ATA290487A - Pharmazeutika enthaltend pyrozole - Google Patents

Pharmazeutika enthaltend pyrozole

Info

Publication number
ATA290487A
ATA290487A AT872904A AT290487A ATA290487A AT A290487 A ATA290487 A AT A290487A AT 872904 A AT872904 A AT 872904A AT 290487 A AT290487 A AT 290487A AT A290487 A ATA290487 A AT A290487A
Authority
AT
Austria
Prior art keywords
pyrozoles
pharmaceuticals containing
pharmaceuticals
containing pyrozoles
Prior art date
Application number
AT872904A
Other languages
English (en)
Other versions
AT390732B (de
Inventor
Richard Anthony Appleton
John Dixon
Sidney Clifford Burford
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB868611102A external-priority patent/GB8611102D0/en
Priority claimed from GB868630906A external-priority patent/GB8630906D0/en
Application filed by Fisons Plc filed Critical Fisons Plc
Publication of ATA290487A publication Critical patent/ATA290487A/de
Application granted granted Critical
Publication of AT390732B publication Critical patent/AT390732B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT0290487A 1986-05-07 1987-11-03 Pharmazeutika enthaltend pyrazole AT390732B (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB868611102A GB8611102D0 (en) 1986-05-07 1986-05-07 Heterocyclic compounds
GB868630906A GB8630906D0 (en) 1986-12-24 1986-12-24 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
ATA290487A true ATA290487A (de) 1989-12-15
AT390732B AT390732B (de) 1990-06-25

Family

ID=26290729

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0290487A AT390732B (de) 1986-05-07 1987-11-03 Pharmazeutika enthaltend pyrazole

Country Status (13)

Country Link
US (1) US4803216A (de)
EP (1) EP0248523B1 (de)
KR (1) KR870011101A (de)
AT (1) AT390732B (de)
AU (1) AU595602B2 (de)
CA (1) CA1305157C (de)
DE (1) DE3773746D1 (de)
DK (1) DK231687A (de)
FI (1) FI871974L (de)
IL (1) IL82421A0 (de)
NO (1) NO871879L (de)
NZ (1) NZ220214A (de)
PT (1) PT84831B (de)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR900100380A (el) * 1989-05-20 1991-10-10 Fisons Plc Μέ?οδος παρασκευής αντι-φλεγμονωδών παραγώγων αμινοφενόλης.
DE4234886A1 (de) * 1992-10-16 1994-04-21 Wella Ag Neue N-Phenylaminopyrazol-Derivate sowie Mittel und Verfahren zur Färbung von Haaren
GB9312853D0 (en) * 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5500439A (en) * 1993-12-09 1996-03-19 Alteon Inc. Aminopyrazoles
DE69526790T2 (de) * 1994-06-24 2003-03-06 Euroceltique S.A., Luxemburg/Luxembourg Verbindungen zur hemmung von phosphodiesrerase iv
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US5591776A (en) * 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
DE69531506T2 (de) * 1994-12-13 2004-06-24 Euroceltique S.A. Arylthioxanthine
JP2001523213A (ja) * 1994-12-13 2001-11-20 ユーロ−セルティーク,エス.エイ. 三置換チオキサンチン類
US6025361A (en) * 1994-12-13 2000-02-15 Euro-Celtique, S.A. Trisubstituted thioxanthines
US6166041A (en) * 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) * 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
US5864037A (en) * 1996-06-06 1999-01-26 Euro-Celtique, S.A. Methods for the synthesis of chemical compounds having PDE-IV inhibitory activity
US5744473A (en) * 1996-09-16 1998-04-28 Euro-Celtique, S.A. PDE IV inhibitors: "bis-compounds"
EP2147679B1 (de) 2001-07-25 2014-06-25 Raptor Pharmaceutical, Inc. Zusammensetzungen für den Blut-Hirn-Schrankentransport
DE602004016964D1 (de) * 2003-02-27 2008-11-20 Smithkline Beecham Corp Neue verbindungen
GB0326601D0 (en) * 2003-11-14 2003-12-17 Novartis Ag Organic compounds
EP2392258B1 (de) 2005-04-28 2014-10-08 Proteus Digital Health, Inc. Pharma-Informatiksystem
JO3019B1 (ar) 2006-04-19 2016-09-05 Janssen Pharmaceutica Nv ثلاثي مستبدل 4،2،1-ثلاثي زولات
CN101594878A (zh) 2006-09-18 2009-12-02 雷普特药品公司 通过给予受体相关蛋白(rap)-缀合物对肝病症的治疗
JO2784B1 (en) 2007-10-18 2014-03-15 شركة جانسين فارماسوتيكا ان. في 5,3,1 - Triazole substitute derivative
ES2424023T3 (es) 2007-10-18 2013-09-26 Janssen Pharmaceutica N.V. 1,2,4-triazoles trisustituidos
CA2714662C (en) 2008-03-19 2016-05-10 Janssen Pharmaceutica Nv Trisubstituted 1,2,4-triazoles as nicotinic acetylcholine receptor modulators
CL2009001125A1 (es) 2008-05-09 2011-02-11 Janssen Pharmaceutica Nv Compuestos derivados de pirazol trisustituido, moduladores alostericos positivos de los receptores ach nicotinicos; composicion farmaceutica que los comprende; proceso de preparacion de la composicion; y su uso en el tratamiento de enfermedades de snc o inflamatorias.
PL3395372T3 (pl) 2009-02-20 2022-07-25 EnhanX Biopharm Inc. Układ do dostarczania leków na bazie glutationu
CN102458374A (zh) 2009-05-06 2012-05-16 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其使用方法
EA020564B1 (ru) 2009-09-17 2014-12-30 Янссен Фармацевтика Нв Замещенные n-фенил-1-(4-пиридинил)-1н-пиразол-3-амины
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
AU2015281799B2 (en) * 2014-06-26 2019-11-28 Central Adelaide Local Health Network Incorporated Enzyme interacting agents
KR102725207B1 (ko) * 2018-02-07 2024-11-01 한국화학연구원 Tnik 저해용 화합물 및 이들의 의약 용도

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD211343A1 (de) * 1982-11-08 1984-07-11 Univ Ernst Moritz Arndt Verfahren zur synthese von pyrazolen
EP0178035B1 (de) * 1984-05-12 1990-01-03 FISONS plc Antiinflammatorische 1,N-Diarylpyrazol-3-amine, deren Zusammensetzungen und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
NO871879D0 (no) 1987-05-06
DK231687D0 (da) 1987-05-06
FI871974A7 (fi) 1987-11-08
FI871974A0 (fi) 1987-05-05
NO871879L (no) 1987-11-09
CA1305157C (en) 1992-07-14
DE3773746D1 (en) 1991-11-21
AU7258487A (en) 1987-11-12
AT390732B (de) 1990-06-25
NZ220214A (en) 1990-06-26
AU595602B2 (en) 1990-04-05
EP0248523A1 (de) 1987-12-09
EP0248523B1 (de) 1991-10-16
IL82421A0 (en) 1987-11-30
PT84831A (en) 1987-06-01
DK231687A (da) 1987-11-08
FI871974L (fi) 1987-11-08
PT84831B (pt) 1990-02-08
KR870011101A (ko) 1987-12-21
US4803216A (en) 1989-02-07

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Legal Events

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