AR004689A1 - Derivados del acido piridazinacetico y del acido tiadiazinacetico, procedimiento para prepararlos, preparaciones farmaceuticas que los contienen yprocedimiento para preparar estas preparaciones farmaceuticas. - Google Patents
Derivados del acido piridazinacetico y del acido tiadiazinacetico, procedimiento para prepararlos, preparaciones farmaceuticas que los contienen yprocedimiento para preparar estas preparaciones farmaceuticas.Info
- Publication number
- AR004689A1 AR004689A1 ARP960104655A AR10465596A AR004689A1 AR 004689 A1 AR004689 A1 AR 004689A1 AR P960104655 A ARP960104655 A AR P960104655A AR 10465596 A AR10465596 A AR 10465596A AR 004689 A1 AR004689 A1 AR 004689A1
- Authority
- AR
- Argentina
- Prior art keywords
- acid
- prepare
- procedure
- pharmaceutical preparations
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/04—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/14—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Derivados del ácido piridazinacético y del ácido tiadiazinacético, por responder a la fórmula I, en la que Y representa -C(R4R4)-C(R4R4)-,-CR4=CR4- o-C(R4R4)-S- R1 representa Het, Ar, R3 o R4, R2 representa Ar o un grupo no sustituído, o bien mono o disustituido en el fenilo con A,R3,OR4, NH2, NHA, NA2, NO2, CN, Hal, NHCOR4, NHSO2R4, COOR4, COR4,CONHSO2R6,O(CH2)nR3, OPh, O(CH2)n OR4 o S(O)mR4, o bien un grupo no sustituído.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19537548A DE19537548A1 (de) | 1995-10-09 | 1995-10-09 | Endothelin-Rezeptor-Antagonisten |
Publications (1)
Publication Number | Publication Date |
---|---|
AR004689A1 true AR004689A1 (es) | 1999-03-10 |
Family
ID=7774384
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP960104655A AR004689A1 (es) | 1995-10-09 | 1996-09-10 | Derivados del acido piridazinacetico y del acido tiadiazinacetico, procedimiento para prepararlos, preparaciones farmaceuticas que los contienen yprocedimiento para preparar estas preparaciones farmaceuticas. |
Country Status (16)
Country | Link |
---|---|
US (1) | US5883090A (es) |
EP (1) | EP0796250A1 (es) |
JP (1) | JPH10511118A (es) |
CN (1) | CN1168137A (es) |
AR (1) | AR004689A1 (es) |
AU (1) | AU7211996A (es) |
BR (1) | BR9606668A (es) |
CA (1) | CA2207243A1 (es) |
CZ (1) | CZ176897A3 (es) |
DE (1) | DE19537548A1 (es) |
HU (1) | HUP9801879A3 (es) |
NO (1) | NO972612L (es) |
PL (1) | PL320638A1 (es) |
SK (1) | SK73597A3 (es) |
WO (1) | WO1997013758A1 (es) |
ZA (1) | ZA968483B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6187920B1 (en) * | 1998-03-26 | 2001-02-13 | Sumitomo Chemical Co., Ltd. | Pyridazinone derivatives |
US6670362B2 (en) * | 2000-09-20 | 2003-12-30 | Pfizer Inc. | Pyridazine endothelin antagonists |
GB0023074D0 (en) * | 2000-09-20 | 2000-11-01 | Pfizer Ltd | Pyridazines |
US6996060B1 (en) | 2001-03-20 | 2006-02-07 | Arraycomm, Inc. | Closing a communications stream between terminals of a communications system |
US7339906B1 (en) * | 2001-03-20 | 2008-03-04 | Arraycomm, Llc | Opening a communications stream between a user terminal and a base station |
DE10155076A1 (de) * | 2001-11-09 | 2003-05-22 | Merck Patent Gmbh | Verwendung von Endothelin-Rezeptor-Antagonisten zur Behandlung von Tumorerkrankungen |
CA2577782A1 (en) * | 2004-08-23 | 2006-03-02 | Wyeth | Pyrrolo-naphthyl acids as pai-1 inhibitors |
BRPI0514544A (pt) | 2004-08-23 | 2008-06-17 | Wyeth Corp | ácidos de oxazol-naftila como moduladores de inibidor tipo-1 de ativador de plasminogênio (pai-1) |
JP2008510816A (ja) | 2004-08-23 | 2008-04-10 | ワイス | チアゾロ−ナフチル酸 |
CN109867613B (zh) * | 2017-12-01 | 2021-08-17 | 中国科学院大连化学物理研究所 | 一种多取代苯甲酸及其合成方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2832780A (en) * | 1955-09-14 | 1958-04-29 | Warner Lambert Pharmaceutical | Hydrazides of pyridazonyl-substituted alkanoic acids |
BR8108745A (pt) * | 1980-08-07 | 1982-07-06 | Diamond Shamrock Corp | Difenilpiridazinonas herbicidas e reguladores do crescimento da planta |
RO117847B1 (ro) * | 1991-11-05 | 2002-08-30 | Smithkline Beecham Corp | Derivati de indan, procedeu de preparare, compozitie farmaceutica care ii contine si metoda de tratament |
ZA939516B (en) * | 1992-12-22 | 1994-06-06 | Smithkline Beecham Corp | Endothelin receptor antagonists |
EP0617001B1 (en) * | 1993-03-19 | 2000-01-26 | Merck & Co. Inc. | Phenoxyphenylacetic acid derivatives |
DE4339868A1 (de) * | 1993-11-23 | 1995-05-24 | Merck Patent Gmbh | Imidazopyridazine |
TW282456B (es) * | 1994-03-10 | 1996-08-01 | Fujisawa Yakusin Kogyo Kk |
-
1995
- 1995-10-09 DE DE19537548A patent/DE19537548A1/de not_active Withdrawn
-
1996
- 1996-09-10 AR ARP960104655A patent/AR004689A1/es unknown
- 1996-09-19 US US08/849,344 patent/US5883090A/en not_active Expired - Fee Related
- 1996-09-19 SK SK735-97A patent/SK73597A3/sk unknown
- 1996-09-19 JP JP9514665A patent/JPH10511118A/ja active Pending
- 1996-09-19 HU HU9801879A patent/HUP9801879A3/hu unknown
- 1996-09-19 CZ CZ971768A patent/CZ176897A3/cs unknown
- 1996-09-19 WO PCT/EP1996/004111 patent/WO1997013758A1/de not_active Application Discontinuation
- 1996-09-19 AU AU72119/96A patent/AU7211996A/en not_active Abandoned
- 1996-09-19 PL PL96320638A patent/PL320638A1/xx unknown
- 1996-09-19 CN CN96191388A patent/CN1168137A/zh active Pending
- 1996-09-19 EP EP96933341A patent/EP0796250A1/de not_active Withdrawn
- 1996-09-19 CA CA002207243A patent/CA2207243A1/en not_active Abandoned
- 1996-09-19 BR BR9606668A patent/BR9606668A/pt not_active Application Discontinuation
- 1996-10-08 ZA ZA968483A patent/ZA968483B/xx unknown
-
1997
- 1997-06-06 NO NO972612A patent/NO972612L/no unknown
Also Published As
Publication number | Publication date |
---|---|
ZA968483B (en) | 1997-05-20 |
HUP9801879A3 (en) | 1999-07-28 |
CA2207243A1 (en) | 1997-04-17 |
CZ176897A3 (en) | 1997-10-15 |
CN1168137A (zh) | 1997-12-17 |
WO1997013758A1 (de) | 1997-04-17 |
SK73597A3 (en) | 1998-05-06 |
NO972612D0 (no) | 1997-06-06 |
MX9704262A (es) | 1997-09-30 |
JPH10511118A (ja) | 1998-10-27 |
HUP9801879A2 (hu) | 1999-06-28 |
PL320638A1 (en) | 1997-10-13 |
DE19537548A1 (de) | 1997-04-10 |
EP0796250A1 (de) | 1997-09-24 |
BR9606668A (pt) | 1997-09-30 |
NO972612L (no) | 1997-08-08 |
US5883090A (en) | 1999-03-16 |
AU7211996A (en) | 1997-04-30 |
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