AT258917B - Verfahren zur Herstellung von neuen Chinazolon-Derivaten - Google Patents

Verfahren zur Herstellung von neuen Chinazolon-Derivaten

Info

Publication number
AT258917B
AT258917B AT774565A AT774565A AT258917B AT 258917 B AT258917 B AT 258917B AT 774565 A AT774565 A AT 774565A AT 774565 A AT774565 A AT 774565A AT 258917 B AT258917 B AT 258917B
Authority
AT
Austria
Prior art keywords
new
production
quinazolone derivatives
quinazolone
derivatives
Prior art date
Application number
AT774565A
Other languages
English (en)
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Application granted granted Critical
Publication of AT258917B publication Critical patent/AT258917B/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT774565A 1963-05-18 1964-05-15 Verfahren zur Herstellung von neuen Chinazolon-Derivaten AT258917B (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DEF39784A DE1231705B (de) 1963-05-18 1963-05-18 Verfahren zur Herstellung von 2, 3-substituierten Chinazolon-(4)-derivaten
DEF0042147 1964-02-28

Publications (1)

Publication Number Publication Date
AT258917B true AT258917B (de) 1967-12-27

Family

ID=25975761

Family Applications (3)

Application Number Title Priority Date Filing Date
AT427764A AT254193B (de) 1963-05-18 1964-05-15 Verfahren zur Herstellung von neuen Chinazolon-Derivaten
AT774665A AT258918B (de) 1963-05-18 1964-05-15 Verfahren zur Herstellung von neuen Chinazolon-Verbindungen
AT774565A AT258917B (de) 1963-05-18 1964-05-15 Verfahren zur Herstellung von neuen Chinazolon-Derivaten

Family Applications Before (2)

Application Number Title Priority Date Filing Date
AT427764A AT254193B (de) 1963-05-18 1964-05-15 Verfahren zur Herstellung von neuen Chinazolon-Derivaten
AT774665A AT258918B (de) 1963-05-18 1964-05-15 Verfahren zur Herstellung von neuen Chinazolon-Verbindungen

Country Status (10)

Country Link
US (1) US3322756A (de)
AT (3) AT254193B (de)
BE (1) BE648093A (de)
CH (3) CH447181A (de)
DE (2) DE1231705B (de)
DK (3) DK104409C (de)
FR (1) FR3806M (de)
GB (1) GB1053063A (de)
NL (1) NL6405448A (de)
SE (3) SE314074B (de)

Families Citing this family (61)

* Cited by examiner, † Cited by third party
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US4113637A (en) * 1974-09-10 1978-09-12 Institut Francais Du Petrole Alkyl-guanidino-heterocyclic compounds, their manufacture and use as additives for fuels and lubricants
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US7671200B2 (en) * 1999-10-27 2010-03-02 Cytokinetics, Inc. Quinazolinone KSP inhibitors
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US6667300B2 (en) 2000-04-25 2003-12-23 Icos Corporation Inhibitors of human phosphatidylinositol 3-kinase delta
US6518277B1 (en) * 2000-04-25 2003-02-11 Icos Corporation Inhibitors of human phosphatidylinositol 3-kinase delta
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US6753428B2 (en) * 2001-11-20 2004-06-22 Cytokinetics, Inc. Process for the racemization of chiral quinazolinones
JP2005529076A (ja) * 2002-02-15 2005-09-29 サイトキネティクス・インコーポレーテッド キナゾリノンの合成
CN100491358C (zh) * 2002-05-09 2009-05-27 赛特凯恩蒂克公司 嘧啶酮类化合物、组合物及方法
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AU2003236527A1 (en) * 2002-06-14 2003-12-31 Cytokinetics, Inc. Compounds, compositions, and methods
AU2003256805A1 (en) * 2002-07-23 2004-02-09 Cytokinetics, Inc. Compounds compositions and methods
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JP2007505121A (ja) * 2003-09-08 2007-03-08 武田薬品工業株式会社 ジペプチジルぺプチダーゼ阻害剤
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CN102127057A (zh) * 2004-03-15 2011-07-20 武田药品工业株式会社 二肽基肽酶抑制剂
PT1761540T (pt) 2004-05-13 2016-12-07 Icos Corp Quinazolinonas como inibidores de fosfatidilinositol-3-cinase delta humana
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AU2010239312A1 (en) * 2009-04-20 2011-11-10 Gilead Calistoga Llc Methods of treatment for solid tumors
KR20120049281A (ko) 2009-07-21 2012-05-16 길리아드 칼리스토가 엘엘씨 Ｐｉ３ｋ 억제제를 이용한 간 장애의 치료
EP3581567A1 (de) 2011-04-10 2019-12-18 Atir Holding S.A. Heterocyclische verbindungen und ihre verwendung bei der behandlung von sexuellen funktionsstörungen
CA2864305C (en) 2012-03-05 2021-02-16 Gilead Calistoga Llc Polymorphic forms of (s)-2-(1-(9h-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3h)-one
EP3083630B1 (de) 2013-12-20 2019-08-21 Gilead Calistoga LLC Prozessverfahren für phosphatidylinositol-3-kinase-hemmer
EP3083623A1 (de) 2013-12-20 2016-10-26 Gilead Calistoga LLC Polymorphe formen eines hydrochloridsalzes aus (s)-2-(9h-purin-6-ylamino)propyl)-5-fluor-3-phenylchinazolin-4 (3h)-on
SG11201609877XA (en) 2014-06-13 2016-12-29 Gilead Sciences Inc Phosphatidylinositol 3-kinase inhibitors

Also Published As

Publication number Publication date
FR3806M (fr) 1966-01-03
SE314074B (de) 1969-09-01
SE314075B (de) 1969-09-01
CH447183A (de) 1967-11-30
DE1249281B (de)
DE1231705B (de) 1967-01-05
SE314076B (de) 1969-09-01
NL6405448A (de) 1964-11-19
BE648093A (de) 1964-11-19
GB1053063A (de)
CH447181A (de) 1967-11-30
DK105765C (da) 1966-11-07
US3322756A (en) 1967-05-30
DK106039C (da) 1966-12-12
DK104409C (da) 1966-05-16
AT258918B (de) 1967-12-27
CH447182A (de) 1967-11-30
AT254193B (de) 1967-05-10

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