AR046879A1 - Derivados de espiroindano - Google Patents

Derivados de espiroindano

Info

Publication number
AR046879A1
AR046879A1 ARP040104593A ARP040104593A AR046879A1 AR 046879 A1 AR046879 A1 AR 046879A1 AR P040104593 A ARP040104593 A AR P040104593A AR P040104593 A ARP040104593 A AR P040104593A AR 046879 A1 AR046879 A1 AR 046879A1
Authority
AR
Argentina
Prior art keywords
optionally substituted
alkyl
alkoxy
aryl
cycloalkyl
Prior art date
Application number
ARP040104593A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR046879A1 publication Critical patent/AR046879A1/es

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/20—N-Aryl derivatives thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/34—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the groups, e.g. biuret; Thio analogues thereof; Urea-aldehyde condensation products
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/20—Spiro-condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Wood Science & Technology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)

Abstract

Derivados de espiroindano, composiciones que los contengan y su uso para controlar insectos, ácaros, nematodes o moluscos. Reivindicación 1: Un compuesto de fórmula (1), donde X es O o NR11, donde R11 es hidrógeno, alquilo opcionalmente sustituido, arilo opcionalmente sustituido o heteroarilo opcionalmente sustituido; Y es una unión simple, C=O, C=S o S(O)m, donde m es 0, 1 ó 2; R1 es hidrógeno, alquilo opcionalmente sustituido, alcoxicarbonilo opcionalmente sustituido, alquilcarbonilo opcionalmente sustituido, aminocarbonilo, alquilaminocarbonilo opcionalmente sustituido, dialquilaminocarbonilo opcionalmente sustituido, arilo opcionalmente sustituido, heteroarilo opcionalmente sustituido, alcoxi opcionalmente sustituido, ariloxi opcionalmente sustituido, heteroariloxi opcionalmente sustituido, heterocicliloxi opcionalmente sustituido, ciano, alquenilo opcionalmente sustituido, alquinilo opcionalmente sustituido, cicloalquilo opcionalmente sustituido, cicloalquenilo opcionalmente sustituido, formilo, heterociclilo opcionalmente sustituido, alquiltio opcionalmente sustituido, NO o NR13R14, donde R13 y R14 son en forma independiente hidrógeno, COR15, alquilo opcionalmente sustituido, arilo opcionalmente sustituido, heteroarilo opcionalmente sustituido, heterociclilo opcionalmente sustituido o R13 y R14 junto con el átomo de N al que están unidos forman un grupo -N=C(R16)-NR17R18; R15 es H, alquilo opcionalmente sustituido, alcoxi opcionalmente sustituido, arilo opcionalmente sustituido, ariloxi opcionalmente sustituido, heteroarilo opcionalmente sustituido, heteroariloxi opcionalmente sustituido o NR19R20; R16, R17 y R18 son cada uno en forma independiente H o alquilo inferior; R10 y R20 son en forma independiente alquilo opcionalmente sustituido, arilo opcionalmente sustituido o heteroarilo opcionalmente sustituido; R2 y R3 son en forma independiente hidrógeno, halógeno, ciano, alquilo opcionalmente sustituido, alcoxi opcionalmente sustituido o arilo opcionalmente sustituido; cada R4 es independientemente halógeno, nitro, ciano, alquilo C1-8 opcionalmente sustituido, alquenilo C2-6 opcionalmente sustituido, alquinilo C2-6 opcionalmente sustituido, alcoxicarbonilo opcionalmente sustituido, alquilcarbonilo opcionalmente sustituido, alquilaminocarbonilo opcionalmente sustituido, dialquilaminocarbonilo opcionalmente sustituido, cicloalquilo C3-7 opcionalmente sustituido, arilo opcionalmente sustituido, heteroarilo opcionalmente sustituido, heterociclilo opcionalmente sustituido, alcoxi opcionalmente sustituido, ariloxi opcionalmente sustituido, heteroariloxi opcionalmente sustituido, alquiltio opcionalmente sustituido o R21R22N, donde R21 y R22 son, independientemente hidrógeno, alquilo C1-8, cicloalquilo C3-7, alquenilo C3-6, alquinilo C3-6, cicloalquil-(C3-7)(alquilo C1-4), haloalquilo C2-6, alcoxi-(C1-6)(alquilo C1-6), alcoxicarbonilo C1-6 o R21 y R22 junto con el átomo de N al que están unidos forman un anillo heterocíclico de cinco, seis o siete miembros que puede contener uno o dos heteroátomos adicionales seleccionados de O, N o S y que puede estar opcionalmente sustituido con uno o dos grupos alquilo C1-6, o 2 grupos adyacentes R4 junto con los átomos de carbono a los que están unidos forman un anillo carbocíclico o heterocíclico de 4, 5, 6 o 7 miembros que puede estar opcionalmente sustituido con halógeno; n es 0, 1, 2, 3 ó 4; cada Ra es independientemente hidrógeno, halógeno, hidroxi, ciano, alquilo C1-8 opcionalmente sustituido, alquenilo C2-6 opcionalmente sustituido, alquinilo C2-6 opcionalmente sustituido, alcoxicarbonilo opcionalmente sustituido, alquilcarbonilo opcionalmente sustituido, alquilaminocarbonilo opcionalmente sustituido, dialquilaminocarbonilo opcionalmente sustituido, cicloalquilo 3-7 opcionalmente sustituido, arilo opcionalmente sustituido, heteroarilo opcionalmente sustituido, heterociclilo opcionalmente sustituido, alcoxi opcionalmente sustituido, ariloxi opcionalmente sustituido, heteroariloxi opcionalmente sustituido, alquiltio opcionalmente sustituido, ariltio opcionalmente sustituido o R23R24N, donde R23 y R24 son, independientemente hidrógeno, alquilo C1- 8, cicloalquilo C3-7, alquenilo C3-6, alquinilo C3-6, cicloalquil-(C3-7)(alquilo C1-4), haloalquilo C2-6, alcoxi-(C1-6)(alquilo C1-6), alcoxicarbonilo C1-6 o R23 y R24 junto con el átomo de N al que están unidos forman un anillo heterocíclico de cinco, seis o siete miembros que puede contener uno o dos heteroátomos adicionales seleccionados de O, N o S y que puede estar opcionalmente sustituido con uno o dos grupos alquilo C1-6, o 2 grupos adyacentes Ra unidos al mismo átomo de carbono al que están unidos son =O o dos grupos Ra unidos a átomos de carbono adyacentes forman una unión, o dos grupos Ra junto con el átomo de carbono al que están unidos forman un anillo de tres a siete miembros, que puede ser saturado o no saturado, y que puede contener uno o dos heteroátomos seleccionados del grupo que consiste en N, O y S; y que puede estar opcionalmente sustituido con uno o dos grupos alquilo C1-6; o dos grupos Ra juntos forman un grupo -CH2-, CHCH- o -CH2-CH2; p es 0, 1, 2, 3, 4, 5 ó 6; q es 0, 1, 2, 3, 4, 5 ó 6 siempre que p+q sea 1, 2, 3, 4 5 ó 6; R8 es alquilo opcionalmente sustituido, alquenilo opcionalmente sustituido, alquinilo opcionalmente sustituido, cicloalquilo opcionalmente sustituido, arilo opcionalmente sustituido, alcoxi opcionalmente sustituido, ariloxi opcionalmente sustituido, alcoxicarbonilo opcionalmente sustituido, alquilcarbonilo opcionalmente sustituido o alquenilcarbonilo opcionalmente sustituido; o sales o N-óxidos de los mismos.
ARP040104593A 2003-12-12 2004-12-09 Derivados de espiroindano AR046879A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0328906.3A GB0328906D0 (en) 2003-12-12 2003-12-12 Chemical compounds

Publications (1)

Publication Number Publication Date
AR046879A1 true AR046879A1 (es) 2005-12-28

Family

ID=30130164

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP040104593A AR046879A1 (es) 2003-12-12 2004-12-09 Derivados de espiroindano

Country Status (10)

Country Link
US (2) US8354423B2 (es)
EP (1) EP1697327B1 (es)
JP (1) JP4819693B2 (es)
AR (1) AR046879A1 (es)
AT (1) ATE516273T1 (es)
BR (1) BRPI0417555B1 (es)
ES (1) ES2369764T3 (es)
GB (1) GB0328906D0 (es)
TW (1) TW200530215A (es)
WO (1) WO2005058836A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI20055288A0 (fi) 2005-06-06 2005-06-06 Nokia Corp Yksittäinen sanomanvälitys
CN101081835B (zh) * 2006-05-30 2011-09-21 上海药明康德新药开发有限公司 一种螺[苯并环-3-酮-1-(4′-哌啶)]模板化合物的合成方法
CN107903265A (zh) * 2017-11-21 2018-04-13 毛琳琳 一种新型螺环类杀虫剂的制备方法及应用

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Also Published As

Publication number Publication date
GB0328906D0 (en) 2004-01-14
EP1697327B1 (en) 2011-07-13
JP2007516253A (ja) 2007-06-21
BRPI0417555B1 (pt) 2013-12-17
EP1697327A1 (en) 2006-09-06
ES2369764T3 (es) 2011-12-05
TW200530215A (en) 2005-09-16
ATE516273T1 (de) 2011-07-15
US20080306101A1 (en) 2008-12-11
BRPI0417555A (pt) 2007-03-27
WO2005058836A1 (en) 2005-06-30
JP4819693B2 (ja) 2011-11-24
US8354423B2 (en) 2013-01-15
US20140031378A1 (en) 2014-01-30

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