AR023884A1 - Derivado de imidazodiazepina, un proceso para su elaboracion, medicamento, y el uso del derivado para elaboracion de medicamentos ansioliticos y /o anticonvulsivos y/o hipnoticos no sedantes. - Google Patents

Derivado de imidazodiazepina, un proceso para su elaboracion, medicamento, y el uso del derivado para elaboracion de medicamentos ansioliticos y /o anticonvulsivos y/o hipnoticos no sedantes.

Info

Publication number
AR023884A1
AR023884A1 ARP000102212A ARP000102212A AR023884A1 AR 023884 A1 AR023884 A1 AR 023884A1 AR P000102212 A ARP000102212 A AR P000102212A AR P000102212 A ARP000102212 A AR P000102212A AR 023884 A1 AR023884 A1 AR 023884A1
Authority
AR
Argentina
Prior art keywords
derivative
preparation
imidazodiazepin
ansiolitic
medication
Prior art date
Application number
ARP000102212A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR023884A1 publication Critical patent/AR023884A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente se relaciona con el compuesto 7-cloro-3-(5-dimetilaminometil-[1,2,4]oxadiazol-3-il)-5-metil-4,5-dihidro-imidazo[1,5-a][1,4]benzodiazepin-6-ona(1) y con el uso del compuesto de la formula (1) para la elaboracion de medicamentos para utilizar como medicamentos ansiolíticos y/o anticunvulsivos y/ohipnoticos no sedantes.
ARP000102212A 1999-05-12 2000-05-08 Derivado de imidazodiazepina, un proceso para su elaboracion, medicamento, y el uso del derivado para elaboracion de medicamentos ansioliticos y /o anticonvulsivos y/o hipnoticos no sedantes. AR023884A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP99109513 1999-05-12

Publications (1)

Publication Number Publication Date
AR023884A1 true AR023884A1 (es) 2002-09-04

Family

ID=8238165

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000102212A AR023884A1 (es) 1999-05-12 2000-05-08 Derivado de imidazodiazepina, un proceso para su elaboracion, medicamento, y el uso del derivado para elaboracion de medicamentos ansioliticos y /o anticonvulsivos y/o hipnoticos no sedantes.

Country Status (17)

Country Link
US (1) US6391873B1 (es)
EP (1) EP1178990B1 (es)
JP (1) JP3706307B2 (es)
KR (1) KR100451610B1 (es)
CN (1) CN1164590C (es)
AR (1) AR023884A1 (es)
AT (1) ATE231865T1 (es)
AU (1) AU769666B2 (es)
BR (1) BR0010495A (es)
CA (1) CA2372040C (es)
DE (1) DE60001313T2 (es)
DK (1) DK1178990T3 (es)
ES (1) ES2189759T3 (es)
MX (1) MXPA01011449A (es)
TR (1) TR200103237T2 (es)
WO (1) WO2000069858A1 (es)
ZA (1) ZA200108913B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5180077B2 (ja) 2006-08-11 2013-04-10 パナソニック株式会社 複数ドライブ装置の遅延対策と省電力制御を行う記録再生装置
US20090054412A1 (en) * 2007-08-20 2009-02-26 John Alan Kemp Treatment of Sleep Disorders
WO2009024324A2 (en) * 2007-08-20 2009-02-26 Evotec Neurosciences Gmbh Treatment of sleep disorders
US20100234359A1 (en) * 2007-08-20 2010-09-16 Evotec Neurosciences Gmbh Treatment of sleep disorders
ES2388708T3 (es) * 2008-01-22 2012-10-17 Eli Lilly And Company Antagonista selectivo del receptor opioide kappa
CN107007559B (zh) * 2017-04-21 2020-05-15 浙江京新药业股份有限公司 一种稳定的口服药物组合物及其制备方法
CN109134471B (zh) * 2017-06-27 2020-05-15 浙江京新药业股份有限公司 一种苯并二氮杂*化合物的固态形式及其制备方法和应用
CN112778220B (zh) * 2019-11-02 2024-06-07 浙江京新药业股份有限公司 一种苯并二氮杂䓬二酮化合物d的制备方法及其中间体
CN113045574B (zh) * 2019-12-26 2024-06-07 浙江京新药业股份有限公司 二氮杂䓬衍生物的制备方法及其中间体
US20220370409A1 (en) 2021-05-04 2022-11-24 Janssen Pharmaceuticals, Inc. Compositions And Methods For The Treatment Of Depression
TW202345796A (zh) 2022-03-07 2023-12-01 美商健生醫藥公司 阿替卡普蘭（ａｔｉｃａｐｒａｎｔ）之形式

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2143246C (en) 1994-03-16 2000-08-22 Thierry Godel Imidazodiazepines
DK0801651T3 (da) * 1995-01-06 2001-10-22 Hoffmann La Roche Hydroxymethyl-imidazodiazepiner og deres estere

Also Published As

Publication number Publication date
AU769666B2 (en) 2004-01-29
TR200103237T2 (tr) 2002-04-22
KR20010112487A (ko) 2001-12-20
DE60001313T2 (de) 2004-01-22
DK1178990T3 (da) 2003-05-26
CA2372040C (en) 2008-12-02
CN1350538A (zh) 2002-05-22
ATE231865T1 (de) 2003-02-15
JP3706307B2 (ja) 2005-10-12
JP2002544277A (ja) 2002-12-24
DE60001313D1 (en) 2003-03-06
US6391873B1 (en) 2002-05-21
KR100451610B1 (ko) 2004-10-06
BR0010495A (pt) 2002-02-13
ZA200108913B (en) 2003-03-26
EP1178990A1 (en) 2002-02-13
ES2189759T3 (es) 2003-07-16
WO2000069858A1 (en) 2000-11-23
CN1164590C (zh) 2004-09-01
MXPA01011449A (es) 2002-06-04
EP1178990B1 (en) 2003-01-29
CA2372040A1 (en) 2000-11-23
AU5211400A (en) 2000-12-05

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