AR208068A1 - Un procedimiento para preparar derivados de acidos 7-acilamido-3-halo-cefem-4-carboxilico los esteres y las sales farmaceuticamente aceptables de los mismos - Google Patents

Un procedimiento para preparar derivados de acidos 7-acilamido-3-halo-cefem-4-carboxilico los esteres y las sales farmaceuticamente aceptables de los mismos

Info

Publication number
AR208068A1
AR208068A1 AR256545A AR25654574A AR208068A1 AR 208068 A1 AR208068 A1 AR 208068A1 AR 256545 A AR256545 A AR 256545A AR 25654574 A AR25654574 A AR 25654574A AR 208068 A1 AR208068 A1 AR 208068A1
Authority
AR
Argentina
Prior art keywords
acilamido
cefem
halo
esters
procedure
Prior art date
Application number
AR256545A
Other languages
English (en)
Spanish (es)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of AR208068A1 publication Critical patent/AR208068A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02Preparation
    • C07D501/04Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR256545A 1973-02-23 1974-01-01 Un procedimiento para preparar derivados de acidos 7-acilamido-3-halo-cefem-4-carboxilico los esteres y las sales farmaceuticamente aceptables de los mismos AR208068A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US33541473A 1973-02-23 1973-02-23

Publications (1)

Publication Number Publication Date
AR208068A1 true AR208068A1 (es) 1976-11-30

Family

ID=23311677

Family Applications (3)

Application Number Title Priority Date Filing Date
AR256545A AR208068A1 (es) 1973-02-23 1974-01-01 Un procedimiento para preparar derivados de acidos 7-acilamido-3-halo-cefem-4-carboxilico los esteres y las sales farmaceuticamente aceptables de los mismos
AR252494A AR200908A1 (es) 1973-02-23 1974-02-22 Procedimiento para preparar acidos 7-acilamido-3-halo-3-cefem-4 carboxilicos, esteres y sales farmaceuticamente aceptables de los mismos
AR256546A AR201709A1 (es) 1973-02-23 1974-11-15 Proceso para preparar 3-halocefalosporinas

Family Applications After (2)

Application Number Title Priority Date Filing Date
AR252494A AR200908A1 (es) 1973-02-23 1974-02-22 Procedimiento para preparar acidos 7-acilamido-3-halo-3-cefem-4 carboxilicos, esteres y sales farmaceuticamente aceptables de los mismos
AR256546A AR201709A1 (es) 1973-02-23 1974-11-15 Proceso para preparar 3-halocefalosporinas

Country Status (34)

Country Link
JP (4) JPS612677B2 (xx)
AR (3) AR208068A1 (xx)
AT (1) AT333952B (xx)
BE (1) BE811494A (xx)
BG (1) BG22404A3 (xx)
BR (1) BR7401385D0 (xx)
CA (1) CA1032532A (xx)
CH (1) CH594686A5 (xx)
CS (1) CS189625B2 (xx)
CY (1) CY1042A (xx)
DD (1) DD110277A5 (xx)
DE (1) DE2408686C2 (xx)
ES (1) ES423532A1 (xx)
FI (1) FI63240C (xx)
FR (1) FR2218878B1 (xx)
GB (1) GB1458293A (xx)
GT (1) GT197432132A (xx)
HK (1) HK19980A (xx)
HU (1) HU167749B (xx)
IE (1) IE38916B1 (xx)
IL (1) IL44263A (xx)
KE (1) KE3026A (xx)
MW (1) MW574A1 (xx)
MY (1) MY8100023A (xx)
NL (1) NL181010C (xx)
NO (2) NO148376C (xx)
OA (1) OA04688A (xx)
PH (1) PH14014A (xx)
PL (1) PL88714B1 (xx)
RO (1) RO64595A (xx)
SE (1) SE411211B (xx)
YU (2) YU36971B (xx)
ZA (1) ZA741190B (xx)
ZM (1) ZM3674A1 (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT342197B (de) * 1975-02-20 1978-03-28 Ciba Geigy Ag Neues verfahren zur herstellung von 3-cephemverbindungen
CH622802A5 (xx) * 1975-08-20 1981-04-30 Ciba Geigy Ag
IE45158B1 (en) * 1976-08-16 1982-06-30 Lilly Co Eli 3-chloro-cephem synthesis
PH17188A (en) * 1977-03-14 1984-06-14 Fujisawa Pharmaceutical Co New cephem and cepham compounds and their pharmaceutical compositions and method of use
JPS62112053U (xx) * 1985-12-27 1987-07-16
JPH0676861B2 (ja) * 1988-05-24 1994-09-28 リンナイ株式会社 温風暖房機の制御装置
IT1255458B (it) * 1992-05-11 1995-11-02 Col Marco Da Procedimento per la preparazione di derivati beta-lattamici alogenati

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2143211B1 (xx) * 1971-06-24 1975-10-31 Fujisawa Pharmaceutical Co

Also Published As

Publication number Publication date
CA1032532A (en) 1978-06-06
NO148376C (no) 1983-09-28
FR2218878A1 (xx) 1974-09-20
JPS49116095A (xx) 1974-11-06
FI63240B (fi) 1983-01-31
AT333952B (de) 1976-12-27
BE811494A (fr) 1974-08-22
DD110277A5 (xx) 1974-12-12
MY8100023A (en) 1981-12-31
KE3026A (en) 1980-03-14
JPS613356B2 (xx) 1986-01-31
IE38916B1 (en) 1978-06-21
NO148376B (no) 1983-06-20
NL7402486A (xx) 1974-08-27
JPS612677B2 (xx) 1986-01-27
JPS56138193A (en) 1981-10-28
IL44263A0 (en) 1974-05-16
SE411211B (sv) 1979-12-10
JPS613357B2 (xx) 1986-01-31
BG22404A3 (xx) 1977-02-20
GT197432132A (es) 1975-08-16
RO64595A (ro) 1981-01-30
NL181010C (nl) 1987-06-01
DE2408686C2 (de) 1986-08-28
DE2408686A1 (de) 1974-09-05
GB1458293A (en) 1976-12-15
MW574A1 (en) 1975-05-13
HU167749B (xx) 1975-12-25
YU99880A (en) 1983-04-27
PH14014A (en) 1980-12-08
AR200908A1 (es) 1974-12-27
NO740607L (no) 1974-08-26
OA04688A (fr) 1980-07-31
IL44263A (en) 1977-10-31
CY1042A (en) 1980-08-01
AR201709A1 (es) 1975-04-08
JPS56138195A (en) 1981-10-28
CH594686A5 (xx) 1978-01-31
ZM3674A1 (en) 1975-11-21
YU46374A (en) 1982-06-18
PL88714B1 (en) 1976-09-30
ATA142474A (de) 1976-04-15
ES423532A1 (es) 1976-06-01
IE38916L (en) 1974-08-23
JPS56138194A (en) 1981-10-28
BR7401385D0 (pt) 1974-11-05
HK19980A (en) 1980-04-25
CS189625B2 (en) 1979-04-30
FR2218878B1 (xx) 1977-03-11
JPS613358B2 (xx) 1986-01-31
AU6591574A (en) 1975-08-28
ZA741190B (en) 1975-09-24
NO792609L (no) 1974-08-26
NL181010B (nl) 1987-01-02
FI63240C (fi) 1983-05-10
YU37347B (en) 1984-08-31
YU36971B (en) 1984-08-31

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