DK231687A - Heterocykliske forbindelser, deres fremstilling og anvendelse, samt laegemidler indeholdende disse forbindelser - Google Patents

Heterocykliske forbindelser, deres fremstilling og anvendelse, samt laegemidler indeholdende disse forbindelser

Info

Publication number
DK231687A
DK231687A DK231687A DK231687A DK231687A DK 231687 A DK231687 A DK 231687A DK 231687 A DK231687 A DK 231687A DK 231687 A DK231687 A DK 231687A DK 231687 A DK231687 A DK 231687A
Authority
DK
Denmark
Prior art keywords
compounds
preparation
pharmaceuticals containing
heterocyclic
heterocyclic compounds
Prior art date
Application number
DK231687A
Other languages
English (en)
Other versions
DK231687D0 (da
Inventor
Richard Anthony Appleton
Sidney Clifford Burford
John Dixon
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB868611102A external-priority patent/GB8611102D0/en
Priority claimed from GB868630906A external-priority patent/GB8630906D0/en
Application filed by Fisons Plc filed Critical Fisons Plc
Publication of DK231687D0 publication Critical patent/DK231687D0/da
Publication of DK231687A publication Critical patent/DK231687A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK231687A 1986-05-07 1987-05-06 Heterocykliske forbindelser, deres fremstilling og anvendelse, samt laegemidler indeholdende disse forbindelser DK231687A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB868611102A GB8611102D0 (en) 1986-05-07 1986-05-07 Heterocyclic compounds
GB868630906A GB8630906D0 (en) 1986-12-24 1986-12-24 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
DK231687D0 DK231687D0 (da) 1987-05-06
DK231687A true DK231687A (da) 1987-11-08

Family

ID=26290729

Family Applications (1)

Application Number Title Priority Date Filing Date
DK231687A DK231687A (da) 1986-05-07 1987-05-06 Heterocykliske forbindelser, deres fremstilling og anvendelse, samt laegemidler indeholdende disse forbindelser

Country Status (13)

Country Link
US (1) US4803216A (da)
EP (1) EP0248523B1 (da)
KR (1) KR870011101A (da)
AT (1) AT390732B (da)
AU (1) AU595602B2 (da)
CA (1) CA1305157C (da)
DE (1) DE3773746D1 (da)
DK (1) DK231687A (da)
FI (1) FI871974L (da)
IL (1) IL82421A0 (da)
NO (1) NO871879L (da)
NZ (1) NZ220214A (da)
PT (1) PT84831B (da)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR900100380A (el) * 1989-05-20 1991-10-10 Fisons Plc Μέ?οδος παρασκευής αντι-φλεγμονωδών παραγώγων αμινοφενόλης.
DE4234886A1 (de) * 1992-10-16 1994-04-21 Wella Ag Neue N-Phenylaminopyrazol-Derivate sowie Mittel und Verfahren zur Färbung von Haaren
GB9312853D0 (en) * 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5500439A (en) * 1993-12-09 1996-03-19 Alteon Inc. Aminopyrazoles
DE69526790T2 (de) * 1994-06-24 2003-03-06 Euroceltique S.A., Luxemburg/Luxembourg Verbindungen zur hemmung von phosphodiesrerase iv
US5591776A (en) * 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
JPH10508032A (ja) * 1994-12-13 1998-08-04 ユーロ−セルティーク,エス.エイ. アリールチオキサンチン類
ATE247655T1 (de) * 1994-12-13 2003-09-15 Euro Celtique Sa Dreifachsubstituierte thioxanthine
US6025361A (en) * 1994-12-13 2000-02-15 Euro-Celtique, S.A. Trisubstituted thioxanthines
US6166041A (en) * 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) * 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
US5864037A (en) 1996-06-06 1999-01-26 Euro-Celtique, S.A. Methods for the synthesis of chemical compounds having PDE-IV inhibitory activity
US5744473A (en) * 1996-09-16 1998-04-28 Euro-Celtique, S.A. PDE IV inhibitors: "bis-compounds"
EP1554572B1 (en) 2001-07-25 2009-10-14 Raptor Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
DE602004016964D1 (de) * 2003-02-27 2008-11-20 Smithkline Beecham Corp Neue verbindungen
GB0326601D0 (en) * 2003-11-14 2003-12-17 Novartis Ag Organic compounds
EP3827747A1 (en) 2005-04-28 2021-06-02 Otsuka Pharmaceutical Co., Ltd. Pharma-informatics system
JO3019B1 (ar) 2006-04-19 2016-09-05 Janssen Pharmaceutica Nv ثلاثي مستبدل 4،2،1-ثلاثي زولات
EP2063905B1 (en) 2006-09-18 2014-07-30 Raptor Pharmaceutical Inc Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates
JO2784B1 (en) 2007-10-18 2014-03-15 شركة جانسين فارماسوتيكا ان. في 5,3,1 - Triazole substitute derivative
RU2474579C2 (ru) 2007-10-18 2013-02-10 Янссен Фармацевтика Нв Тризамещенные 1,2,4-триазолы
AU2009226988B2 (en) 2008-03-19 2013-05-23 Janssen Pharmaceutica Nv Trisubstituted 1, 2, 4 -triazoles as nicotinic acetylcholine receptor modulators
CN102015655A (zh) 2008-05-09 2011-04-13 詹森药业有限公司 作为乙酰胆碱受体调节剂的三取代吡唑类
CN102316902B (zh) 2009-02-20 2014-09-24 to-BBB控股股份有限公司 基于谷胱甘肽的药物递送系统
JP2012526144A (ja) 2009-05-06 2012-10-25 ラボラトリー スキン ケア インコーポレイテッド 活性物質−リン酸カルシウム粒子複合体を含む経皮送達組成物およびその使用方法
WO2011033018A1 (en) 2009-09-17 2011-03-24 Janssen Pharmaceutica Nv Substituted n-phenyl-1-(4-pyridinyl)-1h-pyrazol-3-amines
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
AU2015281799B2 (en) * 2014-06-26 2019-11-28 Central Adelaide Local Health Network Incorporated Enzyme interacting agents
EP3749648B1 (en) * 2018-02-07 2024-10-30 Korea Research Institute of Chemical Technology N-(phenyl)-5-(phenyl)-1h-pyrazol-3-amine derivatives as tnik inhibitors for use in the treatment of cancer

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD211343A1 (de) * 1982-11-08 1984-07-11 Univ Ernst Moritz Arndt Verfahren zur synthese von pyrazolen
ATE49198T1 (de) * 1984-05-12 1990-01-15 Fisons Plc Antiinflammatorische 1,n-diarylpyrazol-3-amine, deren zusammensetzungen und verfahren zu deren herstellung.

Also Published As

Publication number Publication date
NO871879L (no) 1987-11-09
PT84831B (pt) 1990-02-08
US4803216A (en) 1989-02-07
FI871974A7 (fi) 1987-11-08
AU7258487A (en) 1987-11-12
NO871879D0 (no) 1987-05-06
PT84831A (en) 1987-06-01
CA1305157C (en) 1992-07-14
AT390732B (de) 1990-06-25
ATA290487A (de) 1989-12-15
DE3773746D1 (en) 1991-11-21
FI871974A0 (fi) 1987-05-05
EP0248523B1 (en) 1991-10-16
FI871974L (fi) 1987-11-08
EP0248523A1 (en) 1987-12-09
NZ220214A (en) 1990-06-26
KR870011101A (ko) 1987-12-21
AU595602B2 (en) 1990-04-05
IL82421A0 (en) 1987-11-30
DK231687D0 (da) 1987-05-06

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