T1 (de) | 1994-06-15 |
EP0194161B1 (en) | 1994-05-25 |
KR890003839B1 (ko) | 1989-10-05 |
IE860597L (en) | 1986-09-07 |
DK165109C (da) | 1993-03-01 |
ES557198A0 (es) | 1988-01-01 |
KR860007221A (ko) | 1986-10-08 |
AU580391B2 (en) | 1989-01-12 |
NO860852L (no) | 1986-09-08 |
CA1273632A (en) | 1990-09-04 |
US4749704A (en) | 1988-06-07 |
ZA861708B (en) | 1986-11-26 |
EP0194161A3 (en) | 1987-09-02 |
DK165109B (da) | 1992-10-12 |
JPS6270A (ja) | 1987-01-06 |
ES557199A0 (es) | 1988-01-01 |
FI88717C (fi) | 1993-06-28 |
DK106586D0 (da) | 1986-03-07 |
DK106586A (da) | 1986-09-08 |
FI88717B (fi) | 1993-03-15 |
ES552796A0 (es) | 1987-04-16 |
DE3689848D1 (de) | 1994-06-30 |
ES8801221A1 (es) | 1988-01-01 |
AU5448186A (en) | 1986-09-11 |
EP0194161A2 (en) | 1986-09-10 |
IE64504B1 (en) | 1995-08-09 |
ES8801222A1 (es) | 1988-01-01 |
FI860969A (fi) | 1986-09-08 |
DE3689848T2 (de) | 1995-01-12 |
ES8704905A1 (es) | 1987-04-16 |
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