AR230446A1 - Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimiento - Google Patents
Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimientoInfo
- Publication number
- AR230446A1 AR230446A1 AR284380A AR28438081A AR230446A1 AR 230446 A1 AR230446 A1 AR 230446A1 AR 284380 A AR284380 A AR 284380A AR 28438081 A AR28438081 A AR 28438081A AR 230446 A1 AR230446 A1 AR 230446A1
- Authority
- AR
- Argentina
- Prior art keywords
- procedure
- quinolizidines
- substituted
- exclusive use
- prepare new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/02—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH1065478 | 1978-10-13 | ||
CH715679 | 1979-08-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR230446A1 true AR230446A1 (es) | 1984-04-30 |
Family
ID=25700857
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR284384A AR230637A1 (es) | 1978-10-13 | 1981-02-20 | Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas,e intermediarios para su uso exclusivo en el procedimiento |
AR284379A AR230636A1 (es) | 1978-10-13 | 1981-02-20 | Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas e intermediarios para su uso exclusivo en ese procedimiento |
AR284380A AR230446A1 (es) | 1978-10-13 | 1981-02-20 | Procedimiento para preparar nuevas fenil-quinolizidinas 2-substituida e intermediarios para uso exclusivo en dicho procedimiento |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR284384A AR230637A1 (es) | 1978-10-13 | 1981-02-20 | Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas,e intermediarios para su uso exclusivo en el procedimiento |
AR284379A AR230636A1 (es) | 1978-10-13 | 1981-02-20 | Procedimiento para preparar nuevas fenilquinolicidinas 2-substituidas e intermediarios para su uso exclusivo en ese procedimiento |
Country Status (22)
Country | Link |
---|---|
US (6) | US4236010A (es) |
EP (2) | EP0012170B1 (es) |
AR (3) | AR230637A1 (es) |
AT (1) | ATE877T1 (es) |
AU (1) | AU533075B2 (es) |
BR (1) | BR7906543A (es) |
CA (1) | CA1140927A (es) |
CS (2) | CS613879A2 (es) |
CU (1) | CU35149A (es) |
DE (2) | DE2966740D1 (es) |
DK (1) | DK433779A (es) |
ES (7) | ES484930A0 (es) |
FI (2) | FI66611C (es) |
GR (1) | GR73144B (es) |
HU (1) | HU180249B (es) |
IE (1) | IE49082B1 (es) |
IL (1) | IL58415A (es) |
MC (1) | MC1289A1 (es) |
NO (1) | NO152787C (es) |
NZ (1) | NZ191763A (es) |
PH (1) | PH16131A (es) |
PT (1) | PT70309A (es) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MC1289A1 (fr) * | 1978-10-13 | 1980-07-22 | Hoffmann La Roche | Phenyl quinolizidines |
DK116181A (da) * | 1980-04-11 | 1981-10-12 | Hoffmann La Roche | Fremgangsmaade til fremstilling af quinolizidinderivater |
ZW17385A1 (en) * | 1984-11-06 | 1986-02-19 | Hoffmann La Roche | Tricyclic pyridine derivatives |
US4889848A (en) * | 1984-11-06 | 1989-12-26 | Hoffmann-La Roche Inc. | Tricyclic pyridine derivatives |
CA1317945C (en) * | 1985-12-13 | 1993-05-18 | Ulf Fischer | Tricyclic pyridazopyridone derivatives |
DE3614005A1 (de) * | 1986-04-25 | 1987-10-29 | Westfael Elekt Werke | Verfahren zur rauchgasentschwefelung |
EP0294599A3 (de) * | 1987-06-12 | 1990-05-09 | F. Hoffmann-La Roche Ag | Tricyclische Pyridonderivate |
US6992090B2 (en) * | 2003-06-16 | 2006-01-31 | Adolor Corporation | Substituted piperidine compounds and methods of their use |
US7538110B2 (en) | 2005-10-27 | 2009-05-26 | Adolor Corporation | Opioid antagonists |
US20100311782A1 (en) * | 2009-06-08 | 2010-12-09 | Adolor Corporation | Substituted piperidinylpropanoic acid compounds and methods of their use |
