AR066692A1 - Procedimiento para la preparacion de derivados de epotilona por eepoxidacion catalitica selectiva - Google Patents
Procedimiento para la preparacion de derivados de epotilona por eepoxidacion catalitica selectivaInfo
- Publication number
- AR066692A1 AR066692A1 ARP080101279A ARP080101279A AR066692A1 AR 066692 A1 AR066692 A1 AR 066692A1 AR P080101279 A ARP080101279 A AR P080101279A AR P080101279 A ARP080101279 A AR P080101279A AR 066692 A1 AR066692 A1 AR 066692A1
- Authority
- AR
- Argentina
- Prior art keywords
- eepoxidation
- epotilone
- derivatives
- procedure
- preparation
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 230000003197 catalytic effect Effects 0.000 title 1
- 239000000010 aprotic solvent Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000003883 epothilone derivatives Chemical class 0.000 abstract 1
- 238000006735 epoxidation reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102007016046A DE102007016046A1 (de) | 2007-03-30 | 2007-03-30 | Verfahren zur Herstellung von Epothilonderivaten durch selektive katalytische Epoxidierung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR066692A1 true AR066692A1 (es) | 2009-09-09 |
Family
ID=39551678
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080101279A AR066692A1 (es) | 2007-03-30 | 2008-03-28 | Procedimiento para la preparacion de derivados de epotilona por eepoxidacion catalitica selectiva |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US20080242868A1 (https=) |
| EP (1) | EP2142539A2 (https=) |
| JP (1) | JP2010523481A (https=) |
| KR (1) | KR20090125259A (https=) |
| CN (1) | CN101652362B (https=) |
| AR (1) | AR066692A1 (https=) |
| CA (1) | CA2681806A1 (https=) |
| CL (1) | CL2008000901A1 (https=) |
| DE (1) | DE102007016046A1 (https=) |
| PA (1) | PA8773901A1 (https=) |
| TW (1) | TW200902538A (https=) |
| UY (1) | UY30985A1 (https=) |
| WO (1) | WO2008119563A2 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN114539143A (zh) * | 2022-01-28 | 2022-05-27 | 安徽瑞邦生物科技有限公司 | 一种4-氰基吡啶的纯化方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT1140944E (pt) * | 1998-12-22 | 2004-01-30 | Novartis Pharma Gmbh | Derivados de epotilona e sua utilizacao como agentes antitumorais |
| PE20010116A1 (es) | 1999-04-30 | 2001-02-15 | Schering Ag | Derivados de 6-alquenil-, 6-alquinil- y 6-epoxi-epotilona, procedimientos para su preparacion |
| EP1340498A1 (en) * | 2002-03-01 | 2003-09-03 | Schering Aktiengesellschaft | Use of epothilones in the treatment of brain diseases associated with proliferative processes |
| GB0405898D0 (en) * | 2004-03-16 | 2004-04-21 | Novartis Ag | Organic compounds |
-
2007
- 2007-03-30 DE DE102007016046A patent/DE102007016046A1/de not_active Withdrawn
-
2008
- 2008-03-27 UY UY30985A patent/UY30985A1/es not_active Application Discontinuation
- 2008-03-27 CA CA002681806A patent/CA2681806A1/en not_active Abandoned
- 2008-03-27 CN CN2008800103886A patent/CN101652362B/zh not_active Expired - Fee Related
- 2008-03-27 EP EP08734992A patent/EP2142539A2/de not_active Withdrawn
- 2008-03-27 US US12/056,393 patent/US20080242868A1/en not_active Abandoned
- 2008-03-27 WO PCT/EP2008/002652 patent/WO2008119563A2/de not_active Ceased
- 2008-03-27 JP JP2010500148A patent/JP2010523481A/ja not_active Withdrawn
- 2008-03-27 KR KR1020097020329A patent/KR20090125259A/ko not_active Withdrawn
- 2008-03-28 PA PA20088773901A patent/PA8773901A1/es unknown
- 2008-03-28 TW TW097111589A patent/TW200902538A/zh unknown
- 2008-03-28 AR ARP080101279A patent/AR066692A1/es not_active Application Discontinuation
- 2008-03-28 CL CL200800901A patent/CL2008000901A1/es unknown
-
2011
- 2011-11-30 US US13/308,046 patent/US8314248B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| KR20090125259A (ko) | 2009-12-04 |
| US20080242868A1 (en) | 2008-10-02 |
| UY30985A1 (es) | 2008-10-31 |
| US8314248B2 (en) | 2012-11-20 |
| JP2010523481A (ja) | 2010-07-15 |
| WO2008119563A3 (de) | 2009-02-12 |
| CN101652362B (zh) | 2012-10-10 |
| DE102007016046A1 (de) | 2008-10-23 |
| EP2142539A2 (de) | 2010-01-13 |
| CN101652362A (zh) | 2010-02-17 |
| CL2008000901A1 (es) | 2008-10-17 |
| WO2008119563A2 (de) | 2008-10-09 |
| CA2681806A1 (en) | 2008-10-09 |
| US20120077984A1 (en) | 2012-03-29 |
| PA8773901A1 (es) | 2008-11-19 |
| TW200902538A (en) | 2009-01-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY34104A (es) | ?compuestos derivados benzamídicos heterocíclicos, procesos e intermedios para su preparación, composiciones y métodos para su uso?. | |
| CL2017001930A1 (es) | Derivados de 4h-pirrol[3,2-c]piridin-4-ona | |
| CR20120334A (es) | Derivados de imidazopiridina como inhibidores de jak | |
| CL2011000917A1 (es) | Compuestos derivados de tioamida; sus metodos de preparacion y uso de los compuestos para el tratamiento de enfermedades endoparasitarias. | |
| MX2012005358A (es) | Procedimiento para la preparacion de etexilato de dabigatran. | |
| AR088109A1 (es) | Metodo para preparar analogos nucleotidicos antivirales | |
| ECSP088989A (es) | (aza)ciclohexanos carboxilados nuevos como ligandos de receptores de dopamina d3 | |
| MX382656B (es) | 3-oxo-3-(arilamino) propanoatos, proceso para su preparación y su uso en la preparación de pirrolidinonas. | |
| BRPI0820043A8 (pt) | Atividades do receptor de vitamina d e seus usos | |
| BR112012001998A2 (pt) | solução oftálmica, uso de um composto, e, método para preparação de uma solução oftálmica. | |
| CL2007003671A1 (es) | Metodo para la preparacion de derivados del acido 2-amino-5-cianobenzoico, utiles como intermediarios para la preparacion de las correspondientes diamidas cianoantranilicas. | |
| EA201100612A1 (ru) | Новые производные 2-амидотиадиазола | |
| NO20081684L (no) | En forbedret fremgangsmate for fremstilling av okazolidin-beskyttende aminodiolforbindelser anvendbare som mellomprodukter for Florfenicol | |
| ECSP088740A (es) | Derivados de tetrahidronaftalina, procedimientos para prepararlos y su uso como antiinflamatorios | |
| BR112019025028A2 (pt) | Método para preparar um composto. | |
| CL2012000374A1 (es) | Metodo para la preparacion de una composicion saborizante activa que comprende una primera reaccion entre un compuesto amino y un carbonilo, resultando una primera mezcla de intermediarios, una segunda reaccion con un segundo compuesto amino solo o en combinacion con un compuesto carbinilo, resultando una segunda mezcla de intermediarios, reacciones serparadas adicionales con compuestos de otras clases quimicas, ultima reaccion que comprende una mezcla de todas las mezclas de intermediarios anteriores. | |
| BR112013016241A2 (pt) | composto, e, método para fabricar um composto | |
| CR11824A (es) | Derivados heterocíclicos de la urea y sus métodos de empleo | |
| MX2009006750A (es) | Derivados de azaadamantano espirociclicos y metodos de uso. | |
| CL2013000589A1 (es) | Metodo para preparar derivados del acido 3-amino-4-(3,4,5,5-tetrasustituido)-2-oxo-piperidin-1-il)-4-butirico por reaccion entre un acido 3,4-diaminobutanoico y un acido 5-hidroxipentanoico. | |
| AR051341A1 (es) | Proceso para la preparacion de derivados de [1,4,5]-oxadiazepina | |
| WO2010080414A3 (en) | Substituted fno (2-[furan-2-yl] naphthalen-1-ol) derivatives as anti-cancer agents | |
| AR066692A1 (es) | Procedimiento para la preparacion de derivados de epotilona por eepoxidacion catalitica selectiva | |
| UY29434A1 (es) | Derivados de tetrahidronaftalina, procedimientos para su preparación y su uso como inhibidores de la inflamacinn | |
| PA8636101A1 (es) | Metodo para la preparacion de acidos hidroxamicos |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |