AR073252A1 - Piridinas fungicidas - Google Patents
Piridinas fungicidasInfo
- Publication number
- AR073252A1 AR073252A1 ARP090102393A ARP090102393A AR073252A1 AR 073252 A1 AR073252 A1 AR 073252A1 AR P090102393 A ARP090102393 A AR P090102393A AR P090102393 A ARP090102393 A AR P090102393A AR 073252 A1 AR073252 A1 AR 073252A1
- Authority
- AR
- Argentina
- Prior art keywords
- ring
- atoms
- alkyl
- alkoxy
- substituents
- Prior art date
Links
- 125000001424 substituent group Chemical group 0.000 abstract 13
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 12
- 125000000217 alkyl group Chemical group 0.000 abstract 7
- 229910052736 halogen Inorganic materials 0.000 abstract 6
- 150000002367 halogens Chemical class 0.000 abstract 6
- 229910052757 nitrogen Inorganic materials 0.000 abstract 6
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 5
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 5
- -1 cyano, hydroxy, amino Chemical group 0.000 abstract 5
- 125000006413 ring segment Chemical group 0.000 abstract 5
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 4
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 4
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 4
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 4
- 125000003545 alkoxy group Chemical group 0.000 abstract 4
- 125000004429 atom Chemical group 0.000 abstract 4
- 125000004432 carbon atom Chemical group C* 0.000 abstract 4
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 4
- 125000000232 haloalkynyl group Chemical group 0.000 abstract 4
- 125000005842 heteroatom Chemical group 0.000 abstract 4
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 4
- 229910052717 sulfur Inorganic materials 0.000 abstract 4
- 239000011593 sulfur Substances 0.000 abstract 4
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 abstract 3
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 abstract 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 3
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 3
- 125000004183 alkoxy alkyl group Chemical group 0.000 abstract 3
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 3
- 125000005119 alkyl cycloalkyl group Chemical group 0.000 abstract 3
- 229910052799 carbon Inorganic materials 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000000000 cycloalkoxy group Chemical group 0.000 abstract 3
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 abstract 3
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 3
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 abstract 3
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 3
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 3
- 229910052760 oxygen Inorganic materials 0.000 abstract 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000004665 trialkylsilyl group Chemical group 0.000 abstract 3
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 abstract 2
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 abstract 2
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 abstract 2
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 abstract 2
- 125000001627 3 membered heterocyclic group Chemical group 0.000 abstract 2
- 125000001963 4 membered heterocyclic group Chemical group 0.000 abstract 2
- 125000002373 5 membered heterocyclic group Chemical group 0.000 abstract 2
- 125000004070 6 membered heterocyclic group Chemical group 0.000 abstract 2
- 125000006577 C1-C6 hydroxyalkyl group Chemical group 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 abstract 2
- 125000005120 alkyl cycloalkyl alkyl group Chemical group 0.000 abstract 2
- 125000004687 alkyl sulfinyl alkyl group Chemical group 0.000 abstract 2
- 125000004688 alkyl sulfonyl alkyl group Chemical group 0.000 abstract 2
- 125000006350 alkyl thio alkyl group Chemical group 0.000 abstract 2
- 125000000304 alkynyl group Chemical group 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 125000004966 cyanoalkyl group Chemical group 0.000 abstract 2
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 2
- 125000001188 haloalkyl group Chemical group 0.000 abstract 2
- 125000004992 haloalkylamino group Chemical group 0.000 abstract 2
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 abstract 2
- 125000006769 halocycloalkoxy group Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 2
- 125000004434 sulfur atom Chemical group 0.000 abstract 2
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 1
- 125000006559 (C1-C3) alkylamino group Chemical group 0.000 abstract 1
- 125000006595 (C1-C3) alkylsulfinyl group Chemical group 0.000 abstract 1
- 125000006594 (C1-C3) alkylsulfony group Chemical group 0.000 abstract 1
- 125000004455 (C1-C3) alkylthio group Chemical group 0.000 abstract 1
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 1
- 125000004845 (C1-C6) alkylsulfonylamino group Chemical group 0.000 abstract 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 1
- 125000006564 (C4-C8) cycloalkyl group Chemical group 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 125000005083 alkoxyalkoxy group Chemical group 0.000 abstract 1
- 125000005078 alkoxycarbonylalkyl group Chemical group 0.000 abstract 1
- 125000003418 alkyl amino alkoxy group Chemical group 0.000 abstract 1
- 125000000278 alkyl amino alkyl group Chemical group 0.000 abstract 1
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 abstract 1
- 125000005130 alkyl carbonyl thio group Chemical group 0.000 abstract 1
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 abstract 1
- 125000006310 cycloalkyl amino group Chemical group 0.000 abstract 1
- 125000006254 cycloalkyl carbonyl group Chemical group 0.000 abstract 1
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 abstract 1
- 125000004985 dialkyl amino alkyl group Chemical group 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 244000053095 fungal pathogen Species 0.000 abstract 1
- 125000005221 halo alkyl carbonyl amino group Chemical group 0.000 abstract 1
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 abstract 1
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 abstract 1
- 125000004664 haloalkylsulfonylamino group Chemical group 0.000 abstract 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/46—Oxygen atoms
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/26—Radicals substituted by halogen atoms or nitro radicals
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/57—Nitriles
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Abstract
Composiciones que contienen los compuestos de formula (1) y métodos para controlar enfermedades de las plantas causadas por un patogeno fungico, que comprenden aplicar una cantidad eficaz de un compuesto o una composicion de la presente. Reivindicacion 1: Un compuesto caracterizado porque se selecciona entre formula (1), N-oxidos y sales del mismo, donde R1 es halogeno, ciano, hidroxi, amino, alquilo C1-4, alquenilo C2-4, alquinilo C2-4, haloalquilo C1-4, haloalquenilo C2-4, haloalquinilo C2-4, ciclopropilo, halociclopropilo, alcoxialquilo C2-4, alquiltioalquilo C2-4, alquilsulfinilalquilo C2-4, alquilsulfonilalquilo C2-4, alquilcarbonilo C2-4, alcoxicarbonilo C2-4, hidroxialquilo C1-3, alcoxi C1-3, haloalcoxi C1-3, alquiltio C1-3, haloalquiltio C1-3, alquilsulfinilo C1-3, haloalquilsulfinilo C1-3, alquilsulfonilo C1-3, haloalquilsulfonilo C1-3, alquilamino C1-3 o dialquilamino C2-4; cada W e Y es independientemente CH2, O, C(=O), S(=O)n, NR8 o una union directa; R2 es un anillo fenilo opcionalmente sustituido con hasta 5 sustituyentes seleccionados independientemente entre R6; o un anillo heterocíclico de 3, 4, 5 o 6 miembros que contiene miembros del anillo seleccionados entre átomos de carbono y hasta 4 heteroátomos seleccionados entre hasta 2 átomos de oxígeno, hasta 2 de azufre y hasta 3 de nitrogeno, donde hasta 3 átomos de carbono miembros del anillo se seleccionan independientemente entre C(=O) y C(=S), y los átomos de azufre miembros del anillo se seleccionan independientemente entre S(=O)p(=NR9)q, el anillo heterocíclico se sustituye opcionalmente con hasta 5 sustituyentes seleccionados independientemente entre R6 sobre átomos de carbono miembros del anillo y R6a sobre átomos de nitrogeno miembros del anillo; R3 es un anillo fenilo opcionalmente sustituido con hasta 5 sustituyentes seleccionados independientemente entre R7; o un anillo heterocíclico de 3, 4, 5 o 6 miembros que contiene miembros del anillo seleccionados entre átomos de carbono y hasta 4 heteroátomos seleccionados entre hasta 2 átomos de oxígeno, hasta 2 de azufre y hasta 3 de nitrogeno, donde hasta 3 átomos de carbono miembros del anillo se seleccionan independientemente entre C(=O) y C(=S), y los átomos de azufre miembros del anillo se seleccionan independientemente entre S(=O)p(=NR9)q, el anillo heterocíclico se sustituye opcionalmente con hasta 5 sustituyentes seleccionados independientemente entre R7 sobre átomos de carbono miembros del anillo y R7a sobre átomos de nitrogeno miembros del anillo; o cuando Y es una union directa, luego R3 también se selecciona entre halogeno, ciano, hidroxi, amino, nitro, -CHO, alquilo C1-6, alquenilo C2-6, alquinilo C2-6, haloalquilo C1-6, haloalquenilo C2-6, haloalquinilo C2-6, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcicloalquilo C4-8, cicloalquilalquilo C4-8, cicloalquilcicloalquilo C6-12, halocicloalquilalquilo C4-8, alquilcicloalquilalquilo C5-8, cicloalquenilo C3-6, alcoxialquilo C2-6, alquiltioalquilo C2-6, alquilsulfinilalquilo C2-6, alquilsulfonilalquilo C2-6, alquilaminoalquilo C2-6, dialquilaminoalquilo C3-6, alquilcarbonilo C2-6, haloalquilcarbonilo C2-6, cicloalquilcarbonilo C4-6, alcoxicarbonilo C2-6, alquilaminocarbonilo C2-6, dialquilaminocarbonilo C3-8, cianoalquilo C2-6, hidroxialquilo C1-6, hidroxihaloalquilo C2-6, hidroxialquilcarbonilo C2-6, hidroxicarbonilalquilo C2-6, alcoxi C1-6, haloalcoxi, C1-6, cicloalcoxi C3-6, halocicloalcoxi C3-6, alcoxialcoxi C2-6, alcoxicarbonilalquilo C3-6, alquiltio C1-6, haloalquiltio C1-6, alquilsulfinilo C1-6, haloalquilsulfinilo C1-6, alquilsulfonilo C1-6, haloalquilsulfonilo C1-6, trialquilsililo C3-9, alquilamino C1-6, dialquilamino C2-6, haloalquilamino C2-6, halodialquilamino C2-6, cicloalquilamino C3-6, alquilcarbonilamino C2-6, haloalquilcarbonilamino C2-6, alquilsulfonilamino C1-6 y haloalquilsulfonilamino C1-6; R4 es H, halogeno, ciano, hidroxi, alquilo C1-2, haloalquilo C1-2, alquenilo C2, haloalquenilo C2 o alquinilo C2; cada R5, R6 y R7 es independientemente halogeno, ciano, hidroxi, amino, nitro, -CHO, alquilo C1-6, alquenilo C2-6, alquinilo C2-6, haloalquilo C1-6, alquilcarbonilo C2-6, haloalquilcarbonilo C2-6, alcoxicarbonilo C2-6, alquilaminocarbonilo C2-6, dialquilaminocarbonilo C3-6, alquilaminoalcoxi C2-6, haloalquenilo C2-6, haloalquinilo C2-6, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcicloalquilo C4-8, cicloalquilalquilo C4-8, alquilcicloalquilalquilo C5-8, alcoxialquilo C2-6, cianoalquilo C2-6, hidroxialquilo C1-6, alcoxi C1-6, haloalcoxi C1-6, cicloalcoxi C3-6, halocicloalcoxi C3-6, alquilcarboniloxi C2-6, alquiltio C1-6, haloalquiltio C1-6, alquilsulfinilo C1-6, haloalquilsulfinilo C1-6, alquilsulfonilo C1-6, haloalquilsulfonilo C1-6, trialquilsililo C3-9, alquilcarboniltio C2-6, alquilamino C1-6 o dialquilamino C2-6; cada R6a y R7a es independientemente ciano, alquilo C1-6, alquenilo C2-6, alquinilo C2-6, haloalquilo C1-6, alquilcarbonilo C2-6, haloalquilcarbonilo C2-6, alcoxicarbonilo C2-6, alquilaminocarbonilo C2-6, dialquilaminocarbonilo C3-6, haloalquenilo C2-6, haloalquinilo C2-6, cicloalquilo C3-6, halocicloalquilo C3-6, alquilcicloalquilo C4-8, cicloalquilalquilo C4-8, alquilcicloalquilalquilo C5-8, alcoxialquilo C2-6, alcoxi C1-6, haloalcoxi C1-6, cicloalcoxi C3-6, halocicloalcoxi C3-6, alquiltio C1-6, haloalquiltio C1-6, alquilsulfonilo C1-6, haloalquilsulfonilo C1-6 o trialquilsililo C3-9; o un par de sustituyentes R5 unidos a átomos del anillo adyacentes, un par de sustituyentes seleccionados entre R6 y R6a sustituyentes unidos a átomos del anillo adyacentes, y un par de sustituyentes seleccionados entre R7 y R7a sustituyentes unidos a átomos del anillo adyacentes pueden cada uno independientemente tomarse junto con los átomos a los cuales se encuentran unidos para formar un anillo fusionado de 5, 6 o 7 miembros, cada anillo fusionado contiene miembros del anillo seleccionados entre carbono y hasta 4 heteroátomos seleccionados entre hasta 2 oxígeno, hasta 2 azufre y hasta 3 nitrogeno, y opcionalmente sustituidos con hasta 3 sustituyentes independientemente seleccionados entre el grupo que consiste en alquilo C1-2, halogeno, ciano, nitro y alcoxi C1-2 sobre carbonos miembros del anillo y a partir del grupo que consiste en alquilo C1-2, ciano y alcoxi C1-2 sobre nitrogenos miembros del anillo; o un par de sustituyentes R6 unidos al mismo átomo del anillo y un par de sustituyentes R7 unidos al mismo átomo del anillo pueden cada uno independientemente tomarse junto con el átomo al cual se encuentran unidos para formar un anillo espirocíclico de 5, 6 o 7 miembros, cada anillo espirocíclico contiene miembros del anillo seleccionados entre carbono, hasta 4 heteroátomos seleccionados entre hasta 2 oxígeno, hasta 2 azufre y hasta 3 nitrogeno, y opcionalmente sustituidos con hasta 3 sustituyentes independientemente seleccionados entre el grupo que consiste en alquilo C1-2, halogeno, ciano, nitro y alcoxi C1-2 sobre carbonos miembros del anillo y a partir del grupo que consiste en alquilo C1-2, ciano y alcoxi C1-2 sobre nitrogenos miembros del anillo; cada R8 y R9 es independientemente H o alquilo C1-3; m es un entero seleccionado entre 0, 1, 2, 3, 4 y 5; cada n es independientemente un entero seleccionado entre 0, 1 y 2; y p y q son independientemente 0, 1 o 2 en cada instancia de S(=O)p(=NR9)q, con la condicion de que la suma de p y q es 0, 1 o 2; con la condicion de que cuando Y es una union directa y R3 es un anillo fenilo sustituido con dos sustituyentes alcoxi unidos en las posiciones meta, luego R4 es H.
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