US8143273B2 (en) * | 2010-06-22 | 2012-03-27 | Hoffman-La Roche Inc. | Quinolizidine and indolizidine derivatives |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3031454A (en) * | 1962-04-24 | Hexahydro quinolizeses | ||
CA668487A (en) * | 1963-08-13 | H. Tilford Charles | Hexahydro quinolizines | |
GB1096589A (en) * | 1964-03-31 | 1967-12-29 | Chugai Pharmaceutical Co Ltd | Novel quinolizidine derivatives or salts thereof and process for preparing the same |
DE1470084A1 (de) * | 1964-08-19 | 1969-05-29 | Merck Ag E | Verfahren zur Herstellung von substituierten Piperidin-derivaten |
US3394141A (en) * | 1965-11-12 | 1968-07-23 | Fabio Sparatore | Z-benzyaminobenzimidazoles |
US3852452A (en) * | 1970-02-10 | 1974-12-03 | Ayerst Mckenna & Harrison | Benzocycloheptaisoquinoline derivatives as cns depressants |
MC1289A1 (fr) * | 1978-10-13 | 1980-07-22 | Hoffmann La Roche | Phenyl quinolizidines |
-
1979
- 1979-10-05 MC MC791408A patent/MC1289A1/xx unknown
- 1979-10-05 NZ NZ191763A patent/NZ191763A/en unknown
- 1979-10-08 AU AU51545/79A patent/AU533075B2/en not_active Ceased
- 1979-10-08 IL IL58415A patent/IL58415A/xx unknown
- 1979-10-09 CS CS796861A patent/CS613879A2/cs unknown
- 1979-10-09 CA CA000337172A patent/CA1140927A/en not_active Expired
- 1979-10-10 HU HU79HO2187A patent/HU180249B/hu unknown
- 1979-10-10 PH PH23149A patent/PH16131A/en unknown
- 1979-10-11 EP EP79103907A patent/EP0012170B1/de not_active Expired
- 1979-10-11 ES ES484930A patent/ES484930A0/es active Granted
- 1979-10-11 AT AT79103907T patent/ATE877T1/de not_active IP Right Cessation
- 1979-10-11 CU CU7935149A patent/CU35149A/es unknown
- 1979-10-11 DE DE8181106675T patent/DE2966740D1/de not_active Expired
- 1979-10-11 DE DE7979103907T patent/DE2962580D1/de not_active Expired
- 1979-10-11 GR GR60236A patent/GR73144B/el unknown
- 1979-10-11 EP EP81106675A patent/EP0044573B1/de not_active Expired
- 1979-10-12 PT PT70309A patent/PT70309A/pt unknown
- 1979-10-12 FI FI793182A patent/FI66611C/fi not_active IP Right Cessation
- 1979-10-12 DK DK433779A patent/DK433779A/da not_active Application Discontinuation
- 1979-10-12 BR BR7906543A patent/BR7906543A/pt unknown
- 1979-10-12 NO NO793300A patent/NO152787C/no unknown
- 1979-10-12 IE IE1943/79A patent/IE49082B1/en unknown
- 1979-10-15 US US06/085,096 patent/US4236010A/en not_active Expired - Lifetime
-
1980
- 1980-05-12 US US06/148,646 patent/US4272627A/en not_active Expired - Lifetime
- 1980-07-08 ES ES493195A patent/ES493195A0/es active Granted
- 1980-07-08 ES ES493199A patent/ES493199A0/es active Granted
- 1980-07-08 ES ES493202A patent/ES493202A0/es active Granted
- 1980-07-08 ES ES493204A patent/ES493204A0/es active Granted
- 1980-07-08 ES ES493198A patent/ES8105997A1/es not_active Expired
- 1980-07-08 ES ES493196A patent/ES8105992A1/es not_active Expired
- 1980-12-18 US US06/217,863 patent/US4306067A/en not_active Expired - Fee Related
- 1980-12-18 US US06/217,888 patent/US4316030A/en not_active Expired - Fee Related
- 1980-12-18 US US06/217,887 patent/US4329467A/en not_active Expired - Fee Related
- 1980-12-18 US US06/217,864 patent/US4338444A/en not_active Expired - Fee Related
-
1981
- 1981-02-20 AR AR284384A patent/AR230637A1/es active
- 1981-02-20 AR AR284379A patent/AR230636A1/es active
- 1981-02-20 AR AR284380A patent/AR230446A1/es active
-
1984
- 1984-04-05 FI FI841359A patent/FI70017C/fi not_active IP Right Cessation
- 1984-08-13 CS CS846138A patent/CS241050B2/cs unknown
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