AR083251A1 - Imidazoles fungicidas - Google Patents

Imidazoles fungicidas

Info

Publication number
AR083251A1
AR083251A1 ARP110103612A ARP110103612A AR083251A1 AR 083251 A1 AR083251 A1 AR 083251A1 AR P110103612 A ARP110103612 A AR P110103612A AR P110103612 A ARP110103612 A AR P110103612A AR 083251 A1 AR083251 A1 AR 083251A1
Authority
AR
Argentina
Prior art keywords
independently
alkoxy
ring
alkyl
haloalkyl
Prior art date
Application number
ARP110103612A
Other languages
English (en)
Inventor
Andrew Edmund Taggi
James Francis Bereznak
Tuzhong Chen
Moumita Kar
Jeffrey Keith Long
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Publication of AR083251A1 publication Critical patent/AR083251A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/68—Halogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cultivation Of Plants (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Composiciones que contienen los compuestos de la fórmula (1) y los métodos para controlar las enfermedades de las plantas causadas por un patógeno fúngico; donde el método comprende aplicar una cantidad efectiva de un compuesto o una composición de la solicitud.Reivindicación 1: Un compuesto caracterizado porque se selecciona entre la fórmula (1), N-óxidos y las sales de los mismos, en donde Q1 es un anillo fenilo sustituido con entre 1 y 4 sustituyentes que se seleccionan de forma independiente entre R5a; o un anillo tienilo, pirazolilo, imidazolilo, tiazolilo, piridinilo, piridazinilo o pirimidinilo o un sistema de anillos quinazolinilo, donde cada anillo o sistema de anillos opcionalmente está sustituido con hasta 4 sustituyentes que se seleccionan de forma independiente entre R5a en los miembros del anillo que son átomos de carbono y R5b en los miembros del anillo que son átomos de nitrógeno; Q2 es un anillo fenilo sustituido con entre 1 y 4 sustituyentes que se seleccionan de forma independiente entre R5a; o un anillo tienilo, pirazolilo, imidazolilo, tiazolilo, piridinilo, piridazinilo o pirimidinilo o un sistema de anillos quinazolinilo, donde cada anillo o sistema de anillos opcionalmente está sustituido con hasta 4 sustituyentes que se seleccionan de forma independiente entre R5a en los miembros del anillo que son átomos de carbono y R5b en los miembros del anillo que son átomos de nitrógeno; R1 y R2 son cada uno de forma independiente H, halógeno, ciano, nitro, alquilo C1-3, alquenilo C2-3, alquinilo C2-3, haloalquilo C1-3, haloalquenilo C2-3, ciclopropilo, halociclopropilo, hidroxialquilo C1-3, cianoalquilo C2-3, alcoxialquilo C2-3, alcoxi C1-3, alcoxi C1-3, alquiltio C1-3 o haloalquiltio C1-3; R3 es halógeno, -OR6 o -SCºN; R4 es H o alquilo C1-6; cada R5a es de forma independiente halógeno, ciano, hidroxi, nitro, alquilo C1-3, alquenilo C2-3, alquinilo C2-3, haloalquilo C1-3, haloalquenilo C2-3, ciclopropilo, halociclopropilo, cianoalquilo C2-3, alquiltio C1-3, haloalquiltio C1-3, alquilsulfinilo C1-3, haloalquilsulfinilo C1-3, alquilsulfonilo C1-3, haloalquilsulfonilo C1-3, alcoxi C1-3, alcoxi C1-3, alquilcarboniloxi C2-4, alquilcarbonilo C2-3, alquilamino C1-3, dialquilamino C2-4, alquilcarbonilamino C2-3, trialquilsililo C3-6, -CH(=O), -NHCH(=O), -C(=S)NH2, -SCºN o -T-U-V; cada R5b es de forma independiente ciano, alquilo C1-3, alquenilo C2-3, alquinilo C2-3, haloalquilo C1-3, ciclopropilo, alcoxialquilo C2-3, alquilaminoalquilo C2-3, dialquilaminoalquilo C3-4, alcoxi C1-3, alquilcarbonilo C2-3 o alcoxicarbonilo C2-3; R6 es H, -CH(=O), alquilo C1-6, alquenilo C2-6, alquinilo C3-6, haloalquilo C1-6, cicloalquilo C3-6, halocicloalquilo C3-6, alcoxialquilo C2-6, cianoalquilo C2-6, alquilcarbonilo C2-6, alcoxicarbonilo C2-6, (alquiltio)carbonilo C2-6, cicloalquilcarbonilo C4-8, cicloalcoxicarbonilo C4-8, (cicloalquiltio)carbonilo C4-8, alcoxi C2-6(tiocarbonilo) o cicloalcoxi C4-8(tiocarbonilo); cada T es de forma independiente O, S(=O)n, N(R7) o un enlace directo; cada U es de forma independiente alquileno C2-6, alquenileno C2-6, alquinileno C3-6, cicloalquileno C3-6 o cicloalquenileno C3-6, en donde hasta 3 átomos de carbono se seleccionan de forma independiente de C(=O), cada uno opcionalmente sustituido con hasta 5 sustituyentes que se seleccionan de forma independiente entre halógeno, ciano, nitro, hidroxi, alquilo C1-6, haloalquilo C1-6, alcoxi C1-6 y haloalcoxi C1-6; cada V es de forma independiente ciano, N(R8a)(R8b), OR9 o S(=O)nR9; cada R7 es de forma independiente H, alquilo C1-6, haloalquilo C1-6, alquilcarbonilo C2-6, alcoxicarbonilo C2-6, (alquiltio C2-6)carbonilo, alcoxi C2-6(tiocarbonilo), cicloalquilcarbonilo C4-8, cicloalcoxicarbonilo C4-8, (cicloalquiltio C4-8)carbonilo o cicloalcoxi C4-8(tiocarbonilo); cada R8a y R8b es de forma independiente H, alquilo C1-6, haloalquilo C1-6, alquenilo C2-6, alquinilo C3-6, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcarbonilo C2-6, alcoxicarbonilo C2-6, (alquiltio C2-6)carbonilo, alcoxi C2-6(tiocarbonilo), cicloalquilcarbonilo C4-8, cicloalcoxicarbonilo C4-8, (cicloalquiltio C4-8)carbonilo o cicloalcoxi C4-8(tiocarbonilo); o un par de R8a y R8b se toman junto con el átomo de nitrógeno al cual se unen para formar un anillo heterocíclico de entre 4 y 7 miembros, donde el anillo opcionalmente está sustituido con hasta 5 sustituyentes que se seleccionan de forma independiente entre R10, cada R9 es de forma independiente H, alquilo C1-6, haloalquilo C1-6, alquenilo C2-6, alquinilo C3-6, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcarbonilo C2-6, alcoxicarbonilo C2-6, (alquiltio C2-6)carbonilo, alcoxi C2-6(tiocarbonilo), cicloalquilcarbonilo C4-8, cicloalcoxicarbonilo C4-8, (cicloalquiltio C4-8)carbonilo o cicloalcoxi C4-8(tiocarbonilo); cada R10 es de forma independiente halógeno, alquilo C1-6, haloalquilo C1-6 o alcoxi C1-6; cada n es de forma independiente 0, 1 ó 2; con la condición de que: (a) cuando Q1 y Q2 son ambos fenilos sustituidos con entre 1 y 4 sustituyentes que se seleccionan de forma independiente entre R5a, entonces al menos un sustituyente R5a se une en una posición orto; y (b) cuando R1 es H, entonces R2 es distinto de H.
ARP110103612A 2010-09-29 2011-09-29 Imidazoles fungicidas AR083251A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US38767110P 2010-09-29 2010-09-29

Publications (1)

Publication Number Publication Date
AR083251A1 true AR083251A1 (es) 2013-02-13

Family

ID=44801173

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP110103612A AR083251A1 (es) 2010-09-29 2011-09-29 Imidazoles fungicidas

Country Status (12)

Country Link
US (1) US20130143929A1 (es)
EP (1) EP2621907A1 (es)
JP (1) JP2013541535A (es)
KR (1) KR20130099268A (es)
CN (1) CN103153962A (es)
AR (1) AR083251A1 (es)
AU (1) AU2011307289A1 (es)
BR (1) BR112013007635A2 (es)
MX (1) MX2013003390A (es)
TW (1) TW201216849A (es)
UY (1) UY33635A (es)
WO (1) WO2012044650A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR075713A1 (es) 2009-03-03 2011-04-20 Du Pont Pirazoles fungicidas
US8809372B2 (en) 2011-09-30 2014-08-19 Asana Biosciences, Llc Pyridine derivatives
GB201417962D0 (en) * 2014-10-10 2014-11-26 Redag Crop Prot Ltd Agricultural chemicals
CN112047895B (zh) * 2019-06-06 2024-05-14 东莞市东阳光农药研发有限公司 三唑类化合物及其制备方法和应用
CN112986460A (zh) * 2021-04-15 2021-06-18 秦皇岛海关技术中心 植物源食品中双胍三辛烷基苯磺酸盐残留量的检测方法

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Also Published As

Publication number Publication date
AU2011307289A1 (en) 2013-02-21
US20130143929A1 (en) 2013-06-06
WO2012044650A1 (en) 2012-04-05
KR20130099268A (ko) 2013-09-05
UY33635A (es) 2012-04-30
BR112013007635A2 (pt) 2016-07-26
JP2013541535A (ja) 2013-11-14
MX2013003390A (es) 2013-05-31
TW201216849A (en) 2012-05-01
EP2621907A1 (en) 2013-08-07
CN103153962A (zh) 2013-06-12

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