AR113107A1 - Formulación de uso tópico para el control y la prevención de parásitos en animales - Google Patents

Formulación de uso tópico para el control y la prevención de parásitos en animales

Info

Publication number
AR113107A1
AR113107A1 ARP180102538A ARP180102538A AR113107A1 AR 113107 A1 AR113107 A1 AR 113107A1 AR P180102538 A ARP180102538 A AR P180102538A AR P180102538 A ARP180102538 A AR P180102538A AR 113107 A1 AR113107 A1 AR 113107A1
Authority
AR
Argentina
Prior art keywords
trifluoromethyl
chloro
phenyl
ethyl
tetrafluoro
Prior art date
Application number
ARP180102538A
Other languages
English (en)
Inventor
Barthel Franziska Dr
Petra Ohage-Spitzlei
Wolfgang Wiehl Dr
Original Assignee
Bayer Animal Health Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Animal Health Gmbh filed Critical Bayer Animal Health Gmbh
Publication of AR113107A1 publication Critical patent/AR113107A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N59/00—Biocides, pest repellants or attractants, or plant growth regulators containing elements or inorganic compounds
    • A01N59/26—Phosphorus; Compounds thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Reivindicación 1: Una formulación líquida que contiene un principio activo que contiene flúor eficaz contra parásitos y fosfato de trietilo. Reivindicación 5: Una formulación líquida de acuerdo con la reivindicación 1, en el que el principio activo fluorado se selecciona del grupo: 2-cloro-N-ciclopropilo-5-[1-[4-(1,1,1,2,3,3,3-heptafluoropropan-2-ilo)-2-metil-6-(trifluorometil)fenil]-1H-pirazol-4-ilo]benzamida, 2-cloro-N-(1-cianociclopropil)-5-[1-[4-(1,1,1,2,3,3,3-heptafluoropropan-2-ilo)-2-metil-6-(trifluorometil)fenil]-1H-pirazol-4-ilo]benzamida, 2-cloro-N-ciclopropilo-5-[4-[2,6-dimetil-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]-fenil]pirazol-1-ilo]benzamida, 2-cloro-N-(1-cianociclopropil)-5-[4-[2,6-dicloro-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]fenil]pirazol-1-ilo]benzamida, 2-cloro-5-[3-[2-cloro-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]-6-(trifluorometil)fenil]isoxazol-5-ilo]-N-ciclopropilbenzamida, 2-cloro-N-(1-cianociclopropil)-5-[3-[2-metil-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]-6-(trifluorometil)fenil]isoxazol-5-ilo]benzamida, 2-cloro-N-(1-cianociclopropil)-5-[1-[2,6-dicloro-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]fenil]pirrol-3-ilo]benzamida, 2-cloro-5-[3-[2-cloro-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]-6-(trifluorometil)fenil]pirrol-1-ilo]-N-ciclopropilbenzamida, 2-cloro-5-[1-[2-cloro-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]-6-(trifluorometoxi)fenil]-1H-pirazol-4-ilo]-N-ciclopropilo-3-piridincarboxamida (compuesto 1), 2-cloro-5-[1-[2-cloro-4-[1,2,2,2-tetrafluoro-1-(trifluorometil)etil]-6-(trifluorometil)fenil]-1H-pirazol-4-ilo]-N-ciclopropilo-3-piridincarboxamida (compuesto 2), tigolaner, fluralaner, afoxolaner (WO2009126668), sarolaner, lotilaner, fluxametamide, pyriprole, fipronil.
ARP180102538A 2017-09-06 2018-09-06 Formulación de uso tópico para el control y la prevención de parásitos en animales AR113107A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP17189706 2017-09-06

Publications (1)

Publication Number Publication Date
AR113107A1 true AR113107A1 (es) 2020-01-29

Family

ID=59811131

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP180102538A AR113107A1 (es) 2017-09-06 2018-09-06 Formulación de uso tópico para el control y la prevención de parásitos en animales

Country Status (22)

