AR054737A1 - Piperidinas sustituidas pesticidas. - Google Patents
Piperidinas sustituidas pesticidas.Info
- Publication number
- AR054737A1 AR054737A1 ARP060100580A ARP060100580A AR054737A1 AR 054737 A1 AR054737 A1 AR 054737A1 AR P060100580 A ARP060100580 A AR P060100580A AR P060100580 A ARP060100580 A AR P060100580A AR 054737 A1 AR054737 A1 AR 054737A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- substituted
- alkoxy
- group
- halogen
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
- A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/58—1,2-Diazines; Hydrogenated 1,2-diazines
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Abstract
Reivindicacion 1: Uso de derivados de piperidina sustituidos de formula (1), o de una sal de dichos derivados aceptable para uso pesticida, para el control de plagas: donde: A es un haloalquileno-(C1-3) o alquileno-(C1-3) recto o ramificado; R1 es arilo-(C6-14), no sustituido o sustituido con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo-(C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12 y NR13R14; o es alquilo-(C1-6), cicloalquilo- (C3-7), cicloalquenilo-(C3-7), no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12, NR13R14, OH y oxo; o un heterociclilo o heteroarilo, no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo-(C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12, OH y oxo; R2 y R3 son independientemente H o alquilo-(C1-3); o donde R2 y R3 juntos pueden formar un puente alquileno-(C1-6); R4 y R5 son de modo independiente H, alquilo-(C1-6), alquenilo-(C2-6), o alcoxi-(C1-6); donde en el caso de que R4 y R5 sean independientemente alquilo-(C1-6), alquenilo-(C2-6), o alcoxi-(C1-6), ambos grupos juntos pueden formar un anillo de 4 a 7 miembros, con el átomo de carbono en la posicion 4 (C-4) del anillo piperidina; y donde los residuos pueden estar no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo-(C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12 y NR13R14, o en el caso de que R4 sea H o alquilo-(C1-6), R5 también puede ser OH, OCOR8, OCOOR9, OCO-COOalquilo-(C1-4), COOalquilo-(C1-4), COOH, CH2Fenilo, no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo-(C1-6), alcoxi(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O) pR12, o en el caso de que R5 sea un par de electrones de union, R4 puede formar junto con R5 un residuo X, seleccionado del grupo que consiste en O, S, N-OH, N-O-alquilo-(C1-6), N-O-CO-R8, N-O-COOR9; R7es H, alquilo-(C1-3), alquenilo-(C2-4); no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo-(C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12 y NR13R14 o donde los residuos R7 y R5 y los átomos de carbono en la posicion 3 (C-3) y en la posicion 4 (C-4) del anillo piperidina forman un residuo cicloalquilo-(C3-7), cicloalquenilo-(C3-7), o arilo-(C6-14); no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo- (C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12 y NR13R14; R8 es H, alquenilo-(C2-6), alquinilo-(C2-6), cicloalquilo-(C3-7) o alquilo(C1-6); no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, cicloalquilo-(C3-7), alcoxi-(C1-6), alquiltio(C1-6), OH, CN, NO2, R10, R11, S(O)pR12 y NR13R14; R9 es H, alquenilo-(C3-6), alquinilo-(C3-6), cicloalquilo-(C3-7) o alquilo(C1-6); no sustituidos o sustituidos con uno o más radicales seleccionados del grupo que consiste en halogeno, cicloalquilo-(C3-7), alcoxi-(C1-6), alquiltio-(C1-6), OH, CN, NO2, R10, R11, S(O)pR12 y NR13R14; R10 es arilo-(C6-14), no sustituido o sustituido con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo(C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12 y NR13R14; R11 es un radical heterociclilo o heteroaromático saturado o insaturado, no sustituido o sustituido con uno o más radicales seleccionados del grupo que consiste en halogeno, alquilo-(C1-6), haloalquilo-(C1-6), alcoxi-(C1-6), haloalcoxi-(C1-6), CN, NO2, S(O)pR12, OH y oxo; R12 es alquilo-(C1-6) o haloalquilo-(C1-6);R13 y R14 son de modo independiente H, alquilo-(C1-6), haloalquilo-(C1-6), alquenilo-(C2-6), alquinilo-(C2-6), cicloalquilo-(C3-7), o cicloalquilo-(C3-7)-alquilo-(C1-6); o un grupo donde R13 y R14 junto con el N forman un anillo heteroarilo o heterociclilo de 4 a 8 miembros, que puede contener uno o dos heteroátomos más; y donde: n es 0 o 1; y p es 0; 1 o 2.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP05003623A EP1692939A1 (en) | 2005-02-19 | 2005-02-19 | Pesticidal substituted piperidines |
Publications (1)
Publication Number | Publication Date |
---|---|
AR054737A1 true AR054737A1 (es) | 2007-07-11 |
Family
ID=35160081
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP060100580A AR054737A1 (es) | 2005-02-19 | 2006-02-17 | Piperidinas sustituidas pesticidas. |
Country Status (9)
Country | Link |
---|---|
US (1) | US20090082389A1 (es) |
EP (2) | EP1692939A1 (es) |
JP (1) | JP2008530159A (es) |
CN (1) | CN101132695B (es) |
AR (1) | AR054737A1 (es) |
BR (1) | BRPI0607864A2 (es) |
CA (1) | CA2588153C (es) |
MX (1) | MX2007010090A (es) |
WO (1) | WO2006087162A1 (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5258777B2 (ja) * | 2006-11-24 | 2013-08-07 | ノバルティス アーゲー | 害虫の駆除および阻止用組成物 |
MX2010002449A (es) * | 2007-08-31 | 2010-09-07 | Purdue Pharma Lp | Compuestos de piperidina tipo quinoxalina sustituida y uso de los mismsos. |
JP5369854B2 (ja) | 2008-04-21 | 2013-12-18 | 住友化学株式会社 | 有害節足動物防除組成物および縮合複素環化合物 |
AP2653A (en) * | 2008-12-12 | 2013-04-25 | Syngenta Participations Ag | Spiroheterocyclic N-oxypiperidines as pesticides |
WO2012083190A1 (en) * | 2010-12-17 | 2012-06-21 | The Rockefeller University | Insect odorant receptor antagonists |
PL2817302T3 (pl) * | 2012-02-21 | 2016-06-30 | Acraf | Związki 1H-indazolo-3-karboksyamidowe jako inhibitory kinazy syntazy glikogenu 3-beta |
WO2017201683A1 (en) * | 2016-05-25 | 2017-11-30 | Merck Sharp & Dohme Corp. | Substituted tetrahydroisoquinoline compounds useful as gpr120 agonists |
TW201841890A (zh) * | 2017-04-05 | 2018-12-01 | 日商阿格諾卡那休股份有限公司 | 新穎1-苯基哌啶衍生物及以其為有效成份之農園藝用藥劑 |
CN106957246B (zh) * | 2017-04-13 | 2019-06-25 | 云南大学 | 卤代苯胺类化合物及其制备方法和应用 |
KR102128782B1 (ko) * | 2018-09-20 | 2020-07-01 | 한양대학교 에리카산학협력단 | 트로페인(Tropane) 알칼로이드 화합물 및 순차적 산화반응을 이용한 이의 제조방법 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2435458A (en) * | 1943-12-09 | 1948-02-03 | Onyx Oil & Chemical Company | Cationic isoquinoline pesticide |
US3790595A (en) * | 1972-01-28 | 1974-02-05 | Lilly Co Eli | 4-substituted-5,7-dinitro-2-(alpha,alpha-difluoroalkyl)benzimidazole compounds |
AU4690979A (en) * | 1978-05-16 | 1979-11-29 | F. Hoffmann-La Roche Ag | Heterocyclic compounds |
DE2947649A1 (de) * | 1979-11-27 | 1981-08-06 | C.F. Spiess & Sohn GmbH & Co, 6719 Kleinkarlbach | Insektizide mittel |
JPH0778050B2 (ja) * | 1986-02-01 | 1995-08-23 | 日本ケミフア株式会社 | 新規なアルキレンジアミン誘導体およびグルタミン酸遮断剤 |
US5070196A (en) * | 1986-02-01 | 1991-12-03 | Nippon Chemiphar Co., Ltd. | Alkylenediamine derivatives |
ZA87690B (en) * | 1986-02-01 | 1987-09-30 | Nippon Chemiphar Co | Novel alkylenediamine derivatives |
DE4236126A1 (de) * | 1991-10-28 | 1993-04-29 | Ciba Geigy Ag | Cyclische buttersaeureamide |
JP2003508412A (ja) * | 1999-08-27 | 2003-03-04 | アベンティス・クロップサイエンス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | 農薬としてのアザビシクロおよびアザシクロオキシム、並びにアミン化合物 |
EP1420644B1 (de) * | 2001-08-23 | 2006-05-31 | Bayer CropScience S.A. | Substituierte propargylamine |
DE102004010086A1 (de) * | 2003-05-06 | 2004-09-16 | Syngenta Participations Ag | Substiuierte Piperidinderivate |
JP4595381B2 (ja) * | 2003-05-12 | 2010-12-08 | 住友化学株式会社 | ピリミジン化合物及びその有害生物防除用途 |
JP2004346016A (ja) * | 2003-05-22 | 2004-12-09 | Otsuka Chemical Co Ltd | トリフルオロメチルキノキサリン化合物、その製造方法、及び有害生物防除剤 |
EP1654249A1 (en) * | 2003-08-07 | 2006-05-10 | Pharmacia & Upjohn Company LLC | Anthelmintic and insecticide pyrimidine derivatives |
JP2006001914A (ja) * | 2004-06-21 | 2006-01-05 | Ishihara Sangyo Kaisha Ltd | ピリミジン系化合物、それらの製造方法及びそれらを含有する有害生物防除剤 |
-
2005
- 2005-02-19 EP EP05003623A patent/EP1692939A1/en not_active Withdrawn
-
2006
- 2006-02-14 CA CA2588153A patent/CA2588153C/en not_active Expired - Fee Related
- 2006-02-14 BR BRPI0607864-8A patent/BRPI0607864A2/pt not_active Application Discontinuation
- 2006-02-14 WO PCT/EP2006/001320 patent/WO2006087162A1/en active Application Filing
- 2006-02-14 MX MX2007010090A patent/MX2007010090A/es unknown
- 2006-02-14 JP JP2007555514A patent/JP2008530159A/ja active Pending
- 2006-02-14 EP EP06706927A patent/EP1848274A1/en not_active Withdrawn
- 2006-02-14 CN CN2006800015937A patent/CN101132695B/zh not_active Expired - Fee Related
- 2006-02-17 AR ARP060100580A patent/AR054737A1/es unknown
-
2007
- 2007-08-17 US US11/840,388 patent/US20090082389A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2588153C (en) | 2014-11-18 |
EP1848274A1 (en) | 2007-10-31 |
BRPI0607864A2 (pt) | 2009-10-20 |
MX2007010090A (es) | 2007-10-10 |
WO2006087162A1 (en) | 2006-08-24 |
CN101132695B (zh) | 2012-10-03 |
US20090082389A1 (en) | 2009-03-26 |
JP2008530159A (ja) | 2008-08-07 |
EP1692939A1 (en) | 2006-08-23 |
CA2588153A1 (en) | 2006-08-24 |
CN101132695A (zh) | 2008-02-27 |
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