ATA212290A - Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon - Google Patents

Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon

Info

Publication number
ATA212290A
ATA212290A AT0212290A AT212290A ATA212290A AT A212290 A ATA212290 A AT A212290A AT 0212290 A AT0212290 A AT 0212290A AT 212290 A AT212290 A AT 212290A AT A212290 A ATA212290 A AT A212290A
Authority
AT
Austria
Prior art keywords
trifluormethyl
pyrrolidinone
piperidinyl
pyrimidinyl
methyl
Prior art date
Application number
AT0212290A
Other languages
English (en)
Other versions
AT397961B (de
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ATA212290A publication Critical patent/ATA212290A/de
Application granted granted Critical
Publication of AT397961B publication Critical patent/AT397961B/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Silicon Polymers (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
AT0212290A 1989-10-27 1990-10-22 Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon AT397961B (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/427,546 US4963678A (en) 1989-10-27 1989-10-27 Process for large-scale production of BMY 21502

Publications (2)

Publication Number Publication Date
ATA212290A true ATA212290A (de) 1993-12-15
AT397961B AT397961B (de) 1994-08-25

Family

ID=23695332

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0212290A AT397961B (de) 1989-10-27 1990-10-22 Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon

Country Status (12)

Country Link
US (1) US4963678A (de)
KR (1) KR910007917A (de)
CN (1) CN1032916C (de)
AT (1) AT397961B (de)
EG (1) EG19764A (de)
ES (1) ES2026059A6 (de)
FI (1) FI95467C (de)
GR (1) GR1001125B (de)
HU (1) HU206878B (de)
NO (1) NO177303C (de)
PT (1) PT95711B (de)
YU (1) YU203290A (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU206878B (en) * 1989-10-27 1993-01-28 Bristol Myers Squibb Co Process for producing 1-//1-/2-/trifluoromethyl/-4-pyrimidinyl/-4-piperidinyl/-methyl/-2-pirrolidinone
AT398972B (de) * 1989-10-27 1995-02-27 Bristol Myers Squibb Co Verfahren zur herstellung von 1-((diazinylpiperidinyl)-methyl)-2-pyrrolidinon n
US5098904A (en) * 1990-06-27 1992-03-24 Bristol-Myers Squibb Company Cerebral function enhancing pyrimidinyl derivatives
US5401744A (en) * 1993-10-04 1995-03-28 Bristol-Myers Squibb Company Useful hemi-hydrate form of a cerebral function enhancing agent
US5538985A (en) * 1994-01-27 1996-07-23 Mitsui Toatsu Chemicals, Inc. Pyrrolidinone derivatives
CN100488952C (zh) 2001-03-15 2009-05-20 巴斯福股份公司 5-苯基嘧啶、其制备方法和中间体产物及其在防治有害真菌中的用途
US7073271B2 (en) * 2002-02-14 2006-07-11 Faro Technologies Inc. Portable coordinate measurement machine
CN106883185B (zh) * 2015-12-15 2021-07-09 重庆博腾制药科技股份有限公司 一种4-氯-2-三氟甲基嘧啶的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4826843A (en) * 1985-07-08 1989-05-02 Bristol-Myers Cerebral function enhancing diazinylpiperidine derivatives
NZ216720A (en) * 1985-07-08 1990-09-26 Bristol Myers Co Diazinylpiperidine derivatives and pharmaceutical compositions
DE3703103A1 (de) * 1987-02-03 1988-08-11 Bayer Ag Mittel gegen fischparsiten
HU206878B (en) * 1989-10-27 1993-01-28 Bristol Myers Squibb Co Process for producing 1-//1-/2-/trifluoromethyl/-4-pyrimidinyl/-4-piperidinyl/-methyl/-2-pirrolidinone

Also Published As

Publication number Publication date
GR900100776A (en) 1992-03-20
NO904587D0 (no) 1990-10-24
FI905225A0 (fi) 1990-10-24
NO177303B (no) 1995-05-15
ES2026059A6 (es) 1992-04-01
US4963678A (en) 1990-10-16
HU910050D0 (en) 1991-08-28
KR910007917A (ko) 1991-05-30
GR1001125B (el) 1993-04-28
PT95711A (pt) 1991-09-13
FI95467B (fi) 1995-10-31
EG19764A (en) 1996-01-31
YU203290A (sh) 1993-10-20
FI95467C (fi) 1996-02-12
CN1051175A (zh) 1991-05-08
NO904587L (no) 1991-04-29
PT95711B (pt) 1997-12-31
CN1032916C (zh) 1996-10-02
NO177303C (no) 1995-08-23
AT397961B (de) 1994-08-25
HU206878B (en) 1993-01-28

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee