AR082787A1 - Lactonas macrociclicas y su uso y sus combinaciones con otras sustancias activas - Google Patents
Lactonas macrociclicas y su uso y sus combinaciones con otras sustancias activasInfo
- Publication number
- AR082787A1 AR082787A1 ARP110103139A ARP110103139A AR082787A1 AR 082787 A1 AR082787 A1 AR 082787A1 AR P110103139 A ARP110103139 A AR P110103139A AR P110103139 A ARP110103139 A AR P110103139A AR 082787 A1 AR082787 A1 AR 082787A1
- Authority
- AR
- Argentina
- Prior art keywords
- macrociclic
- lactons
- combinations
- active substances
- filarias
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/12—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
- C07D493/20—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Gastroenterology & Hepatology (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Para controlar filarias endoparásitas y nemátodos gastrointestinales. Se prefiere el uso para controlar el gusano del corazón del perro (Dirofilaria immitis). Se refiere además a derivados de los compuestos de fórmula (1) y (2).Reivindicación 1: Compuestos de fórmula (1) y (2) para controlar filarias endoparasitarias y nemátodos gastrointestinales.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10174655 | 2010-08-31 | ||
DE102010064245A DE102010064245A1 (de) | 2010-12-28 | 2010-12-28 | Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen |
Publications (1)
Publication Number | Publication Date |
---|---|
AR082787A1 true AR082787A1 (es) | 2013-01-09 |
Family
ID=44509397
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP110103139A AR082787A1 (es) | 2010-08-31 | 2011-08-29 | Lactonas macrociclicas y su uso y sus combinaciones con otras sustancias activas |
Country Status (3)
Country | Link |
---|---|
AR (1) | AR082787A1 (es) |
UY (1) | UY33577A (es) |
WO (1) | WO2012028556A1 (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2523284C9 (ru) * | 2012-05-31 | 2014-10-10 | Автономная Некоммерческая Организация "Научно-Исследовательский Центр Биотехнологии Антибиотиков И Других Биологически Активных Веществ "Биоан" | Способ модификации макролидного антибиотика олигомицина а с помощью реакции [3+2]-диполярного циклоприсоединения азида и алкинов. 33-дезокис-33-(триазол-1-ил)-олигомицины а и их биологическая активность |
WO2016139331A1 (en) | 2015-03-05 | 2016-09-09 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods and pharmaceutical compositions for the treatment of melanoma |
SI3298027T1 (sl) | 2015-05-20 | 2021-08-31 | Boehringer Ingelheim Animal Health USA Inc. | Antihelmintične depsipeptidne spojine |
WO2017116702A1 (en) | 2015-12-28 | 2017-07-06 | Merial, Inc. | Anthelmintic depsipeptide compounds |
WO2017144546A1 (en) | 2016-02-23 | 2017-08-31 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods and pharmaceutical compositions for the treatment of nasopharyngeal carcinoma |
CN110167921A (zh) | 2016-11-16 | 2019-08-23 | 勃林格殷格翰动物保健美国公司 | 驱蠕虫缩肽化合物 |
CN109431983A (zh) * | 2018-11-30 | 2019-03-08 | 合肥中龙神力动物药业有限公司 | 一种兽用复方伊维菌素注射液及其制备方法 |
EP3956446A1 (en) | 2019-04-17 | 2022-02-23 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods and compositions for treatment of nlrp3 inflammasome mediated il-1beta dependent disorders |
WO2021198511A1 (en) | 2020-04-03 | 2021-10-07 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods and compositions for treatment of sars-cov-2 infection |
WO2022008597A1 (en) | 2020-07-08 | 2022-01-13 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Methods and pharmaceutical composition for the treatment of infectious diseases |
Family Cites Families (37)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5920285A (ja) | 1982-07-23 | 1984-02-01 | Sankyo Co Ltd | ミルベマイシンdの5−二塩基酸エステル誘導体及びその塩 |
JPS60126289A (ja) | 1983-11-14 | 1985-07-05 | Sankyo Co Ltd | ミルベマイシン類の5−カ−ボネ−ト誘導体 |
EP0185623A1 (de) | 1984-12-21 | 1986-06-25 | Ciba-Geigy Ag | Milbemycin-Derivate zur Bekämpfung von Insekten und Parasiten |
AU596586B2 (en) | 1985-04-30 | 1990-05-10 | American Cyanamid Company | Chemical derivatives of antibiotics S541 |
ES2059366T3 (es) | 1986-03-12 | 1994-11-16 | American Cyanamid Co | Compuestos macrolidos. |
GB8606105D0 (en) | 1986-03-12 | 1986-04-16 | Glaxo Group Ltd | Chemical compounds |
EP0260537A1 (en) | 1986-09-12 | 1988-03-23 | American Cyanamid Company | 13-Deoxy-23-oxo(keto) and 23-imino derivatives of 13-deoxy C-076-aglycone compounds |
EP0259779B1 (en) | 1986-09-12 | 1994-08-10 | American Cyanamid Company | 23-Oxo (Keto) and 23-imino Derivatives of LL-F28249 Compounds |
US4916154A (en) | 1986-09-12 | 1990-04-10 | American Cyanamid Company | 23-Imino derivatives of LL-F28249 compounds |
GB8721377D0 (en) | 1987-09-11 | 1987-10-21 | Glaxo Group Ltd | Chemical compounds |
PT88465B (pt) | 1987-09-11 | 1992-11-30 | American Cyanamid Co | Processo para a preparacao de um composto macrolido |
NO176766C (no) | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
CA2132199C (en) | 1992-03-17 | 2000-01-18 | Hitoshi Nishiyama | Depsipeptide derivative, production thereof and use thereof |
US5229416A (en) | 1992-04-29 | 1993-07-20 | Merck & Co., Inc. | Avermectin difluoro derivatives |
DE4317458A1 (de) | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
GB9226525D0 (en) * | 1992-12-19 | 1993-02-10 | Pfizer Ltd | Antiparasitic agents |
NZ261630A (en) | 1993-02-19 | 1998-05-27 | Meiji Seika Kaisha | Heteromacrocyclic compound and use as an assthelmintie |
DE4317457A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4317432A1 (de) | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
ES2170101T3 (es) | 1993-09-06 | 2002-08-01 | Fujisawa Pharmaceutical Co | Compuesto ciclodepsipeptido. |
DE4342907A1 (de) | 1993-12-16 | 1995-06-22 | Bayer Ag | Neue cyclische Depsipeptide mit 18 Ringatomen und ihre Verwendung zur Bekämpfung von Endoparasiten |
DE4401389A1 (de) | 1994-01-19 | 1995-07-20 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 12 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 12 Ringatomen und Verfahren zu ihrer Herstellung |
DE4406025A1 (de) | 1994-02-24 | 1995-08-31 | Bayer Ag | Milchsäure-haltige cyclische Depsipeptide mit 18 Ringatomen als endoparasitizide Mittel und Verfahren zu ihrer Herstellung |
DE4412492A1 (de) | 1994-04-12 | 1995-10-19 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen |
DE4437198A1 (de) | 1994-10-18 | 1996-04-25 | Bayer Ag | Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden |
DE19520275A1 (de) * | 1995-06-02 | 1996-12-05 | Bayer Ag | Endoparasitizide Mittel |
JP3985050B2 (ja) | 1995-06-30 | 2007-10-03 | アステラス製薬株式会社 | デプシペプチド誘導体その製造法およびその新規中間体 |
CZ295705B6 (cs) | 1995-09-22 | 2005-10-12 | Bayer Aktiengesellschaft | Cyklodepsipeptidové deriváty sloučeniny PF1022 a farmaceutický prostředek s jejich obsahem |
DE19545639A1 (de) | 1995-12-07 | 1997-06-12 | Bayer Ag | Verfahren zur Herstellung von substituierten Arylmilchsäure-haltigen Cyclodepsipeptiden mit 24 Ringatomen |
WO1998037088A1 (en) | 1997-02-19 | 1998-08-27 | Meiji Seika Kaisha Ltd. | Derivatives of cyclodepsipeptide, pf1022 substance |
DE19713626A1 (de) | 1997-04-02 | 1998-10-08 | Bayer Ag | Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung |
NZ501478A (en) | 1997-06-04 | 2001-05-25 | Bayer Ag | 8,20-bis-(substituted benzyl)-desoxycyclodepsipeptides and their use for combatting endoparasites |
DE19811559A1 (de) | 1998-03-17 | 1999-09-23 | Bayer Ag | Cyclooctadepsipeptide |
DE19828047A1 (de) | 1998-06-24 | 1999-12-30 | Bayer Ag | Substituierte Cyclooctadepsipeptide |
DE19840320A1 (de) | 1998-09-04 | 2000-03-09 | Bayer Ag | Aza-Cyclodepsipeptide |
DE10359798A1 (de) * | 2003-12-19 | 2005-07-21 | Bayer Healthcare Ag | Cyclohexadepsipeptide zur Bekämpfung von Endoparasiten und ein Verfahren zu ihrer Herstellung |
CN101619067B (zh) | 2009-03-25 | 2011-02-09 | 东北农业大学 | 大环内酯类化合物及其制备方法 |
-
2011
- 2011-08-26 WO PCT/EP2011/064761 patent/WO2012028556A1/en active Application Filing
- 2011-08-29 UY UY0001033577A patent/UY33577A/es not_active Application Discontinuation
- 2011-08-29 AR ARP110103139A patent/AR082787A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
UY33577A (es) | 2012-03-30 |
WO2012028556A1 (en) | 2012-03-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |