DK116181A - Fremgangsmaade til fremstilling af quinolizidinderivater - Google Patents
Fremgangsmaade til fremstilling af quinolizidinderivaterInfo
- Publication number
- DK116181A DK116181A DK116181A DK116181A DK116181A DK 116181 A DK116181 A DK 116181A DK 116181 A DK116181 A DK 116181A DK 116181 A DK116181 A DK 116181A DK 116181 A DK116181 A DK 116181A
- Authority
- DK
- Denmark
- Prior art keywords
- procedure
- preparation
- quinolizidine derivatives
- quinolizidine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/02—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH278480 | 1980-04-11 | ||
CH70181 | 1981-02-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK116181A true DK116181A (da) | 1981-10-12 |
Family
ID=25685419
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK116181A DK116181A (da) | 1980-04-11 | 1981-03-13 | Fremgangsmaade til fremstilling af quinolizidinderivater |
Country Status (18)
Country | Link |
---|---|
US (2) | US4391978A (da) |
EP (1) | EP0037990B1 (da) |
AU (1) | AU540599B2 (da) |
CA (1) | CA1142933A (da) |
CS (1) | CS222696B2 (da) |
DE (1) | DE3167549D1 (da) |
DK (1) | DK116181A (da) |
ES (1) | ES501232A0 (da) |
FI (1) | FI67700C (da) |
HU (1) | HU185633B (da) |
IE (1) | IE51108B1 (da) |
IL (1) | IL62592A (da) |
MC (1) | MC1392A1 (da) |
NO (1) | NO153258C (da) |
NZ (1) | NZ196682A (da) |
PH (1) | PH19199A (da) |
PT (1) | PT72840B (da) |
ZW (1) | ZW5581A1 (da) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK116181A (da) * | 1980-04-11 | 1981-10-12 | Hoffmann La Roche | Fremgangsmaade til fremstilling af quinolizidinderivater |
EP0094744A1 (en) * | 1982-04-23 | 1983-11-23 | Beecham Group Plc | Azabicyclobenzamides, their preparation and their pharmaceutical compositions |
US4716172A (en) * | 1986-04-10 | 1987-12-29 | Mcneilab, Inc. | 4-substituted octahydroquinolizine analgesic compounds and octahydroquinolizinium intermediates |
US6770658B2 (en) | 1998-09-09 | 2004-08-03 | Inflazyme Pharmaceuticals Ltd. | Substituted γ-phenyl-Δ-lactams and uses related thereto |
KR100917545B1 (ko) * | 2004-11-30 | 2009-09-16 | 에프. 호프만-라 로슈 아게 | 당뇨병 치료를 위한 dpp-ⅳ 억제제로서의 치환된벤조퀴놀리진 |
CN111566105A (zh) | 2018-01-08 | 2020-08-21 | 豪夫迈·罗氏有限公司 | 作为MAGL抑制剂的八氢吡啶并[1,2-α]吡嗪类化合物 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3394141A (en) * | 1965-11-12 | 1968-07-23 | Fabio Sparatore | Z-benzyaminobenzimidazoles |
US3852452A (en) * | 1970-02-10 | 1974-12-03 | Ayerst Mckenna & Harrison | Benzocycloheptaisoquinoline derivatives as cns depressants |
US3692791A (en) * | 1970-05-18 | 1972-09-19 | American Home Prod | SUBSTITUTED 2-t-BUTYL-OCTAHYDRO-2H-QUINOLIZINES |
US3948923A (en) * | 1972-03-06 | 1976-04-06 | Bayer Aktiengesellschaft | Pentahydroqunolizine derivatives |
US3997547A (en) * | 1975-07-14 | 1976-12-14 | Morton-Norwich Products, Inc. | Phenylimino-2H-quinolizines |
GB1593146A (en) * | 1976-11-05 | 1981-07-15 | Beecham Group Ltd | Octahydro-quinolizinyl benzamide derivatives |
NZ191763A (en) * | 1978-10-13 | 1984-05-31 | Hoffmann La Roche | 7-beta-phenyl-quinolidines, intermediates and pharmaceutical compositions |
DK116181A (da) * | 1980-04-11 | 1981-10-12 | Hoffmann La Roche | Fremgangsmaade til fremstilling af quinolizidinderivater |
US4339582A (en) * | 1981-08-18 | 1982-07-13 | Miles Laboratories, Inc. | Quinolizidine-propionanilide compounds |
-
1981
- 1981-03-13 DK DK116181A patent/DK116181A/da not_active Application Discontinuation
- 1981-03-17 ZW ZW55/81A patent/ZW5581A1/xx unknown
- 1981-03-31 NZ NZ196682A patent/NZ196682A/en unknown
- 1981-04-03 CA CA000374633A patent/CA1142933A/en not_active Expired
- 1981-04-03 EP EP81102536A patent/EP0037990B1/de not_active Expired
- 1981-04-03 DE DE8181102536T patent/DE3167549D1/de not_active Expired
- 1981-04-06 IL IL62592A patent/IL62592A/xx unknown
- 1981-04-06 AU AU69107/81A patent/AU540599B2/en not_active Ceased
- 1981-04-07 MC MC811510A patent/MC1392A1/xx unknown
- 1981-04-08 HU HU81900A patent/HU185633B/hu unknown
- 1981-04-09 FI FI811102A patent/FI67700C/fi not_active IP Right Cessation
- 1981-04-09 PH PH25479A patent/PH19199A/en unknown
- 1981-04-09 US US06/252,540 patent/US4391978A/en not_active Expired - Fee Related
- 1981-04-10 NO NO811263A patent/NO153258C/no unknown
- 1981-04-10 IE IE822/81A patent/IE51108B1/en unknown
- 1981-04-10 PT PT72840A patent/PT72840B/pt unknown
- 1981-04-10 ES ES501232A patent/ES501232A0/es active Granted
- 1981-04-13 CS CS812791A patent/CS222696B2/cs unknown
-
1983
- 1983-03-11 US US06/474,233 patent/US4684731A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
IL62592A0 (en) | 1981-06-29 |
NO153258C (no) | 1986-02-12 |
CS222696B2 (en) | 1983-07-29 |
FI811102L (fi) | 1981-10-12 |
FI67700B (fi) | 1985-01-31 |
NZ196682A (en) | 1984-03-30 |
PT72840A (en) | 1981-05-01 |
AU540599B2 (en) | 1984-11-29 |
FI67700C (fi) | 1985-05-10 |
PT72840B (en) | 1983-01-10 |
ES8207175A1 (es) | 1982-09-16 |
US4391978A (en) | 1983-07-05 |
ES501232A0 (es) | 1982-09-16 |
ZW5581A1 (en) | 1981-11-18 |
IE51108B1 (en) | 1986-10-01 |
MC1392A1 (fr) | 1982-04-27 |
EP0037990B1 (de) | 1984-12-05 |
IL62592A (en) | 1984-12-31 |
IE810822L (en) | 1981-10-11 |
CA1142933A (en) | 1983-03-15 |
PH19199A (en) | 1986-01-31 |
DE3167549D1 (en) | 1985-01-17 |
NO153258B (no) | 1985-11-04 |
AU6910781A (en) | 1981-10-15 |
HU185633B (en) | 1985-03-28 |
NO811263L (no) | 1981-10-12 |
EP0037990A1 (de) | 1981-10-21 |
US4684731A (en) | 1987-08-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |