AR212012A1 - PROCEDURE FOR THE PREPARATION OF N, N-DIMETHYL-ALPHA-PHENYL-M-DIOXANE-5-METHYLAMINES AND 1- (ALPHA-DIOXAN-5-IL) -BENZYL-PYRROLIDINE OR PIPERIDINE AND THEIR ACID SALTS OF ADDITION PHARMACEUTICALLY ACCEPTABLE - Google Patents

PROCEDURE FOR THE PREPARATION OF N, N-DIMETHYL-ALPHA-PHENYL-M-DIOXANE-5-METHYLAMINES AND 1- (ALPHA-DIOXAN-5-IL) -BENZYL-PYRROLIDINE OR PIPERIDINE AND THEIR ACID SALTS OF ADDITION PHARMACEUTICALLY ACCEPTABLE

Info

Publication number
AR212012A1
AR212012A1 AR258799A AR25879975A AR212012A1 AR 212012 A1 AR212012 A1 AR 212012A1 AR 258799 A AR258799 A AR 258799A AR 25879975 A AR25879975 A AR 25879975A AR 212012 A1 AR212012 A1 AR 212012A1
Authority
AR
Argentina
Prior art keywords
alpha
methylamines
dioxan
pyrrolidine
piperidine
Prior art date
Application number
AR258799A
Other languages
Spanish (es)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of AR212012A1 publication Critical patent/AR212012A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
AR258799A 1972-12-08 1975-05-14 PROCEDURE FOR THE PREPARATION OF N, N-DIMETHYL-ALPHA-PHENYL-M-DIOXANE-5-METHYLAMINES AND 1- (ALPHA-DIOXAN-5-IL) -BENZYL-PYRROLIDINE OR PIPERIDINE AND THEIR ACID SALTS OF ADDITION PHARMACEUTICALLY ACCEPTABLE AR212012A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US31322172A 1972-12-08 1972-12-08

Publications (1)

Publication Number Publication Date
AR212012A1 true AR212012A1 (en) 1978-04-28

Family

ID=23214841

Family Applications (3)

Application Number Title Priority Date Filing Date
AR251422A AR206306A1 (en) 1972-12-08 1973-01-01 PROCEDURE FOR THE PREPARATION OF META-DIOXANE-5-METHYLAMINES AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OF ADDITION
AR251423A AR212416A1 (en) 1972-12-08 1973-12-07 PROCEDURE FOR THE PREPARATION OF N-METHYL ALPHA-PHENYL-O 3-PYRIDYL-5-M-DIOXANE-METHYLAMINE COMPOUNDS AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS
AR258799A AR212012A1 (en) 1972-12-08 1975-05-14 PROCEDURE FOR THE PREPARATION OF N, N-DIMETHYL-ALPHA-PHENYL-M-DIOXANE-5-METHYLAMINES AND 1- (ALPHA-DIOXAN-5-IL) -BENZYL-PYRROLIDINE OR PIPERIDINE AND THEIR ACID SALTS OF ADDITION PHARMACEUTICALLY ACCEPTABLE

Family Applications Before (2)

Application Number Title Priority Date Filing Date
AR251422A AR206306A1 (en) 1972-12-08 1973-01-01 PROCEDURE FOR THE PREPARATION OF META-DIOXANE-5-METHYLAMINES AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OF ADDITION
AR251423A AR212416A1 (en) 1972-12-08 1973-12-07 PROCEDURE FOR THE PREPARATION OF N-METHYL ALPHA-PHENYL-O 3-PYRIDYL-5-M-DIOXANE-METHYLAMINE COMPOUNDS AND ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS

Country Status (27)

Country Link
JP (2) JPS5734835B2 (en)
AR (3) AR206306A1 (en)
AT (2) AT332396B (en)
BE (1) BE808340A (en)
BG (4) BG21223A3 (en)
CA (2) CA1014560A (en)
CH (4) CH605903A5 (en)
CS (3) CS193480B2 (en)
CY (1) CY1017A (en)
DD (3) DD115653A5 (en)
DE (1) DE2361340C2 (en)
DK (1) DK134717B (en)
ES (4) ES421291A1 (en)
FR (1) FR2209578B1 (en)
GB (2) GB1455997A (en)
HK (1) HK60479A (en)
HU (2) HU168620B (en)
IE (1) IE40226B1 (en)
IL (1) IL43773A (en)
KE (1) KE2976A (en)
MY (1) MY8000064A (en)
NL (1) NL7316839A (en)
PH (2) PH15197A (en)
SE (3) SE403377B (en)
SU (4) SU578001A3 (en)
YU (3) YU35447B (en)
ZA (1) ZA739207B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9376409B2 (en) * 2012-05-09 2016-06-28 Boehringer Ingelheim International Gmbh Methods for making oxetan-3-ylmethanamines
LV14983B (en) * 2013-10-15 2015-06-20 Olainfarm, A/S Method for producing intermediates of phenibut

Also Published As

Publication number Publication date
BE808340A (en) 1974-06-07
SU663305A3 (en) 1979-05-15
BG21409A3 (en) 1976-05-20
CA1024150A (en) 1978-01-10
YU36171B (en) 1982-02-25
CS222209B2 (en) 1983-05-27
DK134717B (en) 1977-01-03
DE2361340A1 (en) 1974-06-12
BG26205A4 (en) 1979-02-15
JPS4987680A (en) 1974-08-22
SE428378B (en) 1983-06-27
DD110864A5 (en) 1975-01-12
ATA1026073A (en) 1975-10-15
BG22386A3 (en) 1977-02-20
SE417196B (en) 1981-03-02
SE7701795L (en) 1977-02-17
CS193480B2 (en) 1979-10-31
IL43773A0 (en) 1974-03-14
NL7316839A (en) 1974-06-11
JPS4987681A (en) 1974-08-22
YU318573A (en) 1981-06-30
HU168620B (en) 1976-06-28
YU318473A (en) 1980-09-25
YU35447B (en) 1981-02-28
FR2209578B1 (en) 1977-09-02
FR2209578A1 (en) 1974-07-05
HK60479A (en) 1979-08-31
DD109625A5 (en) 1974-11-12
MY8000064A (en) 1980-12-31
AT330773B (en) 1976-07-26
YU109380A (en) 1981-04-30
BG21223A3 (en) 1976-03-20
SE7701796L (en) 1977-02-17
SE403377B (en) 1978-08-14
CH614439A5 (en) 1979-11-30
AT332396B (en) 1976-09-27
SU587861A3 (en) 1978-01-05
CH605903A5 (en) 1978-10-13
ES444911A1 (en) 1977-09-01
ES421291A1 (en) 1976-07-01
HU168763B (en) 1976-07-28
IL43773A (en) 1979-05-31
YU36020B (en) 1981-11-13
IE40226B1 (en) 1979-04-11
KE2976A (en) 1979-07-20
CH619219A5 (en) 1980-09-15
AR206306A1 (en) 1976-07-15
CY1017A (en) 1979-11-23
JPS5734835B2 (en) 1982-07-26
ES421290A1 (en) 1976-07-01
ZA739207B (en) 1975-07-30
CA1014560A (en) 1977-07-26
ATA1026173A (en) 1976-01-15
GB1455998A (en) 1976-11-17
SU578001A3 (en) 1977-10-25
JPS5742633B2 (en) 1982-09-09
AR212416A1 (en) 1978-07-14
DE2361340C2 (en) 1983-11-24
CH630914A5 (en) 1982-07-15
AU6321773A (en) 1975-06-05
CS222208B2 (en) 1983-05-27
GB1455997A (en) 1976-11-17
DK134717C (en) 1977-05-31
IE40226L (en) 1974-06-08
PH15197A (en) 1982-09-17
SU648081A3 (en) 1979-02-15
ES444716A1 (en) 1977-05-16
PH14923A (en) 1982-01-29
DD115653A5 (en) 1975-10-12

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