AR126766A1 - Método para tratar endometriosis y proporcionar una anticoncepción eficaz - Google Patents
Método para tratar endometriosis y proporcionar una anticoncepción eficazInfo
- Publication number
- AR126766A1 AR126766A1 ARP220102164A ARP220102164A AR126766A1 AR 126766 A1 AR126766 A1 AR 126766A1 AR P220102164 A ARP220102164 A AR P220102164A AR P220102164 A ARP220102164 A AR P220102164A AR 126766 A1 AR126766 A1 AR 126766A1
- Authority
- AR
- Argentina
- Prior art keywords
- drospirenone
- provide effective
- effective contraception
- endometriosis
- treat endometriosis
- Prior art date
Links
- 201000009273 Endometriosis Diseases 0.000 title abstract 3
- METQSPRSQINEEU-UHFFFAOYSA-N dihydrospirorenone Natural products CC12CCC(C3(CCC(=O)C=C3C3CC33)C)C3C1C1CC1C21CCC(=O)O1 METQSPRSQINEEU-UHFFFAOYSA-N 0.000 abstract 4
- METQSPRSQINEEU-HXCATZOESA-N drospirenone Chemical compound C([C@]12[C@H]3C[C@H]3[C@H]3[C@H]4[C@@H]([C@]5(CCC(=O)C=C5[C@@H]5C[C@@H]54)C)CC[C@@]31C)CC(=O)O2 METQSPRSQINEEU-HXCATZOESA-N 0.000 abstract 4
- 229960004845 drospirenone Drugs 0.000 abstract 4
- 230000002051 biphasic effect Effects 0.000 abstract 3
- 201000000736 Amenorrhea Diseases 0.000 abstract 1
- 206010001928 Amenorrhoea Diseases 0.000 abstract 1
- 208000005171 Dysmenorrhea Diseases 0.000 abstract 1
- 206010013935 Dysmenorrhoea Diseases 0.000 abstract 1
- 208000000450 Pelvic Pain Diseases 0.000 abstract 1
- 231100000540 amenorrhea Toxicity 0.000 abstract 1
- 239000003433 contraceptive agent Substances 0.000 abstract 1
- 230000002254 contraceptive effect Effects 0.000 abstract 1
- 230000001939 inductive effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pregnancy & Childbirth (AREA)
Abstract
La presente invención se refiere a drospirenona para su uso en un método para tratar endometriosis, dolor pélvico asociado a endometriosis (DPAE) y/o dismenorrea, que comprende administrar drospirenona en un régimen bifásico. La presente invención se refiere además al uso de drospirenona administrada en un régimen bifásico de este tipo como anticonceptivo y para inducir amenorrea, así como a una composición farmacéutica y a un kit que comprende drospirenona administrada en un régimen bifásico de este tipo.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP21382757.9A EP4134082A1 (en) | 2021-08-12 | 2021-08-12 | Method for treating endometriosis and providing effective contraception |
Publications (1)
Publication Number | Publication Date |
---|---|
AR126766A1 true AR126766A1 (es) | 2023-11-08 |
Family
ID=77358188
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP220102164A AR126766A1 (es) | 2021-08-12 | 2022-08-11 | Método para tratar endometriosis y proporcionar una anticoncepción eficaz |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP4134082A1 (es) |
KR (1) | KR20240047421A (es) |
CN (1) | CN118076358A (es) |
AR (1) | AR126766A1 (es) |
AU (1) | AU2022327756A1 (es) |
CA (1) | CA3228483A1 (es) |
CO (1) | CO2024001947A2 (es) |
IL (1) | IL310634A (es) |
PE (1) | PE20240811A1 (es) |
TW (1) | TW202320801A (es) |
WO (1) | WO2023017109A1 (es) |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2652761C2 (de) | 1976-11-16 | 1985-11-21 | Schering AG, 1000 Berlin und 4709 Bergkamen | 15,16-Methylen-Spirolactone, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel |
DE19633685C1 (de) | 1996-08-12 | 1997-10-09 | Schering Ag | Verfahren zur Herstellung von Drospirenon (6beta,7beta;15 beta,16beta-Dimethyl-en-3-oxo-17alpha-pregn-4-en-21,17-carbolacton, DRSP) sowie 7alpha-(3-Hydroxy-1-propyl)-6beta,7beta;15beta, 16beta-dimethylen-5beta-androstan-3beta,5,17beta-triol (ZK 92836) und 6beta,7beta;15beta,16beta-dimethylen-5beta-hydroxy-3-oxo-17alpha-androstan-21,17-carbolacton (90965) als Zwischenprodukte des Verfahrens |
ITMI20042338A1 (it) | 2004-12-06 | 2005-03-06 | Ind Chimica Srl | Processo per la preparazione di drospirenone |
US10849857B2 (en) * | 2010-07-28 | 2020-12-01 | Laboratorios Leon Farma Sa | Pharmaceutical compositions comprising active drugs, contraceptive kits comprising active drugs, and methods of administering the same |
AR081670A1 (es) | 2010-06-29 | 2012-10-10 | Leon Farma Sa Lab | Composicion farmaceutica que comprende drospirenona y kit anticonceptivo |
ES2970532T3 (es) | 2015-06-23 | 2024-05-29 | Laboratorios Leon Farma Sa | Anticonceptivo basado en drospirenona para una paciente que presenta exceso de peso |
KR20220144885A (ko) * | 2016-08-05 | 2022-10-27 | 에스테트라, 소시에떼 아 레스폰서빌리떼 리미떼 | 월경통 및 생리통의 관리방법 |
JP2018083806A (ja) * | 2016-11-11 | 2018-05-31 | 持田製薬株式会社 | 月経困難症治療用組成物 |
-
2021
- 2021-08-12 EP EP21382757.9A patent/EP4134082A1/en not_active Withdrawn
-
2022
- 2022-08-11 AR ARP220102164A patent/AR126766A1/es unknown
- 2022-08-11 CN CN202280066560.XA patent/CN118076358A/zh active Pending
- 2022-08-11 CA CA3228483A patent/CA3228483A1/en active Pending
- 2022-08-11 PE PE2024000240A patent/PE20240811A1/es unknown
- 2022-08-11 WO PCT/EP2022/072511 patent/WO2023017109A1/en active Application Filing
- 2022-08-11 AU AU2022327756A patent/AU2022327756A1/en active Pending
- 2022-08-11 IL IL310634A patent/IL310634A/en unknown
- 2022-08-11 TW TW111130168A patent/TW202320801A/zh unknown
- 2022-08-11 KR KR1020247008289A patent/KR20240047421A/ko unknown
-
2024
- 2024-02-22 CO CONC2024/0001947A patent/CO2024001947A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
AU2022327756A1 (en) | 2024-03-14 |
IL310634A (en) | 2024-04-01 |
KR20240047421A (ko) | 2024-04-12 |
CO2024001947A2 (es) | 2024-03-07 |
CN118076358A (zh) | 2024-05-24 |
TW202320801A (zh) | 2023-06-01 |
EP4134082A1 (en) | 2023-02-15 |
WO2023017109A1 (en) | 2023-02-16 |
PE20240811A1 (es) | 2024-04-18 |
CA3228483A1 (en) | 2024-02-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PE20190739A1 (es) | Procedimiento de tratamiento de dismenorrea y dolor menstrual | |
AR057060A1 (es) | Composiciones de tanaproget que contienen etinil estradiol | |
CO2021000174A2 (es) | Composiciones tópicas para el alivio del dolor | |
EA200600964A1 (ru) | Фармацевтический препарат для непрерывного гормонального лечения в течение периода времени более длительного, чем 21-28 дней, включающий две композиции эстрогена и/или прогестина | |
AR082998A1 (es) | Asociacion farmaceutica para tratar y/o prevenir mioma y/o endometriosis, uso de resveratrol y progestogeno, composicion farmaceutica para tratamiento y/o prevencion de mioma y/o endometriosis, medicamento para tratamiento y/o prevencion de mioma y/o endometriosis, kit y metodo para tratamiento y/o prevencion de mioma y/o endometriosis | |
PE20211588A1 (es) | Compuestos y sus usos para aliviar sintomas asociados a la menopausia | |
MA26843A1 (fr) | NOUVELLES COMPOSITIONS ESTRO-PROGESTATIVES TOPIQUES à EFFET SYSTÉMIQUE | |
EA200700500A1 (ru) | Совокупность лекарственных форм и способ её введения | |
BRPI0416700A (pt) | métodos para tratar obesidade, para alcançar perda de peso desejável, para evitar ganho de peso indesejável, e para facilitar a perda de peso em um indivìduo não sofrendo de depressão, métodos de manutenção de um peso estável e de redução do peso corporal em um indivìduo, composição farmacêutica, e, kit | |
CA2468748A1 (en) | Oral contraceptives to prevent pregnancy and diminish premenstrual symptomatology | |
PE20040068A1 (es) | Decanoato, undecanoato y dodecanoato de etonogestrel | |
EE05259B1 (et) | Antiprogestiinide kasutamine hormoons?ltuvate haiguste proflaktikaks ja raviks | |
UY38067A (es) | Péptidos de la cadena b de la relaxina modificados y su uso terapéutico | |
AR126766A1 (es) | Método para tratar endometriosis y proporcionar una anticoncepción eficaz | |
CR8010A (es) | Regimenes de contraceptivos transdermicos extendidos | |
BRPI0808599A2 (pt) | "ácido nucléico, vacina, composição farmacêutica, uso de um ácido nucléico e método para estimular uma imunoresposta versus um epítopo das células t" | |
AR120976A1 (es) | Sistema para proporcionar un control de la natalidad | |
ES2211996T3 (es) | Agentes de union a receptores de acido hialuronico y su uso para el tratamiento de tumores o de reestenosis. | |
HRP20090256T1 (en) | Use of estradiolvalerate and dienogest for oral treatment of dysfunctional uterine bleeding in a contraceptive method | |
BR112022014529A2 (pt) | Absorção celular | |
BR112023003317A2 (pt) | Composições e métodos para o tratamento da colangite biliar primária | |
BR112022012081A2 (pt) | Método para tratar câncer, kit, e, uso de uma combinação terapêutica | |
BR112022007168A2 (pt) | Método para tratar câncer, kit, conjugado de anticorpo-fármaco, usos de um conjugado de anticorpo-fármaco e de um agente à base de platina, e, agente à base de platina | |
EP4151210A3 (en) | Pyridine-carboline derivatives as mchr1 antagonists for use in therapy | |
CN108721406A (zh) | 一种治疗急性扭挫伤的外用敷剂及其制备方法 |