AR080923A1 - Proceso para la preparacion de amidas del acido pirazolcarboxilico - Google Patents
Proceso para la preparacion de amidas del acido pirazolcarboxilicoInfo
- Publication number
- AR080923A1 AR080923A1 ARP110101327A ARP110101327A AR080923A1 AR 080923 A1 AR080923 A1 AR 080923A1 AR P110101327 A ARP110101327 A AR P110101327A AR P110101327 A ARP110101327 A AR P110101327A AR 080923 A1 AR080923 A1 AR 080923A1
- Authority
- AR
- Argentina
- Prior art keywords
- formula
- compound
- bromine
- chlorine
- until
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 17
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 7
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 7
- 229910052794 bromium Chemical group 0.000 abstract 7
- 229910052801 chlorine Inorganic materials 0.000 abstract 7
- 239000000460 chlorine Substances 0.000 abstract 7
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 7
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 3
- 239000003054 catalyst Substances 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- HEDRZPFGACZZDS-UHFFFAOYSA-N Chloroform Chemical compound ClC(Cl)Cl HEDRZPFGACZZDS-UHFFFAOYSA-N 0.000 abstract 2
- KDLHZDBZIXYQEI-UHFFFAOYSA-N Palladium Chemical compound [Pd] KDLHZDBZIXYQEI-UHFFFAOYSA-N 0.000 abstract 2
- 239000003446 ligand Substances 0.000 abstract 2
- NAWXUBYGYWOOIX-SFHVURJKSA-N (2s)-2-[[4-[2-(2,4-diaminoquinazolin-6-yl)ethyl]benzoyl]amino]-4-methylidenepentanedioic acid Chemical compound C1=CC2=NC(N)=NC(N)=C2C=C1CCC1=CC=C(C(=O)N[C@@H](CC(=C)C(O)=O)C(O)=O)C=C1 NAWXUBYGYWOOIX-SFHVURJKSA-N 0.000 abstract 1
- RYGMFSIKBFXOCR-UHFFFAOYSA-N Copper Chemical compound [Cu] RYGMFSIKBFXOCR-UHFFFAOYSA-N 0.000 abstract 1
- PGTKVMVZBBZCKQ-UHFFFAOYSA-N Fulvene Chemical compound C=C1C=CC=C1 PGTKVMVZBBZCKQ-UHFFFAOYSA-N 0.000 abstract 1
- 239000005922 Phosphane Substances 0.000 abstract 1
- XYFCBTPGUUZFHI-UHFFFAOYSA-N Phosphine Chemical compound P XYFCBTPGUUZFHI-UHFFFAOYSA-N 0.000 abstract 1
- 229910052802 copper Inorganic materials 0.000 abstract 1
- 239000010949 copper Substances 0.000 abstract 1
- 229910052751 metal Inorganic materials 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 125000002524 organometallic group Chemical group 0.000 abstract 1
- 229910052763 palladium Inorganic materials 0.000 abstract 1
- 229910000064 phosphane Inorganic materials 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C17/00—Preparation of halogenated hydrocarbons
- C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
- C07C17/263—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
- C07C17/2635—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions involving a phosphorus compound, e.g. Wittig synthesis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C17/00—Preparation of halogenated hydrocarbons
- C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
- C07C17/30—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C17/00—Preparation of halogenated hydrocarbons
- C07C17/35—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction
- C07C17/354—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction by hydrogenation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
- C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10160439 | 2010-04-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR080923A1 true AR080923A1 (es) | 2012-05-16 |
Family
ID=43984050
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP110101327A AR080923A1 (es) | 2010-04-20 | 2011-04-18 | Proceso para la preparacion de amidas del acido pirazolcarboxilico |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8524915B2 (OSRAM) |
| EP (1) | EP2560960B1 (OSRAM) |
| JP (1) | JP6153864B2 (OSRAM) |
| CN (1) | CN102858749B (OSRAM) |
| AR (1) | AR080923A1 (OSRAM) |
| BR (1) | BR112012026456B1 (OSRAM) |
| ES (1) | ES2458935T3 (OSRAM) |
| IL (1) | IL222400A (OSRAM) |
| MX (1) | MX2012012009A (OSRAM) |
| TW (1) | TWI480041B (OSRAM) |
| UY (1) | UY33341A (OSRAM) |
| WO (1) | WO2011131544A1 (OSRAM) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI534126B (zh) * | 2011-01-25 | 2016-05-21 | 先正達合夥公司 | 用於製備吡唑羧酸醯胺之方法 |
| CN103483407B (zh) * | 2013-10-10 | 2015-11-18 | 宁夏启元药业有限公司 | 一种硫氰酸红霉素萃取结晶用复合溶媒及萃取结晶方法 |
| GB201403438D0 (en) * | 2014-02-27 | 2014-04-16 | Syngenta Participations Ag | Polymorphs |
| CN105985254B (zh) * | 2015-02-17 | 2018-03-16 | 上海中科绿碳化工科技有限公司 | 一种制备甲酰胺类化合物的方法 |
| CN106588745B (zh) * | 2016-12-02 | 2019-06-14 | 杭州百昂锐地科技有限公司 | 一种苯并烯氟菌唑的中间体及其制备方法和应用 |
| AU2023309261A1 (en) | 2022-07-22 | 2024-12-12 | Syngenta Crop Protection Ag | Solid form of a heterocyclic amide derivative |
| WO2025157998A1 (en) | 2024-01-26 | 2025-07-31 | Syngenta Crop Protection Ag | Chemical process |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH075487B2 (ja) | 1985-11-14 | 1995-01-25 | 住友化学工業株式会社 | １―ブロモ―２―クロロ―４―フルオロベンゼンの製造法 |
| US5093347A (en) | 1991-01-28 | 1992-03-03 | Monsanto Company | 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use |
| US7223879B2 (en) | 1998-07-10 | 2007-05-29 | Massachusetts Institute Of Technology | Ligands for metals and improved metal-catalyzed processes based thereon |
| AU2006308128B2 (en) * | 2005-10-25 | 2011-07-28 | Syngenta Crop Protection Ag | Heterocyclic amide derivatives useful as microbiocides |
| DK1963251T3 (da) * | 2005-12-12 | 2012-11-26 | Syngenta Participations Ag | Fremgangsmåde til fremstilling af aminer |
| CA2667499A1 (en) | 2006-10-25 | 2008-05-02 | Syngenta Limited | Process for the production of substituted bromobenzenes |
| US8227619B2 (en) | 2008-05-14 | 2012-07-24 | Syngenta Limited | Process for the preparation of amides |
| WO2010072631A1 (en) * | 2008-12-24 | 2010-07-01 | Syngenta Limited | Methods for the preparation of fungicides |
| RU2012146246A (ru) * | 2010-03-31 | 2014-05-10 | Актелион Фармасьютиклз Лтд | Антибактериальные производные изохинолин-3-илмочевины |
| CN102906072B (zh) * | 2010-04-20 | 2014-07-02 | 先正达参股股份有限公司 | 吡唑羧酸酰胺的制备方法 |
| EP2560957B1 (en) * | 2010-04-20 | 2014-05-07 | Syngenta Participations AG | Process for the preparation of pyrazole carboxylic acid amides |
| WO2011131546A1 (en) * | 2010-04-20 | 2011-10-27 | Syngenta Participations Ag | Process for the preparation of pyrazole carboxylic acid amides |
-
2011
- 2011-04-14 JP JP2013505408A patent/JP6153864B2/ja active Active
- 2011-04-14 US US13/642,511 patent/US8524915B2/en active Active
- 2011-04-14 EP EP11715687.7A patent/EP2560960B1/en active Active
- 2011-04-14 CN CN201180019764.XA patent/CN102858749B/zh active Active
- 2011-04-14 WO PCT/EP2011/055870 patent/WO2011131544A1/en not_active Ceased
- 2011-04-14 MX MX2012012009A patent/MX2012012009A/es active IP Right Grant
- 2011-04-14 ES ES11715687.7T patent/ES2458935T3/es active Active
- 2011-04-14 BR BR112012026456-7A patent/BR112012026456B1/pt active IP Right Grant
- 2011-04-15 UY UY0001033341A patent/UY33341A/es active IP Right Grant
- 2011-04-18 AR ARP110101327A patent/AR080923A1/es active IP Right Grant
- 2011-04-19 TW TW100113508A patent/TWI480041B/zh active
-
2012
- 2012-10-11 IL IL222400A patent/IL222400A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| ES2458935T3 (es) | 2014-05-07 |
| EP2560960B1 (en) | 2014-02-26 |
| MX2012012009A (es) | 2012-12-17 |
| US20130041160A1 (en) | 2013-02-14 |
| UY33341A (es) | 2011-12-01 |
| US8524915B2 (en) | 2013-09-03 |
| JP6153864B2 (ja) | 2017-06-28 |
| CN102858749B (zh) | 2014-07-02 |
| EP2560960A1 (en) | 2013-02-27 |
| BR112012026456B1 (pt) | 2017-06-27 |
| JP2013527840A (ja) | 2013-07-04 |
| TW201210590A (en) | 2012-03-16 |
| BR112012026456A2 (pt) | 2015-09-08 |
| WO2011131544A1 (en) | 2011-10-27 |
| IL222400A (en) | 2015-04-30 |
| CN102858749A (zh) | 2013-01-02 |
| TWI480041B (zh) | 2015-04-11 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR080923A1 (es) | Proceso para la preparacion de amidas del acido pirazolcarboxilico | |
| AR080921A1 (es) | Proceso para la preparacion de amidas de acido pirazolcarboxilico | |
| AR076974A1 (es) | Metodo para sintetizar pirfenidona | |
| IN2014DN06596A (OSRAM) | ||
| MY149709A (en) | Process for manufacturing acrolein or acrylic acid from glycerin | |
| UA106739C2 (uk) | Спосіб одержання каталізаторів фішера-тропша та їх застосування | |
| UY32142A (es) | Preparación de una quinoliniloxidifenilciclopropanodicarboxamida | |
| CL2011002085A1 (es) | Proceso para produccion de quimicos a partir de lignina, que comprende la depolimerizacion de la lignina mediante hidrogenacion catalitica para obtener hidrocraburos ciclicos, que luego se someten a reaccion catalitica de desoxigenacion y deshidrogenacion para convertir los hidrocarburos ciclicos en compuestos aromaticos. | |
| DE502007002576D1 (de) | Verfahren zur herstellung kupferhaltiger metallorganischer gerüstmaterialien | |
| IN2014DN10249A (OSRAM) | ||
| EP2772956A8 (en) | Material for positive hole injection transport layer, ink for positive hole injection transport layer, device, and production methods for same | |
| MX2012012005A (es) | Proceso para preparar amidas de acidos carboxilicos pirazolicos. | |
| ECSP11011004A (es) | Proceso para la preparación de benzonorbornenos | |
| JP2013525317A5 (OSRAM) | ||
| DE502006009282D1 (de) | Verfahren zur substitution von indenofluorenen | |
| PE20130252A1 (es) | Intermedios de agomelatina y metodo de preparacion de estos | |
| AR080924A1 (es) | Proceso para la preparacion de amidas del acido pirazolcarboxilico | |
| CR9771A (es) | Proceso para la produccion de anilinas | |
| GB201312783D0 (en) | Bis(Trifluoromethanesulfonyl)Ethyl-bearing compound and acid catalyst and method for preparing same | |
| MX2010008663A (es) | Procedimiento para preparar bifenilanilidas sustituidas. | |
| EA028190B9 (ru) | Монооксид азота в качестве катализатора цис/транс-изомеризации ненасыщенных соединений | |
| EA201491463A1 (ru) | Способ получения соединения по новой реакции присоединения михаэля с применением воды или различных кислот в качестве добавки | |
| MD4443B1 (ro) | Procedeu de sinteză a 3,4-dimetoxibiciclo[4.2.0]octa-1,3,5-trien-7-carbonitrilului şi aplicarea lui în sinteza ivabradinei şi a sărurilor sale de adiţie cu un acid acceptabil farmaceutic | |
| TH115394A (th) | กระบวนการสำหรับการจัดเตรียมของเบนโซนอร์บอร์นีน | |
| EA201070131A1 (ru) | Способ получения аминов |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration |