AR208068A1 - A PROCEDURE FOR PREPARING DERIVATIVES OF 7-ACILAMIDO-3-HALO-CEFEM-4-CARBOXYL ACIDS, THE ESTERS AND THE PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF - Google Patents

A PROCEDURE FOR PREPARING DERIVATIVES OF 7-ACILAMIDO-3-HALO-CEFEM-4-CARBOXYL ACIDS, THE ESTERS AND THE PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF

Info

Publication number
AR208068A1
AR208068A1 AR256545A AR25654574A AR208068A1 AR 208068 A1 AR208068 A1 AR 208068A1 AR 256545 A AR256545 A AR 256545A AR 25654574 A AR25654574 A AR 25654574A AR 208068 A1 AR208068 A1 AR 208068A1
Authority
AR
Argentina
Prior art keywords
acilamido
cefem
halo
esters
procedure
Prior art date
Application number
AR256545A
Other languages
Spanish (es)
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of AR208068A1 publication Critical patent/AR208068A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02Preparation
    • C07D501/04Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR256545A 1973-02-23 1974-01-01 A PROCEDURE FOR PREPARING DERIVATIVES OF 7-ACILAMIDO-3-HALO-CEFEM-4-CARBOXYL ACIDS, THE ESTERS AND THE PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AR208068A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US33541473A 1973-02-23 1973-02-23

Publications (1)

Publication Number Publication Date
AR208068A1 true AR208068A1 (en) 1976-11-30

Family

ID=23311677

Family Applications (3)

Application Number Title Priority Date Filing Date
AR256545A AR208068A1 (en) 1973-02-23 1974-01-01 A PROCEDURE FOR PREPARING DERIVATIVES OF 7-ACILAMIDO-3-HALO-CEFEM-4-CARBOXYL ACIDS, THE ESTERS AND THE PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
AR252494A AR200908A1 (en) 1973-02-23 1974-02-22 PROCEDURE FOR PREPARING 7-ACILAMIDO-3-HALO-3-CEFEM-4 CARBOXYL ACIDS, ESTERS AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
AR256546A AR201709A1 (en) 1973-02-23 1974-11-15 PROCESS TO PREPARE 3-HALOCEPHALOSPORINS

Family Applications After (2)

Application Number Title Priority Date Filing Date
AR252494A AR200908A1 (en) 1973-02-23 1974-02-22 PROCEDURE FOR PREPARING 7-ACILAMIDO-3-HALO-3-CEFEM-4 CARBOXYL ACIDS, ESTERS AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
AR256546A AR201709A1 (en) 1973-02-23 1974-11-15 PROCESS TO PREPARE 3-HALOCEPHALOSPORINS

Country Status (34)

Country Link
JP (4) JPS612677B2 (en)
AR (3) AR208068A1 (en)
AT (1) AT333952B (en)
BE (1) BE811494A (en)
BG (1) BG22404A3 (en)
BR (1) BR7401385D0 (en)
CA (1) CA1032532A (en)
CH (1) CH594686A5 (en)
CS (1) CS189625B2 (en)
CY (1) CY1042A (en)
DD (1) DD110277A5 (en)
DE (1) DE2408686C2 (en)
ES (1) ES423532A1 (en)
FI (1) FI63240C (en)
FR (1) FR2218878B1 (en)
GB (1) GB1458293A (en)
GT (1) GT197432132A (en)
HK (1) HK19980A (en)
HU (1) HU167749B (en)
IE (1) IE38916B1 (en)
IL (1) IL44263A (en)
KE (1) KE3026A (en)
MW (1) MW574A1 (en)
MY (1) MY8100023A (en)
NL (1) NL181010C (en)
NO (2) NO148376C (en)
OA (1) OA04688A (en)
PH (1) PH14014A (en)
PL (1) PL88714B1 (en)
RO (1) RO64595A (en)
SE (1) SE411211B (en)
YU (2) YU36971B (en)
ZA (1) ZA741190B (en)
ZM (1) ZM3674A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT342197B (en) * 1975-02-20 1978-03-28 Ciba Geigy Ag NEW PROCESS FOR PRODUCING 3-CEPHEM CONNECTIONS
CH622802A5 (en) * 1975-08-20 1981-04-30 Ciba Geigy Ag
IE45158B1 (en) * 1976-08-16 1982-06-30 Lilly Co Eli 3-chloro-cephem synthesis
PH17188A (en) * 1977-03-14 1984-06-14 Fujisawa Pharmaceutical Co New cephem and cepham compounds and their pharmaceutical compositions and method of use
JPS62112053U (en) * 1985-12-27 1987-07-16
JPH0676861B2 (en) * 1988-05-24 1994-09-28 リンナイ株式会社 Control device for hot air heater
IT1255458B (en) * 1992-05-11 1995-11-02 Col Marco Da PROCEDURE FOR THE PREPARATION OF HALOGENATED BETA-LACTAMIC DERIVATIVES

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2265798C2 (en) * 1971-06-24 1985-09-26 Fujisawa Pharmaceutical Co., Ltd., Osaka Process for the preparation of oxoazetidine derivatives

Also Published As

Publication number Publication date
PL88714B1 (en) 1976-09-30
JPS56138193A (en) 1981-10-28
NL181010C (en) 1987-06-01
FR2218878B1 (en) 1977-03-11
CA1032532A (en) 1978-06-06
GB1458293A (en) 1976-12-15
HU167749B (en) 1975-12-25
NO148376C (en) 1983-09-28
MW574A1 (en) 1975-05-13
YU46374A (en) 1982-06-18
AR201709A1 (en) 1975-04-08
JPS613356B2 (en) 1986-01-31
CY1042A (en) 1980-08-01
JPS56138194A (en) 1981-10-28
FR2218878A1 (en) 1974-09-20
ATA142474A (en) 1976-04-15
MY8100023A (en) 1981-12-31
BG22404A3 (en) 1977-02-20
IE38916B1 (en) 1978-06-21
ZM3674A1 (en) 1975-11-21
HK19980A (en) 1980-04-25
BR7401385D0 (en) 1974-11-05
IE38916L (en) 1974-08-23
IL44263A (en) 1977-10-31
NL7402486A (en) 1974-08-27
DE2408686C2 (en) 1986-08-28
JPS613357B2 (en) 1986-01-31
CS189625B2 (en) 1979-04-30
JPS56138195A (en) 1981-10-28
AU6591574A (en) 1975-08-28
FI63240C (en) 1983-05-10
NO148376B (en) 1983-06-20
AR200908A1 (en) 1974-12-27
CH594686A5 (en) 1978-01-31
OA04688A (en) 1980-07-31
RO64595A (en) 1981-01-30
ES423532A1 (en) 1976-06-01
DE2408686A1 (en) 1974-09-05
JPS49116095A (en) 1974-11-06
IL44263A0 (en) 1974-05-16
YU36971B (en) 1984-08-31
FI63240B (en) 1983-01-31
AT333952B (en) 1976-12-27
GT197432132A (en) 1975-08-16
YU99880A (en) 1983-04-27
SE411211B (en) 1979-12-10
JPS612677B2 (en) 1986-01-27
DD110277A5 (en) 1974-12-12
BE811494A (en) 1974-08-22
PH14014A (en) 1980-12-08
NO740607L (en) 1974-08-26
NO792609L (en) 1974-08-26
YU37347B (en) 1984-08-31
ZA741190B (en) 1975-09-24
KE3026A (en) 1980-03-14
NL181010B (en) 1987-01-02
JPS613358B2 (en) 1986-01-31

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