AR061477A1 - Metodos para utilizar un derivado de tiazol - Google Patents

Metodos para utilizar un derivado de tiazol

Info

Publication number
AR061477A1
AR061477A1 ARP070102637A ARP070102637A AR061477A1 AR 061477 A1 AR061477 A1 AR 061477A1 AR P070102637 A ARP070102637 A AR P070102637A AR P070102637 A ARP070102637 A AR P070102637A AR 061477 A1 AR061477 A1 AR 061477A1
Authority
AR
Argentina
Prior art keywords
tetomilast
beta2
receptor agonist
adrenergic receptor
disorder
Prior art date
Application number
ARP070102637A
Other languages
English (en)
Inventor
Kazuhiro Saito
H Nagamoto
N A Molfino
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of AR061477A1 publication Critical patent/AR061477A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/008Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/04Drugs for disorders of the respiratory system for throat disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Otolaryngology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente se refiere a un método para tratar una enfermedad, trastorno o afeccion en un paciente que comprende administrar a un paciente una cantidad efectiva para uso terapéutico de un derivado de tiazol, tetomilast. La presente además se refiere a la administracion de al menos un agonista del receptor beta2-adrenérgico con tetomilast para tratar una enfermedad, trastorno o afeccion. Además se refiere a la administracion de un esteroide antiinflamatorio con tetomilast y al menos un agonista del receptor beta2-adrenérgico para tratar una enfermedad, trastorno o afeccion. Reivindicacion 42: Una composicion farmacéutica caracterizada porque comprende tetomilast y al menos un agonista del receptor beta2-adrenérgico. Reivindicacion 46: La composicion farmacéutica de la reivindicacion 45, caracterizada porque el agonista del receptor beta2-adrenérgico se selecciona de salmeterol o albuterol y donde el esteroide antiinflamatorio es fluticasona.
ARP070102637A 2006-06-19 2007-06-15 Metodos para utilizar un derivado de tiazol AR061477A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US81454506P 2006-06-19 2006-06-19

Publications (1)

Publication Number Publication Date
AR061477A1 true AR061477A1 (es) 2008-08-27

Family

ID=38514103

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070102637A AR061477A1 (es) 2006-06-19 2007-06-15 Metodos para utilizar un derivado de tiazol

Country Status (17)

Country Link
US (1) US20120010179A1 (es)
EP (2) EP2040686A1 (es)
JP (3) JP2009541203A (es)
KR (3) KR20090021176A (es)
CN (2) CN102512676A (es)
AR (1) AR061477A1 (es)
AU (1) AU2007261951B2 (es)
BR (1) BRPI0713388A2 (es)
CA (1) CA2655296A1 (es)
IL (2) IL195894A0 (es)
MX (1) MX2008015380A (es)
PH (1) PH12014501074A1 (es)
RU (1) RU2542502C2 (es)
SG (1) SG184752A1 (es)
TW (2) TWI436761B (es)
WO (1) WO2007148806A1 (es)
ZA (1) ZA200810635B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7056916B2 (en) 2002-11-15 2006-06-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments for the treatment of chronic obstructive pulmonary disease
US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
ES2530991T3 (es) 2005-08-15 2015-03-09 Boehringer Ingelheim Int Procedimiento para la obtención de betamiméticos
JP2011513203A (ja) * 2008-03-14 2011-04-28 大塚製薬株式会社 Mmp−2及び/又はmmp−9阻害剤
TW201542207A (zh) * 2013-10-03 2015-11-16 Otsuka Pharma Co Ltd 嚴重氣喘治療劑

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1130017T3 (da) 1990-11-30 2005-10-10 Otsuka Pharma Co Ltd Azolderivater og deres anvendelse som superoxidradikalinhibitorer
ATE418536T1 (de) * 1996-08-12 2009-01-15 Celgene Corp Neue immunotherapeutische mittel und deren verwendung in der reduzierung von cytokinenspiegel
MY128323A (en) 1996-09-30 2007-01-31 Otsuka Pharma Co Ltd Thiazole derivatives for inhibition of cytokine production and of cell adhesion
AU777012B2 (en) * 1999-08-21 2004-09-30 Takeda Gmbh Synergistic combination of PDE inhibitors and beta 2 adrenoceptor agonist
EP1411936B1 (en) 2001-07-24 2005-09-28 Otsuka Pharmaceutical Co., Ltd. Use of thiazole derivatives for the manufacture of a medicament for the treatment of chronic obstructive pulmonary disease
JP3713577B2 (ja) * 2001-07-24 2005-11-09 大塚製薬株式会社 慢性閉塞性肺疾患治療薬
GB0123951D0 (en) * 2001-10-05 2001-11-28 Glaxo Group Ltd Therapies for treating respiratory diseases
WO2003037349A1 (en) * 2001-10-31 2003-05-08 Merck Patent Gmbh Type 4 phosphodiesterase inhibitors and uses thereof
US20040014563A1 (en) 2002-07-19 2004-01-22 Deere & Company, A Delaware Corporation Transmission shift control with engine torque control
ES2257152B1 (es) * 2004-05-31 2007-07-01 Laboratorios Almirall S.A. Combinaciones que comprenden agentes antimuscarinicos y agonistas beta-adrenergicos.
US20080269239A1 (en) * 2004-11-11 2008-10-30 Argenta Discovery Ltd. Pyrimidine Compounds as Histamine Modulators
CA2603433A1 (en) * 2005-03-30 2006-10-05 Schering Corporation Medicaments and methods combining an anticholinergic, a corticosteroid, and a long acting beta agonist

Also Published As

Publication number Publication date
BRPI0713388A2 (pt) 2012-03-27
JP2013047281A (ja) 2013-03-07
WO2007148806A1 (en) 2007-12-27
KR20090021176A (ko) 2009-02-27
KR20130014645A (ko) 2013-02-07
SG184752A1 (en) 2012-10-30
ZA200810635B (en) 2010-03-31
EP2040686A1 (en) 2009-04-01
TWI436761B (zh) 2014-05-11
IL195894A0 (en) 2009-09-01
TW201023916A (en) 2010-07-01
MX2008015380A (es) 2008-12-15
AU2007261951A1 (en) 2007-12-27
US20120010179A1 (en) 2012-01-12
CA2655296A1 (en) 2007-12-27
CN101472570A (zh) 2009-07-01
CN102512676A (zh) 2012-06-27
IL237789A0 (en) 2015-05-31
RU2009101317A (ru) 2010-07-27
PH12014501074A1 (en) 2015-09-28
AU2007261951B2 (en) 2011-03-31
TW200815054A (en) 2008-04-01
EP2522340A1 (en) 2012-11-14
KR20150016344A (ko) 2015-02-11
JP2009541203A (ja) 2009-11-26
JP2015083596A (ja) 2015-04-30
RU2542502C2 (ru) 2015-02-20

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