AP3413A - Adenosine a1 agonists for the treatment of glaucoma and ocular hypertension - Google Patents
Adenosine a1 agonists for the treatment of glaucoma and ocular hypertensionInfo
- Publication number
- AP3413A AP3413A AP2013006753A AP2013006753A AP3413A AP 3413 A AP3413 A AP 3413A AP 2013006753 A AP2013006753 A AP 2013006753A AP 2013006753 A AP2013006753 A AP 2013006753A AP 3413 A AP3413 A AP 3413A
- Authority
- AP
- ARIPO
- Prior art keywords
- glaucoma
- adenosine
- agonists
- treatment
- ocular hypertension
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10175151 | 2010-09-02 | ||
PCT/EP2011/064829 WO2012028585A1 (fr) | 2010-09-02 | 2011-08-29 | Agonistes du récepteur a1 à l'adénosine destinés au traitement du glaucome et de l'hypertension oculaire |
Publications (2)
Publication Number | Publication Date |
---|---|
AP2013006753A0 AP2013006753A0 (en) | 2013-02-28 |
AP3413A true AP3413A (en) | 2015-09-30 |
Family
ID=44582992
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2013006753A AP3413A (en) | 2010-09-02 | 2011-08-29 | Adenosine a1 agonists for the treatment of glaucoma and ocular hypertension |
Country Status (30)
Country | Link |
---|---|
US (3) | US20120058983A1 (fr) |
EP (1) | EP2611415B1 (fr) |
JP (1) | JP5875585B2 (fr) |
KR (1) | KR20140091457A (fr) |
CN (1) | CN103249400B (fr) |
AP (1) | AP3413A (fr) |
AU (1) | AU2011298430B2 (fr) |
BR (1) | BR112013005224A2 (fr) |
CA (1) | CA2809700A1 (fr) |
CL (2) | CL2013000599A1 (fr) |
CR (1) | CR20130094A (fr) |
CY (1) | CY1117458T1 (fr) |
DK (1) | DK2611415T3 (fr) |
EA (1) | EA028411B1 (fr) |
ES (1) | ES2570659T3 (fr) |
HK (1) | HK1188138A1 (fr) |
HR (1) | HRP20160532T1 (fr) |
HU (1) | HUE027295T2 (fr) |
MA (1) | MA34489B1 (fr) |
MX (1) | MX2013002396A (fr) |
MY (1) | MY160383A (fr) |
NZ (1) | NZ607624A (fr) |
PL (1) | PL2611415T3 (fr) |
RS (1) | RS54743B1 (fr) |
SG (1) | SG187974A1 (fr) |
SI (1) | SI2611415T1 (fr) |
TW (1) | TWI516266B (fr) |
UA (1) | UA111947C2 (fr) |
WO (1) | WO2012028585A1 (fr) |
ZA (1) | ZA201302340B (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20140128974A (ko) | 2012-01-26 | 2014-11-06 | 이노텍 파마슈티컬스 코포레이션 | ((2r,3s,4r,5r)-5-(6-(시클로펜틸아미노)-9h-퓨린-9-일)-3,4-디히드록시테트라히드로푸란-2-일) 메틸 니트레이트의 무수 다형체들 및 이들의 제조 방법들 |
US20160317542A1 (en) | 2013-12-09 | 2016-11-03 | Respira Therapeutics, Inc. | Pde5 inhibitor powder formulations and methods relating thereto |
CA2933244A1 (fr) * | 2013-12-12 | 2015-06-18 | Bayer Pharma Aktiengesellschaft | Agonistes a1 de l'adenosine utilises comme medicaments contre les maladies des reins |
EA031723B1 (ru) * | 2014-01-10 | 2019-02-28 | Сантэн Фармасьютикал Ко., Лтд. | Фармацевтическая композиция, содержащая соединение пиридиламиноуксусной кислоты и полиоксиэтиленовое касторовое масло |
ES2744227T3 (es) * | 2015-05-06 | 2020-02-24 | Bayer Pharma AG | Procedimiento para la preparación de monoclorhidrato de L-alanil-L-alaninato de 2-{4-[2-({[2-(4-clorofenil)-1,3-tiazol-4-il]metil}sulfanil)-3,5-diciano-6-(pirrolidin-1-il)piridin-4-il]fenoxi}etilo |
WO2017137528A1 (fr) | 2016-02-12 | 2017-08-17 | Charité - Universitätsmedizin Berlin | Agoniste du récepteur a1 de l'adénosine pour utilisation dans le traitement de l'état de mal épileptique |
CN112545983A (zh) * | 2020-12-18 | 2021-03-26 | 合肥中龙神力动物药业有限公司 | 一种复方硫酸新霉素滴眼液及其制备方法和应用 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102007036076A1 (de) * | 2007-08-01 | 2009-02-05 | Bayer Healthcare Aktiengesellschaft | Dipeptoid-Produgs und ihre Verwendung |
DE102008062561A1 (de) * | 2008-12-16 | 2010-06-24 | Maxon Motor Ag | Bausatz für einen Elektromotor mit einem Drehwinkelgeber |
Family Cites Families (61)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4052510A (en) | 1974-12-18 | 1977-10-04 | Sandoz, Inc. | 4-alkyl-2,6-di(secondary or tertiary alkylamino) pyridines, compositions thereof and methods for treating diabetes and obesity |
TW299333B (fr) | 1992-12-29 | 1997-03-01 | Takeda Pharm Industry Co Ltd | |
DE4334919A1 (de) * | 1993-10-13 | 1995-04-20 | Liedtke Pharmed Gmbh | Grenzwertig wirksame Arzneiformen mit Betablockern |
CN1056611C (zh) | 1994-06-16 | 2000-09-20 | 美国辉瑞有限公司 | 吡唑并吡啶和吡咯并吡啶,其用途和用于制备它们的中间体 |
DE4430638A1 (de) | 1994-08-29 | 1996-03-07 | Bayer Ag | Verwendung von substituierten 4-Phenyl-6-amino-nicotinsäurederivaten als Arzneimittel |
JPH09132529A (ja) | 1995-11-09 | 1997-05-20 | Ono Pharmaceut Co Ltd | 一酸化窒素合成酵素阻害剤 |
CN1158290C (zh) | 1996-01-17 | 2004-07-21 | 诺沃挪第克公司 | 稠合1,2,4-噻二嗪与稠合1,4-噻嗪衍生物、其制备方法及用途 |
WO1997027177A2 (fr) | 1996-01-29 | 1997-07-31 | The United States Of America, Represented By The Secretary, Department Of Health And Human Services | Derives de dihydropyridine-, pyridine-, benzopyrane- mono- et triazoloquinazoline, leur preparation, et utilsation comme antagonistes des recepteurs de l'adenosine |
JPH10324687A (ja) | 1997-02-19 | 1998-12-08 | Nippon Soda Co Ltd | ピロール化合物、製法および農園芸用殺菌剤 |
WO1998054139A1 (fr) | 1997-05-30 | 1998-12-03 | Basf Aktiengesellschaft | Procede de fabrication de thiopyridines substituees |
PL338013A1 (en) | 1997-07-16 | 2000-09-25 | Novo Nordisk As | Derivatives of condensed 1,2,4-thiadiazine, their production and application |
US6632823B1 (en) | 1997-12-22 | 2003-10-14 | Merck & Co., Inc. | Substituted pyridine compounds useful as modulators of acetylcholine receptors |
DE19834044A1 (de) | 1998-07-29 | 2000-02-03 | Bayer Ag | Neue substituierte Pyrazolderivate |
DE19834047A1 (de) | 1998-07-29 | 2000-02-03 | Bayer Ag | Substituierte Pyrazolderivate |
DE19943634A1 (de) | 1999-09-13 | 2001-04-12 | Bayer Ag | Neuartige Dicarbonsäurederivate mit pharmazeutischen Eigenschaften |
DE19943636A1 (de) | 1999-09-13 | 2001-03-15 | Bayer Ag | Neuartige Dicarbonsäurederivate mit pharmazeutischen Eigenschaften |
DE19943635A1 (de) | 1999-09-13 | 2001-03-15 | Bayer Ag | Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften |
DE19947154A1 (de) | 1999-10-01 | 2001-10-04 | Bayer Ag | Substituierte 2-Thio-3,5-dicyano-4-aryl-6-aminopyridine und ihre Verwendung |
ATE293962T1 (de) | 2000-02-25 | 2005-05-15 | Hoffmann La Roche | Adenosin-rezeptor modulatoren |
AU2001269529A1 (en) | 2000-07-18 | 2002-01-30 | Yamanouchi Pharmaceutical Co., Ltd. | Medicine comprising dicyanopyridine derivative |
AR031176A1 (es) | 2000-11-22 | 2003-09-10 | Bayer Ag | Nuevos derivados de pirazolpiridina sustituidos con piridina |
JP2004515543A (ja) | 2000-12-11 | 2004-05-27 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 有害無脊椎動物を防除するためのキナゾリノン類およびピリジニルピリミジノン類 |
JP4405726B2 (ja) | 2000-12-21 | 2010-01-27 | ブリストル−マイヤーズ スクイブ カンパニー | Tecファミリーチロシンキナーゼのチアゾリルインヒビター |
DE10110750A1 (de) | 2001-03-07 | 2002-09-12 | Bayer Ag | Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften |
DE10110749A1 (de) | 2001-03-07 | 2002-09-12 | Bayer Ag | Substituierte Aminodicarbonsäurederivate |
DE10110747A1 (de) | 2001-03-07 | 2002-09-12 | Bayer Ag | Substituierte 2,6-Diamino-3,5-dicyano-4-aryl-pyridine und ihre Verwendung |
DE10134481A1 (de) | 2001-07-16 | 2003-01-30 | Bayer Ag | Substituierte 2-Thio-3,5-dicyano-4-phenyl-6-aminopyridine und ihre Verwendung |
DE10238113A1 (de) * | 2001-12-11 | 2003-06-18 | Bayer Ag | Substituierte 2-Thio-3,5-dicyano-4-phenyl-6-aminopyridine und ihre Verwendung |
JP2003183254A (ja) | 2001-12-20 | 2003-07-03 | Yamanouchi Pharmaceut Co Ltd | 2−アシルアミノ−3,5−ジシアノピリジン誘導体又はその塩 |
AU2003237121A1 (en) | 2002-04-26 | 2003-11-10 | Vertex Pharmaceuticals Incorporated | Pyrrole derivatives as inhibitors of erk2 and uses thereof |
DE10220570A1 (de) | 2002-05-08 | 2003-11-20 | Bayer Ag | Carbamat-substituierte Pyrazolopyridine |
EP1388342A1 (fr) | 2002-08-07 | 2004-02-11 | Aventis Pharma Deutschland GmbH | Dérivés de cycloalkenylamine condensé avec un hététoaryle et acylé et leur utilisation comme produits pharmaceutiques |
EP1545515A1 (fr) | 2002-08-12 | 2005-06-29 | Sugen, Inc. | 3-pyrrolyl-pyridopyrazoles et 3-pyrrolyl-indazoles utilises en tant que nouveaux inhibiteurs de la proteine kinase |
AU2003296414A1 (en) | 2002-12-12 | 2004-07-09 | Pharmacia Corporation | Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors |
AR042667A1 (es) | 2002-12-26 | 2005-06-29 | Taisho Pharmaceutical Co Ltd | Derivados de pirrolopirimidina y pirrolopiridina sustituidos con un grupo amino ciclico |
TW200418829A (en) | 2003-02-14 | 2004-10-01 | Avanir Pharmaceutics | Inhibitors of macrophage migration inhibitory factor and methods for identifying the same |
AR045047A1 (es) | 2003-07-11 | 2005-10-12 | Arena Pharm Inc | Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos |
JP4722851B2 (ja) | 2003-09-23 | 2011-07-13 | メルク・シャープ・エンド・ドーム・コーポレイション | キノリンカリウムチャネル阻害剤 |
US7338951B2 (en) | 2003-11-10 | 2008-03-04 | Synta Pharmaceuticals Corp. | Pyridine compounds |
US20050182105A1 (en) | 2004-02-04 | 2005-08-18 | Nirschl Alexandra A. | Method of using 3-cyano-4-arylpyridine derivatives as modulators of androgen receptor function |
JP2007161585A (ja) | 2004-06-25 | 2007-06-28 | Taisho Pharmaceut Co Ltd | 環状アミノ基で置換されているピロロピリミジン及びピロロピリジン誘導体 |
BRPI0512514A (pt) | 2004-06-25 | 2008-03-11 | Taisho Pharmaceutical Co Ltd | composto, antagonista para receptores de crf, e, uso de um composto |
DE102004032651A1 (de) * | 2004-07-06 | 2006-02-16 | Bayer Healthcare Ag | Verwendung von substituierten 2-Thio-3,5-dicyano-4-phenyl-6-aminopyriden bei der Behandlung von Übelkeit und Erbrechen |
BRPI0515499A (pt) | 2004-09-20 | 2008-07-29 | Xenon Pharmaceuticals Inc | derivados de piridina para a inibição de estearoil-coa-desaturase humana |
JP2008534453A (ja) | 2005-03-24 | 2008-08-28 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | 再灌流傷害および再灌流障害の処置のための置換2−チオ−3,5−ジシアノ−4−フェニル−6−アミノピリジンの使用 |
US7750015B2 (en) | 2005-05-17 | 2010-07-06 | Schering Corporation | Nitrogen-containing heterocyclic compounds and methods of use thereof |
DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
JP2009535307A (ja) | 2006-04-28 | 2009-10-01 | アベキサ・リミテッド | インテグラーゼ阻害剤3 |
WO2008008059A1 (fr) | 2006-07-12 | 2008-01-17 | Locus Pharmaceuticals, Inc. | Agents anti-cancer et leurs utilisations |
DE102006042143A1 (de) | 2006-09-08 | 2008-03-27 | Bayer Healthcare Aktiengesellschaft | Neue substituierte Bipyridin-Derivate und ihre Verwendung |
DE102006056740A1 (de) | 2006-12-01 | 2008-06-05 | Bayer Healthcare Ag | Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung |
DE102006056739A1 (de) | 2006-12-01 | 2008-06-05 | Bayer Healthcare Ag | Substituierte 4-Amino-3,5-dicyano-2-thiopyridine und ihre Verwendung |
JP2008266143A (ja) | 2007-04-16 | 2008-11-06 | Santen Pharmaceut Co Ltd | アデノシン誘導体を有効成分として含有する緑内障治療剤 |
DE102007035367A1 (de) | 2007-07-27 | 2009-01-29 | Bayer Healthcare Ag | Substituierte Aryloxazole und ihre Verwendung |
DE102007036075A1 (de) | 2007-08-01 | 2009-02-05 | Bayer Healthcare Ag | Prodrugs und ihre Verwendung |
DE102008013587A1 (de) | 2008-03-11 | 2009-09-17 | Bayer Schering Pharma Aktiengesellschaft | Heteroaryl-substituierte Dicyanopyridine und ihre Verwendung |
JP2011520997A (ja) | 2008-05-29 | 2011-07-21 | バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト | 2−アルコキシ置換ジシアノピリジン類およびそれらの使用 |
DE102008062567A1 (de) * | 2008-12-16 | 2010-06-17 | Bayer Schering Pharma Aktiengesellschaft | Dipeptoid-Prodrugs und ihre Verwendung |
DE102008062566A1 (de) | 2008-12-16 | 2010-06-17 | Bayer Schering Pharma Aktiengesellschaft | Aminosäureester-Prodrugs und ihre Verwendung |
DE102009006602A1 (de) * | 2009-01-29 | 2010-08-05 | Bayer Schering Pharma Aktiengesellschaft | Alkylamino-substituierte Dicyanopyridine und deren Aminosäureester-Prodrugs |
CN102413832B (zh) * | 2009-05-01 | 2015-11-25 | 伊诺泰克制药公司 | 降低人眼内压的方法 |
-
2011
- 2011-08-16 US US13/210,889 patent/US20120058983A1/en not_active Abandoned
- 2011-08-29 MA MA35698A patent/MA34489B1/fr unknown
- 2011-08-29 ES ES11752517T patent/ES2570659T3/es active Active
- 2011-08-29 PL PL11752517T patent/PL2611415T3/pl unknown
- 2011-08-29 HU HUE11752517A patent/HUE027295T2/en unknown
- 2011-08-29 MY MYPI2013700322A patent/MY160383A/en unknown
- 2011-08-29 WO PCT/EP2011/064829 patent/WO2012028585A1/fr active Application Filing
- 2011-08-29 BR BR112013005224A patent/BR112013005224A2/pt not_active IP Right Cessation
- 2011-08-29 EA EA201300310A patent/EA028411B1/ru not_active IP Right Cessation
