AR047981A1 - Inhibidores de caspasa y sus usos correspondientes - Google Patents

Inhibidores de caspasa y sus usos correspondientes

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Publication number
AR047981A1
AR047981A1 ARP050100737A ARP050100737A AR047981A1 AR 047981 A1 AR047981 A1 AR 047981A1 AR P050100737 A ARP050100737 A AR P050100737A AR P050100737 A ARP050100737 A AR P050100737A AR 047981 A1 AR047981 A1 AR 047981A1
Authority
AR
Argentina
Prior art keywords
aliphatic
group
optionally
ring
cor9
Prior art date
Application number
ARP050100737A
Other languages
English (en)
Spanish (es)
Inventor
Jean-Damien Charrier
Steven Durrant
Michael Mortimore
Donnell Michael O
Alistair Rutherford
Sharn Ramaya
John R Studley
Martin Trudeau
Adam Looker
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34923260&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR047981(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of AR047981A1 publication Critical patent/AR047981A1/es

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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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NO20064344L (no) 2006-10-19
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IL177709A0 (en) 2006-12-31
EP1718639A2 (en) 2006-11-08
TW201217332A (en) 2012-05-01
BRPI0508102A (pt) 2007-07-17
HK1099757A1 (en) 2007-08-24
HK1159614A1 (en) 2012-08-03
TW200540152A (en) 2005-12-16
US20050233979A1 (en) 2005-10-20
ZA200607634B (en) 2008-01-08
TWI362381B (en) 2012-04-21
NZ549665A (en) 2010-09-30
JP2011144203A (ja) 2011-07-28
JP2014140385A (ja) 2014-08-07
US7652153B2 (en) 2010-01-26
EP2270004A1 (en) 2011-01-05
KR20060129069A (ko) 2006-12-14
RU2382780C2 (ru) 2010-02-27
WO2005085236A3 (en) 2005-10-20
AU2005219861A1 (en) 2005-09-15
CA2557645C (en) 2013-09-24
NO20064351L (no) 2006-11-20
US20100105914A1 (en) 2010-04-29
WO2005085236A2 (en) 2005-09-15
CN102161656A (zh) 2011-08-24
AU2005219861B2 (en) 2011-08-11
CA2557645A1 (en) 2005-09-15
CN102161656B (zh) 2013-02-20

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