AR022755A1 - Novedoso proceso - Google Patents
Novedoso procesoInfo
- Publication number
- AR022755A1 AR022755A1 ARP000100813A ARP000100813A AR022755A1 AR 022755 A1 AR022755 A1 AR 022755A1 AR P000100813 A ARP000100813 A AR P000100813A AR P000100813 A ARP000100813 A AR P000100813A AR 022755 A1 AR022755 A1 AR 022755A1
- Authority
- AR
- Argentina
- Prior art keywords
- formula
- compound
- salt
- solvate
- new process
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 150000003839 salts Chemical class 0.000 abstract 3
- 239000012453 solvate Substances 0.000 abstract 2
- BXQNSPXDWSNUKE-UHFFFAOYSA-N 1,3-benzothiazole 1-oxide Chemical class C1=CC=C2S(=O)C=NC2=C1 BXQNSPXDWSNUKE-UHFFFAOYSA-N 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 230000000144 pharmacologic effect Effects 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 150000003512 tertiary amines Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/16—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C317/18—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/10—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C323/11—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/12—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Proceso para preparar compuestos de benzotiazolona con actividad farmacologica de la formula (1) o una sal o solvato de los mismos, donde Ph representa ungrupo fenilo, que consiste en hacer reaccionar un compuesto de la formula (2) o una sal del mismo con un compuesto de la formula (3) en presencia de unsolvente y, optativamente, una base de amina terciaria y, se si desea, convertir el compuesto de la formula (1) a una sal o solvato farmacéuticamente aceptabledel mismo, e intermediarios empleados en su preparacion.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9900693A SE9900693D0 (sv) | 1999-02-26 | 1999-02-26 | Novel process |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR022755A1 true AR022755A1 (es) | 2002-09-04 |
Family
ID=20414646
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP000100813A AR022755A1 (es) | 1999-02-26 | 2000-02-25 | Novedoso proceso |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US20010039351A1 (es) |
| JP (1) | JP2002537389A (es) |
| KR (1) | KR20010108269A (es) |
| CN (1) | CN1341110A (es) |
| AR (1) | AR022755A1 (es) |
| AU (1) | AU3578500A (es) |
| BR (1) | BR0008545A (es) |
| CA (1) | CA2360456A1 (es) |
| CZ (1) | CZ20013068A3 (es) |
| EE (1) | EE200100407A (es) |
| IL (1) | IL144175A0 (es) |
| NO (1) | NO20014126L (es) |
| PL (1) | PL350138A1 (es) |
| SE (1) | SE9900693D0 (es) |
| TR (1) | TR200102447T2 (es) |
| WO (1) | WO2000050413A1 (es) |
| ZA (1) | ZA200105600B (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2329586T3 (es) | 2003-11-21 | 2009-11-27 | Theravance, Inc. | Compuestos que tienen actividad agonista del receptor beta2 adrenergico y antagonista del receptor muscarino. |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5648370A (en) * | 1990-11-20 | 1997-07-15 | Astra Pharmaceuticals Limited | 7-(2-aminoethyl) benzothiazolones |
| GB9211172D0 (en) * | 1992-05-27 | 1992-07-08 | Fisons Plc | Compounds |
-
1999
- 1999-02-26 SE SE9900693A patent/SE9900693D0/xx unknown
-
2000
- 2000-02-22 WO PCT/SE2000/000347 patent/WO2000050413A1/en not_active Application Discontinuation
- 2000-02-22 JP JP2000600996A patent/JP2002537389A/ja active Pending
- 2000-02-22 PL PL00350138A patent/PL350138A1/xx not_active Application Discontinuation
- 2000-02-22 BR BR0008545-6A patent/BR0008545A/pt not_active Application Discontinuation
- 2000-02-22 CZ CZ20013068A patent/CZ20013068A3/cs unknown
- 2000-02-22 CA CA002360456A patent/CA2360456A1/en not_active Abandoned
- 2000-02-22 KR KR1020017010918A patent/KR20010108269A/ko not_active Application Discontinuation
- 2000-02-22 EE EEP200100407A patent/EE200100407A/xx unknown
- 2000-02-22 TR TR2001/02447T patent/TR200102447T2/xx unknown
- 2000-02-22 IL IL14417500A patent/IL144175A0/xx unknown
- 2000-02-22 AU AU35785/00A patent/AU3578500A/en not_active Abandoned
- 2000-02-22 CN CN00804067A patent/CN1341110A/zh active Pending
- 2000-02-25 AR ARP000100813A patent/AR022755A1/es unknown
-
2001
- 2001-04-27 US US09/842,710 patent/US20010039351A1/en not_active Abandoned
- 2001-07-06 ZA ZA200105600A patent/ZA200105600B/en unknown
- 2001-08-24 NO NO20014126A patent/NO20014126L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1341110A (zh) | 2002-03-20 |
| JP2002537389A (ja) | 2002-11-05 |
| ZA200105600B (en) | 2002-10-07 |
| SE9900693D0 (sv) | 1999-02-26 |
| KR20010108269A (ko) | 2001-12-07 |
| CZ20013068A3 (cs) | 2002-01-16 |
| WO2000050413A1 (en) | 2000-08-31 |
| NO20014126D0 (no) | 2001-08-24 |
| IL144175A0 (en) | 2002-05-23 |
| US20010039351A1 (en) | 2001-11-08 |
| PL350138A1 (en) | 2002-11-04 |
| EE200100407A (et) | 2002-10-15 |
| CA2360456A1 (en) | 2000-08-31 |
| NO20014126L (no) | 2001-08-24 |
| TR200102447T2 (tr) | 2002-01-21 |
| AU3578500A (en) | 2000-09-14 |
| BR0008545A (pt) | 2001-11-06 |
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