AR202224A1 - Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas - Google Patents

Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas

Info

Publication number
AR202224A1
AR202224A1 AR254832A AR25483274A AR202224A1 AR 202224 A1 AR202224 A1 AR 202224A1 AR 254832 A AR254832 A AR 254832A AR 25483274 A AR25483274 A AR 25483274A AR 202224 A1 AR202224 A1 AR 202224A1
Authority
AR
Argentina
Prior art keywords
onas
benzodiazepin
procedure
obtaining
Prior art date
Application number
AR254832A
Other languages
English (en)
Spanish (es)
Original Assignee
Crc Ricerca Chim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Crc Ricerca Chim filed Critical Crc Ricerca Chim
Application granted granted Critical
Publication of AR202224A1 publication Critical patent/AR202224A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/28Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AR254832A 1973-07-30 1974-07-22 Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas AR202224A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1105673A CH573928A5 (no) 1973-07-30 1973-07-30

Publications (1)

Publication Number Publication Date
AR202224A1 true AR202224A1 (es) 1975-05-23

Family

ID=4369623

Family Applications (1)

Application Number Title Priority Date Filing Date
AR254832A AR202224A1 (es) 1973-07-30 1974-07-22 Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas

Country Status (21)

Country Link
US (1) US4010153A (no)
JP (1) JPS5041886A (no)
AR (1) AR202224A1 (no)
AT (1) AT337192B (no)
BE (1) BE818047A (no)
CA (1) CA1021778A (no)
CH (1) CH573928A5 (no)
DE (1) DE2436744A1 (no)
DK (1) DK138798B (no)
ES (1) ES428675A1 (no)
FI (1) FI227474A (no)
FR (1) FR2239464B1 (no)
GB (1) GB1481219A (no)
HU (1) HU169180B (no)
IE (1) IE39904B1 (no)
IL (1) IL45289A (no)
NL (1) NL7410256A (no)
NO (1) NO137897C (no)
SE (2) SE7409708L (no)
SU (1) SU528872A3 (no)
ZA (1) ZA744635B (no)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1332410C (en) * 1984-06-26 1994-10-11 Roger M. Freidinger Benzodiazepine analogs
US4820834A (en) * 1984-06-26 1989-04-11 Merck & Co., Inc. Benzodiazepine analogs
LT3324977T (lt) 2015-07-22 2022-10-25 Enanta Pharmaceuticals, Inc. Benzodiazepino dariniai kaip rsv inhibitoriai
US20170226129A1 (en) 2016-01-15 2017-08-10 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
CA3065368A1 (en) 2017-02-16 2018-08-23 Enanta Pharmaceuticals, Inc. Processes for the preparation of benzodiazepine derivatives
WO2018226801A1 (en) 2017-06-07 2018-12-13 Enanta Pharmaceuticals, Inc. Aryldiazepine derivatives as rsv inhibitors
WO2019006295A1 (en) 2017-06-30 2019-01-03 Enanta Pharmaceuticals, Inc. HETEROCYCLIC COMPOUNDS AS RSV INHIBITORS
US10851115B2 (en) 2017-06-30 2020-12-01 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
BR112020006334A2 (pt) 2017-09-29 2020-09-24 Enanta Pharmaceuticals, Inc. combinação de agentes farmacêuticos como inibidores de rsv
WO2019094920A1 (en) 2017-11-13 2019-05-16 Enanta Pharmaceuticals, Inc. Azepin-2-one derivatives as rsv inhibitors
CA3080138A1 (en) * 2017-11-13 2019-05-16 Enanta Pharmaceuticals, Inc. Processes for the resolution of benzodiazepin-2-one and benzoazepin-2-one derivatives
WO2019199908A1 (en) 2018-04-11 2019-10-17 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as rsv inhibitors
UY38614A (es) 2019-03-18 2020-10-30 Enanta Pharm Inc Derivados de benzodiazepinas como inhibidores del rsv
US11179400B2 (en) 2019-04-09 2021-11-23 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as RSV inhibitors
US11505558B1 (en) 2019-10-04 2022-11-22 Enanta Pharmaceuticals, Inc. Antiviral heterocyclic compounds
UY39032A (es) 2020-01-24 2021-07-30 Enanta Pharm Inc Compuestos heterocíclicos como agentes antivirales
WO2022010882A1 (en) 2020-07-07 2022-01-13 Enanta Pharmaceuticals, Inc, Dihydroquinoxaline and dihydropyridopyrazine derivatives as rsv inhibitors
US11945824B2 (en) 2020-10-19 2024-04-02 Enanta Pharmaceuticals, Inc. Heterocyclic compounds as anti-viral agents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3371085A (en) * 1959-12-10 1968-02-27 Hoffmann La Roche 5-aryl-3h-1,4-benzodiazepin-2(1h)-ones
JPS4426302Y1 (no) * 1966-04-22 1969-11-05

Also Published As

Publication number Publication date
FR2239464A1 (no) 1975-02-28
DK138798B (da) 1978-10-30
AT337192B (de) 1977-06-10
IE39904L (en) 1975-01-30
SE7409708L (no) 1975-01-31
SE7510823L (sv) 1975-09-26
ES428675A1 (es) 1976-09-01
IL45289A0 (en) 1974-10-22
IL45289A (en) 1979-12-30
ZA744635B (en) 1975-08-27
CA1021778A (en) 1977-11-29
FR2239464B1 (no) 1978-04-14
CH573928A5 (no) 1976-03-31
DK138798C (no) 1979-04-09
US4010153A (en) 1977-03-01
GB1481219A (en) 1977-07-27
DK393274A (no) 1975-04-01
DE2436744A1 (de) 1975-02-27
JPS5041886A (no) 1975-04-16
NL7410256A (nl) 1975-02-03
NO137897C (no) 1978-05-16
BE818047A (fr) 1974-11-18
HU169180B (no) 1976-10-28
NO742739L (no) 1975-02-24
FI227474A (no) 1975-01-31
ATA567674A (de) 1976-10-15
IE39904B1 (en) 1979-01-31
SU528872A3 (ru) 1976-09-15
NO137897B (no) 1978-02-06

Similar Documents

Publication Publication Date Title
AR213262A1 (es) Procedimiento para la produccion de derivados de 1,1-diaminoetileno
AR208527A1 (es) Procedimiento para la preparacion de 2-acil-4-oxo-polihidro-pirazino(2,1-a)isoquinolinas
AR205249A1 (es) Procedimiento para la sintesis de 1,2 - benzo - tiazin - 3 - carboxamidas
AR210988A1 (es) Procedimiento para la produccion de derivados de 4,6-didesoxi-4-aminoglucopirano.
AR202224A1 (es) Procedimiento para la obtencion de 1,4-benzodiacepin-2-onas
AR198599A1 (es) Procedimiento para la obtencion de formaldehido
AR204926A1 (es) Procedimiento para la preparacion de 2,2,6,6-tetrametil-4-oxopiperidina
AR209263A1 (es) Un procedimiento para la preparacion de 13, 14- dihidro-prostaglandinas
AR203451A1 (es) Procedimiento para la obtencion de nuevas 1,4,5,6,-tetrahidro-piridinas 3-sustituidas
AR202653A1 (es) Preparacion de 2,2,6,6-tetrametil-4-oxopiperidina
AR195391A1 (es) Procedimiento para la preparacion de aldehido 3,4,5-triometoxibenzoico
AR208393A1 (es) Procedimiento para la preparacion de 2,2,6,6-tetrametil-4-oxopiperidina
NO740320L (no) Fremgangsmåte for fremstilling 6-deoksyoksytetracyklin.
AR203653A1 (es) Procedimiento para la obtencion de derivados de 3,4-dihidro-2h-naftalinona-(1)-5-oxi-propil-piperazina
AR208885A1 (es) Procedimiento mejorado para preparar compuestos de 2-amino-5-alquil-1,3,4-tiadiazol
AR197206A1 (es) Procedimiento para preparar 6,7-substituido-quinazolinonas
AR200162A1 (es) Procedimiento para la preparacion de derivados 1,2,4-triazolicos
AR196846A1 (es) Procedimiento para la produccion de compuestos de quinazonalina 2-4diamino-6-sustituidos (0 5,6-disustituidos
AR198586A1 (es) Procedimiento para la produccion de 5-nitro-naftoquinona-(1,4)
AR205800A1 (es) Procedimiento para la preparacion de nuevos derivados de 3,4-difenil-imidazolina
AR202506A1 (es) Procedimiento para la sintesis de 2,6-dehidroxicineol
AR203358A1 (es) Procedimiento para la produccion de nuevas n'-alcilamino-fenil-n,n-dimetilacetamidinas
AR205722A1 (es) Procedimiento para la preparacion de derivados de 17a - substituidos - d - homo - 4 - pregnen - 3,20 - diona
AR213411A1 (es) Procedimiento para la preparacion de 2,6-metano-benzazocinas
AR199146A1 (es) Procedimiento para la obtencion de 16-0-alquil derivados de digitoxosidos de gitoxigenina