AR230446A1 - Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimiento - Google Patents

Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimiento

Info

Publication number
AR230446A1
AR230446A1 AR284380A AR28438081A AR230446A1 AR 230446 A1 AR230446 A1 AR 230446A1 AR 284380 A AR284380 A AR 284380A AR 28438081 A AR28438081 A AR 28438081A AR 230446 A1 AR230446 A1 AR 230446A1
Authority
AR
Argentina
Prior art keywords
procedure
quinolizidines
substituted
exclusive use
prepare new
Prior art date
Application number
AR284380A
Other languages
English (en)
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR230446A1 publication Critical patent/AR230446A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74Oxygen atoms
    • C07D211/76Oxygen atoms attached in position 2 or 6
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D455/00Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/02Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AR284380A 1978-10-13 1981-02-20 Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimiento AR230446A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1065478 1978-10-13
CH715679 1979-08-03

Publications (1)

Publication Number Publication Date
AR230446A1 true AR230446A1 (es) 1984-04-30

Family

ID=25700857

Family Applications (3)

Application Number Title Priority Date Filing Date
AR284380A AR230446A1 (es) 1978-10-13 1981-02-20 Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimiento
AR284379A AR230636A1 (es) 1978-10-13 1981-02-20 Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas e intermediarios para su uso exclusivo en ese procedimiento
AR284384A AR230637A1 (es) 1978-10-13 1981-02-20 Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas,e intermediarios para su uso exclusivo en el procedimiento

Family Applications After (2)

Application Number Title Priority Date Filing Date
AR284379A AR230636A1 (es) 1978-10-13 1981-02-20 Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas e intermediarios para su uso exclusivo en ese procedimiento
AR284384A AR230637A1 (es) 1978-10-13 1981-02-20 Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas,e intermediarios para su uso exclusivo en el procedimiento

Country Status (22)

Country Link
US (6) US4236010A (pt)
EP (2) EP0012170B1 (pt)
AR (3) AR230446A1 (pt)
AT (1) ATE877T1 (pt)
AU (1) AU533075B2 (pt)
BR (1) BR7906543A (pt)
CA (1) CA1140927A (pt)
CS (2) CS613879A2 (pt)
CU (1) CU35149A (pt)
DE (2) DE2962580D1 (pt)
DK (1) DK433779A (pt)
ES (7) ES8200680A1 (pt)
FI (2) FI66611C (pt)
GR (1) GR73144B (pt)
HU (1) HU180249B (pt)
IE (1) IE49082B1 (pt)
IL (1) IL58415A (pt)
MC (1) MC1289A1 (pt)
NO (1) NO152787C (pt)
NZ (1) NZ191763A (pt)
PH (1) PH16131A (pt)
PT (1) PT70309A (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MC1289A1 (fr) * 1978-10-13 1980-07-22 Hoffmann La Roche Phenyl quinolizidines
DK116181A (da) * 1980-04-11 1981-10-12 Hoffmann La Roche Fremgangsmaade til fremstilling af quinolizidinderivater
US4889848A (en) * 1984-11-06 1989-12-26 Hoffmann-La Roche Inc. Tricyclic pyridine derivatives
ZW17385A1 (en) * 1984-11-06 1986-02-19 Hoffmann La Roche Tricyclic pyridine derivatives
CA1317945C (en) * 1985-12-13 1993-05-18 Ulf Fischer Tricyclic pyridazopyridone derivatives
DE3614005A1 (de) * 1986-04-25 1987-10-29 Westfael Elekt Werke Verfahren zur rauchgasentschwefelung
EP0294599A3 (de) * 1987-06-12 1990-05-09 F. Hoffmann-La Roche Ag Tricyclische Pyridonderivate
US6992090B2 (en) * 2003-06-16 2006-01-31 Adolor Corporation Substituted piperidine compounds and methods of their use
US7538110B2 (en) 2005-10-27 2009-05-26 Adolor Corporation Opioid antagonists
US20100311782A1 (en) * 2009-06-08 2010-12-09 Adolor Corporation Substituted piperidinylpropanoic acid compounds and methods of their use
US8143273B2 (en) 2010-06-22 2012-03-27 Hoffman-La Roche Inc. Quinolizidine and indolizidine derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3031454A (en) * 1962-04-24 Hexahydro quinolizeses
CA668487A (en) * 1963-08-13 H. Tilford Charles Hexahydro quinolizines
GB1096589A (en) * 1964-03-31 1967-12-29 Chugai Pharmaceutical Co Ltd Novel quinolizidine derivatives or salts thereof and process for preparing the same
DE1470084A1 (de) * 1964-08-19 1969-05-29 Merck Ag E Verfahren zur Herstellung von substituierten Piperidin-derivaten
US3394141A (en) * 1965-11-12 1968-07-23 Fabio Sparatore Z-benzyaminobenzimidazoles
US3852452A (en) * 1970-02-10 1974-12-03 Ayerst Mckenna & Harrison Benzocycloheptaisoquinoline derivatives as cns depressants
MC1289A1 (fr) * 1978-10-13 1980-07-22 Hoffmann La Roche Phenyl quinolizidines

Also Published As

Publication number Publication date
EP0044573B1 (de) 1984-02-29
US4329467A (en) 1982-05-11
NO152787B (no) 1985-08-12
GR73144B (pt) 1984-02-09
CS241050B2 (en) 1986-03-13
DE2966740D1 (de) 1984-04-05
ES8105997A1 (es) 1981-07-01
ES493204A0 (es) 1981-07-01
AU533075B2 (en) 1983-10-27
US4316030A (en) 1982-02-16
FI841359A0 (fi) 1984-04-05
ES493196A0 (es) 1981-07-01
HU180249B (en) 1983-02-28
ES8106304A1 (es) 1981-06-16
ATE877T1 (de) 1982-05-15
ES8105993A1 (es) 1981-07-01
ES8105994A1 (es) 1981-07-01
FI70017B (fi) 1986-01-31
FI841359A (fi) 1984-04-05
FI66611B (fi) 1984-07-31
FI70017C (fi) 1986-09-12
ES484930A0 (es) 1981-11-16
EP0012170B1 (de) 1982-04-21
DK433779A (da) 1980-04-14
US4236010A (en) 1980-11-25
MC1289A1 (fr) 1980-07-22
AU5154579A (en) 1980-04-17
NZ191763A (en) 1984-05-31
IE791943L (en) 1980-04-13
CA1140927A (en) 1983-02-08
IL58415A0 (en) 1980-01-31
US4338444A (en) 1982-07-06
IL58415A (en) 1982-11-30
ES8200680A1 (es) 1981-11-16
IE49082B1 (en) 1985-07-24
FI66611C (fi) 1984-11-12
CS613879A2 (en) 1985-06-13
US4272627A (en) 1981-06-09
ES8105991A1 (es) 1981-07-01
EP0012170A1 (de) 1980-06-25
ES493198A0 (es) 1981-07-01
PH16131A (en) 1983-07-08
US4306067A (en) 1981-12-15
CU35149A (en) 1983-04-06
NO793300L (no) 1980-04-15
EP0044573A1 (de) 1982-01-27
DE2962580D1 (en) 1982-06-03
AR230636A1 (es) 1984-05-31
NO152787C (no) 1985-11-20
ES493199A0 (es) 1981-06-16
ES493202A0 (es) 1981-07-01
FI793182A (fi) 1980-04-14
PT70309A (en) 1979-11-01
AR230637A1 (es) 1984-05-31
ES493195A0 (es) 1981-07-01
ES8105992A1 (es) 1981-07-01
BR7906543A (pt) 1980-07-15

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