AR220689A1 - Procedimiento para obtener compuestos de n-(2-mercapto,2-benzoiltio,2-alcanoiltio-2-mercapto o 2-alquil)-acetil-tiazolidin o tiazancarboxilicos y sus sales - Google Patents

Procedimiento para obtener compuestos de n-(2-mercapto,2-benzoiltio,2-alcanoiltio-2-mercapto o 2-alquil)-acetil-tiazolidin o tiazancarboxilicos y sus sales

Info

Publication number
AR220689A1
AR220689A1 AR270203A AR27020377A AR220689A1 AR 220689 A1 AR220689 A1 AR 220689A1 AR 270203 A AR270203 A AR 270203A AR 27020377 A AR27020377 A AR 27020377A AR 220689 A1 AR220689 A1 AR 220689A1
Authority
AR
Argentina
Prior art keywords
mercapto
tiazancarboxilicos
benzoiltio
alcanoiltio
tiazolidin
Prior art date
Application number
AR270203A
Other languages
English (en)
Spanish (es)
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Application granted granted Critical
Publication of AR220689A1 publication Critical patent/AR220689A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/041,3-Thiazines; Hydrogenated 1,3-thiazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AR270203A 1976-12-03 1977-11-30 Procedimiento para obtener compuestos de n-(2-mercapto,2-benzoiltio,2-alcanoiltio-2-mercapto o 2-alquil)-acetil-tiazolidin o tiazancarboxilicos y sus sales AR220689A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74728176A 1976-12-03 1976-12-03
US83610777A 1977-09-23 1977-09-23

Publications (1)

Publication Number Publication Date
AR220689A1 true AR220689A1 (es) 1980-11-28

Family

ID=27114718

Family Applications (1)

Application Number Title Priority Date Filing Date
AR270203A AR220689A1 (es) 1976-12-03 1977-11-30 Procedimiento para obtener compuestos de n-(2-mercapto,2-benzoiltio,2-alcanoiltio-2-mercapto o 2-alquil)-acetil-tiazolidin o tiazancarboxilicos y sus sales

Country Status (28)

Country Link
JP (1) JPS5382778A (pt)
AR (1) AR220689A1 (pt)
AT (1) AT363467B (pt)
AU (1) AU518147B2 (pt)
BG (1) BG32269A3 (pt)
CA (1) CA1146940A (pt)
CH (1) CH634062A5 (pt)
DD (1) DD133798A5 (pt)
DE (1) DE2752719C2 (pt)
DK (1) DK152494C (pt)
EG (1) EG13037A (pt)
ES (1) ES464555A1 (pt)
FI (1) FI67378C (pt)
FR (1) FR2372817A1 (pt)
GB (1) GB1578940A (pt)
GR (1) GR72453B (pt)
HK (1) HK55881A (pt)
IE (1) IE46169B1 (pt)
IL (1) IL53352A0 (pt)
IN (1) IN146945B (pt)
IT (1) IT1092179B (pt)
NL (3) NL171055C (pt)
NO (1) NO148416C (pt)
NZ (1) NZ185800A (pt)
PT (1) PT67352B (pt)
RO (2) RO78013A (pt)
SE (1) SE441267B (pt)
YU (1) YU41823B (pt)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2395998A1 (fr) * 1977-06-29 1979-01-26 Yoshitomi Pharmaceutical Nouveaux derives de la thiazolidine et leur application dans le traitement de l'hypertension
JPS5455565A (en) * 1977-10-06 1979-05-02 Santen Pharmaceut Co Ltd Novel thiazolidine derivative
JPS557255A (en) * 1978-07-03 1980-01-19 Santen Pharmaceut Co Ltd Thiazolidine derivative
AU528115B2 (en) * 1978-04-08 1983-04-14 Santen Pharmaceutical Co. Ltd. Antihypertensive 4-thiazolidine/carboxylic acids
JPS5531022A (en) * 1978-08-24 1980-03-05 Yoshitomi Pharmaceut Ind Ltd Hydroxamic acid derivative and its preparation
GR73585B (pt) * 1978-09-11 1984-03-26 Univ Miami
JPS5540622A (en) * 1978-09-14 1980-03-22 Santen Pharmaceut Co Ltd Hypotensive agent
JPS5829950B2 (ja) * 1978-10-05 1983-06-25 ウェルファイド株式会社 環状イミノカルボン酸誘導体およびその塩類
US4483861A (en) * 1978-10-31 1984-11-20 Santen Pharmaceutical Co., Ltd. Antihypertensive sulfur-containing compounds
JPS5562060A (en) * 1978-10-31 1980-05-10 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS55124757A (en) * 1979-03-17 1980-09-26 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS565415A (en) * 1979-06-26 1981-01-20 Santen Pharmaceut Co Ltd Ester-type hypotensor
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
JPS5683483A (en) * 1979-12-13 1981-07-08 Santen Pharmaceut Co Ltd Thiazolidine compound
JPS56139455A (en) * 1980-04-02 1981-10-30 Santen Pharmaceut Co Ltd Sulfur-containing acylaminoacid
DE3152643A1 (de) * 1980-12-29 1982-12-16 Santen Pharmaceutical Co Ltd Heterocyclic 5-membered ring compounds
JPH0662529B2 (ja) * 1984-07-13 1994-08-17 三共株式会社 アミノ酸誘導体
DE3685829T2 (de) * 1985-02-04 1992-12-17 Searle & Co Heterocyclische amide.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446100C3 (de) * 1974-09-26 1982-01-14 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren Phenoxyalkancarbonsäureamide von Thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und Arzneimittel
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
FR2372817B1 (pt) 1981-06-19
DK152494C (da) 1988-07-25
DE2752719C2 (de) 1982-03-25
RO72596B (ro) 1983-07-30
IL53352A0 (en) 1978-01-31
NL171055C (nl) 1983-02-01
IN146945B (pt) 1979-10-20
SE7713722L (sv) 1978-06-04
GB1578940A (en) 1980-11-12
FI67378C (fi) 1985-03-11
CA1146940A (en) 1983-05-24
YU41823B (en) 1988-02-29
IT1092179B (it) 1985-07-06
RO72596A (ro) 1983-08-03
NL8201146A (nl) 1982-07-01
BG32269A3 (en) 1982-06-15
NL7713274A (nl) 1978-06-06
IE46169B1 (en) 1983-03-09
NL8201145A (nl) 1982-07-01
DE2752719A1 (de) 1978-06-08
FR2372817A1 (fr) 1978-06-30
SE441267B (sv) 1985-09-23
FI67378B (fi) 1984-11-30
DK152494B (da) 1988-03-07
PT67352B (fr) 1979-05-15
GR72453B (pt) 1983-11-09
AU518147B2 (en) 1981-09-17
NO774126L (no) 1978-06-06
FI773640A (fi) 1978-06-04
NZ185800A (en) 1980-04-28
JPS5382778A (en) 1978-07-21
RO78013A (ro) 1981-12-25
ES464555A1 (es) 1978-09-01
DD133798A5 (de) 1979-01-24
EG13037A (en) 1980-12-31
NO148416B (no) 1983-06-27
AT363467B (de) 1981-08-10
PT67352A (fr) 1978-01-01
ATA857677A (de) 1981-01-15
NO148416C (no) 1983-10-12
CH634062A5 (en) 1983-01-14
DK538277A (da) 1978-06-04
JPS618834B2 (pt) 1986-03-18
HK55881A (en) 1981-11-20
AU3037977A (en) 1979-05-17
IE46169L (en) 1978-06-03
YU283777A (en) 1983-01-21

Similar Documents

Publication Publication Date Title
AR220525A1 (es) Procedimiento para obtener nuevos derivados de n-(2-mercapto,2-alcanoiltio,2-mercapto-alquil,2-alquiltio-alquiltio o2-alcanoiltioalquil)-acetil-prolina
AR228575A1 (es) Procedimiento para obtener derivados de 7-hidroximetil o 7-carboxicamptotecina y sus sales
AR228444A1 (es) Procedimiento para preparar derivados de 5-bencil-tiazolidin-2,4-diona y sus sales
AR226290A1 (es) Procedimiento para preparar nuetoalquil-(c1-c3)-carbonil)-l-provos derivados de acido-1-(mercaplina,y sus sales
AR220689A1 (es) Procedimiento para obtener compuestos de n-(2-mercapto,2-benzoiltio,2-alcanoiltio-2-mercapto o 2-alquil)-acetil-tiazolidin o tiazancarboxilicos y sus sales
AR220686A1 (es) Procedimiento para obtener derivados de 2 amino-2-desoxi-3-o-(propilcarbamoilmetil)-carbamoilmetil-glucopiranosa y sus sales
AR224495A1 (es) Procedimiento para la preparacion de derivados de 1-fenil-7,8-dihidroxi o 7,8-dialcanoiloxi-1,3,4,5-tetrahidro-1h-3-benzazepina y sus sales
AR221833A1 (es) Procedimiento para obtener derivados de 1-(3-hidroxipirrolidin-3-ilcarbonilamino o 4-hidroxipiperidin-4-ilcarbonilamino-)-2-(3,5-dihidroxi-4-amino-6 hidroximetil-2,3,5,6-tetrahidropiran-2-iloxi)-3-hidroxi-4-(5-hidroxi-6 aminometil-2,3,5,6-tetrahidropiran-2-iloxi)-5-aminociclohexano y sus sales
AR230280A1 (es) Procedimiento para obtener derivados de carboestirilo y sus sales
AR223069A1 (es) Polieterpoliaminas y sus sales,procedimiento para su preparacion y su empleo
AR228144A1 (es) Procedimiento para obtener derivados de 5-fenil-triazolidina-2,4-diona y sus sales
AR215886A1 (es) Procedimiento para la preparacion de derivados de n-(5-tetrazolil)-4-oxo-4h-pirimido(2,1-b)benzotiazol y sales de los mismos
AR218454A1 (es) Procedimiento para preparar derivados de 7-beta-amino o 7-beta-(2-oximino-2-furil o 2-fenilacetamido)-3-(sulfoalquil o 3-sulfoaminalquilo o 3-sulfamilalquil-tetrazol-5-il)tiometil 3-cefem-4-carboxilicos y sus sales
AR220129A1 (es) Procedimiento para la desnitrosacion de n-(1-etilpropil)-n-nitroso-2,6-dinitro-3,4-xilidina
AR227272A1 (es) Procedimiento para la obtencion de compuestos de n-oxaciclil-alquil-piperidil-diaza y sus sales
AR226578A1 (es) Procedimiento para preparar tetrapeptidos de try-d-ala-gly-l-(n alfa-substituido)-phe-amida y sus sales
AR218242A1 (es) Procedimiento para la produccion de derivados de acidos n-(2-(imidazolil o tiazolil-metil-tio)-etil)-amidino formico
AR218951A1 (es) Procedimiento para obtener derivados de acidos 3-(1-metiltetrazolil-tiometil)-7-glicilamido-1-oxadetia-3-cefem-4-carboxilicos y sus sales
AR231539A1 (es) Procedimiento para la elaboracion de nuevos derivados de la curamina o del 4n-1-benzopirano y sus sales
AR224610A1 (es) Procedimiento para obtener derivados,de acidos benzacil-benzimidazol-2-carboxilicos o de 2-hidroximetilo y sus sales
AR213184A1 (es) Procedimiento para preparar derivados de 1,4-etan-6-oxo-perhidroquinoleina y sus sales
AR218452A1 (es) Procedimiento para obtener derivados de 4-(3-(4-piperidil)-propil)-quinoleina y sus sales
AR228036A1 (es) Procedimiento para obtener derivados de 1-tio-alcanoilprolina y sus sales
AR218465A1 (es) Procedimiento para obtener compuestos de 13-(1-sustituido-4-piperiliden)-8,13-dihidro-benzo(e)-naft(2,1-b)-oxepina y sus sales
AR219076A1 (es) Procedimiento para adobar cueros