AR014922A1 - Compuesto derivado de indol util en terapia, proceso para su preparacion, formulaciones farmaceuticas y procedimiento de tratamiento. - Google Patents

Compuesto derivado de indol util en terapia, proceso para su preparacion, formulaciones farmaceuticas y procedimiento de tratamiento.

Info

Publication number
AR014922A1
AR014922A1 ARP980105232A ARP980105232A AR014922A1 AR 014922 A1 AR014922 A1 AR 014922A1 AR P980105232 A ARP980105232 A AR P980105232A AR P980105232 A ARP980105232 A AR P980105232A AR 014922 A1 AR014922 A1 AR 014922A1
Authority
AR
Argentina
Prior art keywords
useful
indol
therapy
preparation
processing procedure
Prior art date
Application number
ARP980105232A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AR014922A1 publication Critical patent/AR014922A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se describe el ácido (S)-(+)-3-{1-(1,3-benzodioxol-5-il)-2-[(2-metoxi-4- metilfenil)sulfonilamino]-2-oxoetil}-1-metil-1h-indol-6-carboxílico, que estáen gran parte libre de su enantiomero (R)- (-), y derivados farmacéuticamente aceptables del mismo.Los compuestos son utiles en el tratamiento de la insuficiencia renal aguda inter alia, reestenosis e hipertension pulmonar. Se describen también procesosde preparacion y formulaciones farmacéuticas y procedimiento de tratamiento que utilizadicho compuesto (I).
ARP980105232A 1997-10-22 1998-10-20 Compuesto derivado de indol util en terapia, proceso para su preparacion, formulaciones farmaceuticas y procedimiento de tratamiento. AR014922A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9722287.1A GB9722287D0 (en) 1997-10-22 1997-10-22 Compounds useful in therapy

Publications (1)

Publication Number Publication Date
AR014922A1 true AR014922A1 (es) 2001-04-11

Family

ID=10820904

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980105232A AR014922A1 (es) 1997-10-22 1998-10-20 Compuesto derivado de indol util en terapia, proceso para su preparacion, formulaciones farmaceuticas y procedimiento de tratamiento.

Country Status (17)

Country Link
US (1) US6211223B1 (es)
AP (1) AP899A (es)
AR (1) AR014922A1 (es)
AU (1) AU1150999A (es)
BG (1) BG104394A (es)
CA (1) CA2308478C (es)
CZ (1) CZ20001514A3 (es)
DZ (1) DZ2628A1 (es)
GB (1) GB9722287D0 (es)
GT (1) GT199800161A (es)
MA (1) MA26556A1 (es)
MY (1) MY117148A (es)
PA (1) PA8461001A1 (es)
TN (1) TNSN98190A1 (es)
TW (1) TW483893B (es)
WO (1) WO1999020623A1 (es)
ZA (1) ZA989574B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9722287D0 (en) 1997-10-22 1997-12-17 Pfizer Ltd Compounds useful in therapy
AR037097A1 (es) 2001-10-05 2004-10-20 Novartis Ag Compuestos acilsulfonamidas, composiciones farmaceuticas y el uso de dichos compuestos para la preparacion de un medicamento
CN106631920B (zh) * 2016-11-17 2018-11-13 贵州大学 一种2-羟基-4-甲基苯磺酸的制备方法
CN114507162A (zh) * 2020-11-16 2022-05-17 尚科生物医药(上海)有限公司 一种制备2-氟-5-甲氧基苯磺酰氯的方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE189217T1 (de) * 1993-03-19 2000-02-15 Merck & Co Inc Phenoxyphenylessigsäurederivate
GB9609641D0 (en) * 1996-05-09 1996-07-10 Pfizer Ltd Compounds useful in therapy
GB9722287D0 (en) 1997-10-22 1997-12-17 Pfizer Ltd Compounds useful in therapy

Also Published As

Publication number Publication date
TW483893B (en) 2002-04-21
CA2308478A1 (en) 1999-04-29
AU1150999A (en) 1999-05-10
GB9722287D0 (en) 1997-12-17
TNSN98190A1 (fr) 2005-03-15
CZ20001514A3 (cs) 2001-09-12
PA8461001A1 (es) 2000-05-24
DZ2628A1 (fr) 2003-03-08
AP899A (en) 2000-11-17
GT199800161A (es) 2000-04-11
ZA989574B (en) 2000-04-25
MY117148A (en) 2004-05-31
AP9801370A0 (en) 1998-12-31
BG104394A (en) 2001-09-28
US6211223B1 (en) 2001-04-03
MA26556A1 (fr) 2004-12-20
WO1999020623A1 (en) 1999-04-29
CA2308478C (en) 2004-12-07

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