Country Link
US (1) US11344532B2 (es)
EP (1) EP3651579A1 (es)
JP (1) JP7305620B2 (es)
KR (1) KR20200044099A (es)
CN (1) CN111050557B (es)
AR (1) AR113107A1 (es)
AU (1) AU2018329158A1 (es)
BR (1) BR112020004339A2 (es)
CA (1) CA3074620A1 (es)
CL (1) CL2020000551A1 (es)
CO (1) CO2020002624A2 (es)
CR (1) CR20200105A (es)
DO (1) DOP2020000052A (es)
IL (1) IL272720A (es)
MX (1) MX2020002496A (es)
MY (1) MY202302A (es)
PH (1) PH12020500431A1 (es)
SG (1) SG11202001304XA (es)
TW (2) TWI794282B (es)
UA (1) UA127622C2 (es)
UY (1) UY37867A (es)
WO (1) WO2019048381A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112022002623A2 (pt) * 2019-08-14 2022-05-03 Vetoquinol Sa Composição, composição compreendendo praziquantel, emodepsida e um componente solvente, método para produzir uma composição e composição para uso
AU2021214719A1 (en) * 2020-01-29 2022-08-25 Elanco Animal Health Gmbh Pharmaceutical composition for controlling parasites on non-human organisms

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4443888A1 (de) 1994-12-09 1996-06-13 Bayer Ag Dermal applizierbare Formulierungen von Parasitiziden
JPH08291004A (ja) * 1995-04-24 1996-11-05 Nippon Kayaku Co Ltd 害虫防除剤組成物
SE517612C2 (sv) 1995-12-20 2002-06-25 Rhone Poulenc Agrochimie Användning av 5-amino-4-etylsulfinyl-1-arylpyrazol föreningar som pesticider
DE10117676A1 (de) 2001-04-09 2002-10-10 Bayer Ag Dermal applizierbare flüssige Formulierungen zur Bekämpfung von parasitierenden Insekten an Tieren
DE10320505A1 (de) 2003-05-08 2004-11-25 Bayer Healthcare Ag Mittel zum Bekämpfen von Parasiten an Tieren
CN1225978C (zh) * 2003-11-03 2005-11-09 浙江新农化工有限公司 含三唑磷和氟虫腈复配杀虫微乳剂及其制备方法
DK1731512T3 (en) 2004-03-05 2015-01-05 Nissan Chemical Ind Ltd Isoxazoline-substituted benzamide AND INSTRUMENTS FOR COMBATING HARMFUL ORGANISMS
EP2072501A1 (en) 2007-12-21 2009-06-24 Bayer CropScience AG Aminobenzamide derivatives as useful agents for controlling animal parasites
TWI518076B (zh) 2008-04-09 2016-01-21 杜邦股份有限公司 製備雜環化合物之方法
ES2395704T3 (es) 2008-12-19 2013-02-14 Novartis Ag Derivados de isoxazolina y su uso como pesticida
NZ601203A (en) * 2010-01-29 2015-01-30 Mitsui Chemicals Agro Inc Composition for exterminating animal parasite and method for exterminating animal parasite
SI2683723T1 (sl) 2011-03-10 2016-07-29 Zoetis Services Llc Spirociklični izoksazolinski derivati kot antiparazitiki
CA2900029C (en) 2013-02-06 2021-03-02 Bayer Cropscience Aktiengesellschaft Halogen-substituted pyrazol derivatives as pest-control agents
SI3066079T1 (sl) 2013-11-05 2018-09-28 Bayer Cropscience Ag Nove spojine za boj proti členonožcem
JP6740239B2 (ja) 2015-03-12 2020-08-12 エフ エム シー コーポレーションＦｍｃ Ｃｏｒｐｏｒａｔｉｏｎ 複素環置換二環式アゾール殺有害生物剤
UY36910A (es) 2015-09-23 2017-04-28 Syngenta Participations Ag Benzamidas de bis isoxazolinas como compuestos insecticidas

Also Published As

Publication number Publication date
IL272720A (en) 2020-04-30
CN111050557A (zh) 2020-04-21
TW201919584A (zh) 2019-06-01
EP3651579A1 (en) 2020-05-20
BR112020004339A2 (pt) 2020-09-08
TWI794282B (zh) 2023-03-01
CR20200105A (es) 2020-04-22
TW202335661A (zh) 2023-09-16
MX2020002496A (es) 2020-07-20
US11344532B2 (en) 2022-05-31
UA127622C2 (uk) 2023-11-08
CL2020000551A1 (es) 2020-11-06
RU2020112629A (ru) 2021-10-06
WO2019048381A1 (en) 2019-03-14
CN111050557B (zh) 2023-08-01
UY37867A (es) 2019-03-29
MY202302A (en) 2024-04-23
PH12020500431A1 (en) 2020-11-09
AU2018329158A8 (en) 2020-03-12
JP2020532563A (ja) 2020-11-12
RU2020112629A3 (es) 2021-12-28
US20210059986A1 (en) 2021-03-04
AU2018329158A1 (en) 2020-03-05
DOP2020000052A (es) 2020-08-16
JP7305620B2 (ja) 2023-07-10
CA3074620A1 (en) 2019-03-14
CO2020002624A2 (es) 2020-04-13
KR20200044099A (ko) 2020-04-28
SG11202001304XA (en) 2020-03-30

Similar Documents

Publication Publication Date Title
CO2017000689A2 (es) Composición insecticida, acaricida, nematicida, molusquicida, microbicida, o bactericida y método para controlar plagas
AR113107A1 (es) Formulación de uso tópico para el control y la prevención de parásitos en animales
EA201992550A1 (ru) Фунгицидные смеси, содержащие замещенные 3-фенил-5-(трифторметил)-1,2,4-оксадиазолы
PE20191005A1 (es) 1,2,4-triazolonas 2,4,5-trisustituidas
NZ592224A (en) Acrylamido derivatives useful as inhibitors of the mitochondrial permeability transition
RU2470920C2 (ru) Фторосодержащее сераорганическое соединение и содержащая его пестицидная композиция
PE20220253A1 (es) Benzamidas sustituidas con 1,3-tiazol-2-ilo
JP2016528201A5 (es)
AR104735A1 (es) Terapia combinada de un anticuerpo anti-cd20 con un inhibidor de bcl-2 y un inhibidor de mdm2, método de tratamiento, uso
PE20140837A1 (es) Compuestos fungicidas 2-[2-cloro-4-(4-cloro-fenoxi)-fenil]-1-[1,2,4]triazol-1-il-etanol alquilo sustituidos
PE20210928A1 (es) Mezclas pesticidas que comprenden indazoles
NZ719975A (en) Active compound combinations comprising a (thio)carboxamide derivative and a fungicidal compound
MX2022000708A (es) Formulaciones orales de inhibidores de sarcomeros cardiacos.
CL2009000578A1 (es) Formulacion herbicida sinergica que comprende piroxasulfona y pendimetalin; uso y metodo que la emplea para controlar vegetacion indeseada.
AR102987A1 (es) Combinaciones de compuestos activos que comprenden un derivado de (tio)carboxamida y compuesto(s) fungicida(s)
PE20191792A1 (es) Derivados de isoxazol como agonistas del receptor nuclear y usos de los mismos
EA202191833A1 (ru) Композиции и способы применения 2-(4-хлорфенил)-n-((2-(2,6-диоксопиперидин-3-ил)-1-оксоизоиндолин-5-ил)метил)-2,2-дифторацетамида
BR112017009282A2 (pt) misturas fungicidas, composição pesticida, métodos para controlar pragas fitopatogênicas, para melhorar a fitossanidade e para proteção de material de propagação de plantas contra pragas, e, material de propagação de plantas.
BR112021023074A2 (pt) Tratamento de disfunção sistólica e insuficiência cardíaca com fração de ejeção reduzida com o composto (r)-4-(l-(1-((3-(difluorometil)-l--1-metil-1h-pirazol-4-il)sulfonil)-l-1-fluoroetil)-n-(isoxazol-3-il)piperidina-l-1-carboxamida
ZA202101186B (en) A stable liquid agrochemical formulation
UY36964A (es) Combinaciones de principios activos que comprenden un derivado de (tio) carboxamida y un compuesto funguicida
AR105952A1 (es) Composiciones herbicidas que comprenden n-(tetrazol-5-il)-on-(1,3,4-oxadiazol-2-il)arilamidas y un derivado de 3-isoxazolidinona
JP2018516873A5 (es)
EA202092018A1 (ru) Фунгицидные композиции мефентрифлуконазола
EA201890207A1 (ru) Термодинамически стабильная кристаллическая модификация 2-хлор-3-(метилсульфанил)-n-(1-метил-1h-тетразол-5-ил)-4-(трифторметил)бензамида