AR231984A1 - Procedimiento para elaborar compuestos del ester del acido 7-beta-(2-(2-amino-4-tiazolil)-2-(sin)-metoxiimino-acetamido-3 cefem-4 - Google Patents

Procedimiento para elaborar compuestos del ester del acido 7-beta-(2-(2-amino-4-tiazolil)-2-(sin)-metoxiimino-acetamido-3 cefem-4

Info

Publication number
AR231984A1
AR231984A1 AR291999A AR29199983A AR231984A1 AR 231984 A1 AR231984 A1 AR 231984A1 AR 291999 A AR291999 A AR 291999A AR 29199983 A AR29199983 A AR 29199983A AR 231984 A1 AR231984 A1 AR 231984A1
Authority
AR
Argentina
Prior art keywords
metoxiimino
tiazolil
cefem
acetamido
sin
Prior art date
Application number
AR291999A
Other languages
English (en)
Spanish (es)
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Application granted granted Critical
Publication of AR231984A1 publication Critical patent/AR231984A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR291999A 1980-12-12 1983-01-31 Procedimiento para elaborar compuestos del ester del acido 7-beta-(2-(2-amino-4-tiazolil)-2-(sin)-metoxiimino-acetamido-3 cefem-4 AR231984A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH919680 1980-12-12

Publications (1)

Publication Number Publication Date
AR231984A1 true AR231984A1 (es) 1985-04-30

Family

ID=4349398

Family Applications (1)

Application Number Title Priority Date Filing Date
AR291999A AR231984A1 (es) 1980-12-12 1983-01-31 Procedimiento para elaborar compuestos del ester del acido 7-beta-(2-(2-amino-4-tiazolil)-2-(sin)-metoxiimino-acetamido-3 cefem-4

Country Status (18)

Country Link
EP (1) EP0054512A3 (OSRAM)
JP (1) JPS57123190A (OSRAM)
KR (1) KR830007683A (OSRAM)
AR (1) AR231984A1 (OSRAM)
AU (1) AU7846681A (OSRAM)
DD (1) DD208155A5 (OSRAM)
DK (1) DK550081A (OSRAM)
ES (6) ES8303424A1 (OSRAM)
FI (1) FI813946A7 (OSRAM)
GB (1) GB2111043B (OSRAM)
GR (1) GR76967B (OSRAM)
HU (1) HU185985B (OSRAM)
IE (1) IE52008B1 (OSRAM)
IL (1) IL64506A (OSRAM)
NO (1) NO814232L (OSRAM)
NZ (1) NZ199255A (OSRAM)
PT (1) PT74119B (OSRAM)
ZA (1) ZA818622B (OSRAM)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES507942A0 (es) * 1980-12-15 1983-02-01 Fujisawa Pharmaceutical Co Un procedimiento para preparar derivados del acido 7-acilaminocefalosporanico .
JPS57156495A (en) * 1981-03-23 1982-09-27 Kyoto Yakuhin Kogyo Kk Cephalosporin derivative and remedy for microbism used in oral administration
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
JPS59116291A (ja) * 1982-12-06 1984-07-05 Fujisawa Pharmaceut Co Ltd 7−置換−3−セフエム−4−カルボン酸エステルおよびその製法
US5202454A (en) * 1986-07-11 1993-04-13 Societe Nationale Des Poudres Et Explosifs Process for the manufacture of 1-bromoalkyl hydrocarbyl carbonates
KR0173796B1 (ko) * 1989-10-28 1999-02-01 기까미 기즈히꼬 세팔로스포린 화합물 및 그의 제조방법
CN101239989B (zh) * 1996-07-26 2012-12-12 吉联亚科学股份有限公司 核苷酸类似物
EP1585527A1 (en) 2003-01-14 2005-10-19 Gilead Sciences, Inc. Compositions and methods for combination antiviral therapy
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3965099A (en) * 1974-06-26 1976-06-22 Smithkline Corporation Cephalosporin esters with antibacterial activity
JPS5321192A (en) * 1976-08-10 1978-02-27 Takeda Chem Ind Ltd Cephalosporin derivatives and their preparation
US4370326A (en) * 1977-09-13 1983-01-25 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds and composition
MA18686A1 (fr) * 1978-07-07 1980-10-01 Ciba Geigy Ag Composes aminothiazoliques
ZA793391B (en) * 1978-07-07 1980-06-25 Ciba Geigy Ag Aminothiazole compounds
JPS5543011A (en) * 1978-09-20 1980-03-26 Shionogi & Co Ltd 7-halothiazolylalkoxyiminoacetamido-3-cephem compound
GR78221B (OSRAM) * 1980-02-01 1984-09-26 Ciba Geigy Ag

Also Published As

Publication number Publication date
ES516592A0 (es) 1983-08-01
DD208155A5 (de) 1984-03-28
GR76967B (OSRAM) 1984-09-04
ES516594A0 (es) 1983-11-16
ES516590A0 (es) 1983-11-16
ES507907A0 (es) 1983-02-01
IL64506A (en) 1985-05-31
ES8401078A1 (es) 1983-11-16
IL64506A0 (en) 1982-03-31
HU185985B (en) 1985-04-28
EP0054512A2 (de) 1982-06-23
JPS57123190A (en) 1982-07-31
PT74119B (de) 1983-12-19
GB2111043A (en) 1983-06-29
ES8307820A1 (es) 1983-08-01
NO814232L (no) 1982-06-14
FI813946L (fi) 1982-06-13
ES516593A0 (es) 1983-11-16
ES8401079A1 (es) 1983-11-16
EP0054512A3 (de) 1983-08-03
GB2111043B (en) 1985-02-06
ES8303424A1 (es) 1983-02-01
PT74119A (de) 1982-01-01
JPH0314038B2 (OSRAM) 1991-02-25
IE812915L (en) 1982-06-12
KR830007683A (ko) 1983-11-04
ES8401080A1 (es) 1983-11-16
DK550081A (da) 1982-06-13
FI813946A7 (fi) 1982-06-13
ES8401077A1 (es) 1983-11-16
AU7846681A (en) 1982-06-17
NZ199255A (en) 1985-08-30
ZA818622B (en) 1982-10-27
IE52008B1 (en) 1987-05-13
ES516591A0 (es) 1983-11-16

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