- 2011-08-29 EP EP11752517.0A patent/EP2611415B1/fr active Active
- 2011-08-29 SG SG2013014691A patent/SG187974A1/en unknown
- 2011-08-29 CN CN201180052857.2A patent/CN103249400B/zh not_active Expired - Fee Related
- 2011-08-29 MX MX2013002396A patent/MX2013002396A/es active IP Right Grant
- 2011-08-29 SI SI201130809A patent/SI2611415T1/sl unknown
- 2011-08-29 KR KR1020137007797A patent/KR20140091457A/ko not_active Application Discontinuation
- 2011-08-29 CA CA2809700A patent/CA2809700A1/fr not_active Abandoned
- 2011-08-29 DK DK11752517.0T patent/DK2611415T3/en active
- 2011-08-29 AU AU2011298430A patent/AU2011298430B2/en not_active Ceased
- 2011-08-29 US US13/819,790 patent/US9040566B2/en not_active Expired - Fee Related
- 2011-08-29 RS RS20160304A patent/RS54743B1/sr unknown
- 2011-08-29 UA UAA201303837A patent/UA111947C2/uk unknown
- 2011-08-29 NZ NZ607624A patent/NZ607624A/en not_active IP Right Cessation
- 2011-08-29 AP AP2013006753A patent/AP3413A/xx active
- 2011-08-29 JP JP2013526433A patent/JP5875585B2/ja not_active Expired - Fee Related
- 2011-09-01 TW TW100131416A patent/TWI516266B/zh not_active IP Right Cessation
-
2013
- 2013-03-01 CL CL2013000599A patent/CL2013000599A1/es unknown
- 2013-03-04 CR CR20130094A patent/CR20130094A/es unknown
- 2013-03-28 ZA ZA2013/02340A patent/ZA201302340B/en unknown
-
2014
- 2014-02-12 HK HK14101303.4A patent/HK1188138A1/xx not_active IP Right Cessation
-
2015
- 2015-05-07 US US14/705,967 patent/US20150306084A1/en not_active Abandoned
-
2016
- 2016-05-05 CY CY20161100371T patent/CY1117458T1/el unknown
- 2016-05-13 CL CL2016001164A patent/CL2016001164A1/es unknown
- 2016-05-19 HR HRP20160532TT patent/HRP20160532T1/hr unknown
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102007036076A1 (de) * | 2007-08-01 | 2009-02-05 | Bayer Healthcare Aktiengesellschaft | Dipeptoid-Produgs und ihre Verwendung |
DE102008062561A1 (de) * | 2008-12-16 | 2010-06-24 | Maxon Motor Ag | Bausatz für einen Elektromotor mit einem Drehwinkelgeber |
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
HK1188138A1 (en) | Adenosine a1 agonists for the treatment of glaucoma and ocular hypertension a1 | |
HK1201042A1 (en) | Compositions for the treatment of dry eye | |
EP2303184A4 (fr) | Traitement d'association du glaucome | |
HK1200367A1 (en) | 4-pregenen-11ss-17-21-triol-3, 20-dione derivatives for the treatment of ocular conditions 4--11ss-17-21--320- | |
EP2654745A4 (fr) | Composition pour le traitement d'états pathologiques de la peau | |
ZA201303829B (en) | 2-piperazin-1-yl-4h-1,3-benzothiazin-4-one derivatives and their use for the treatment of mammalian infections | |
EP2515926A4 (fr) | Compositions et méthodes pour le traitement de maladies ophtalmiques liées à une angiogenèse | |
EP2563119A4 (fr) | Procédé et médicament pour la prévention et le traitement de l'hypertension oculaire et du glaucome | |
EP2623494A4 (fr) | Agent pour le traitement de maladies oculaires | |
PL2838417T3 (pl) | Urządzenie i sposób do nieinwazyjnego pomiaru stanu napięcia, biochemicznych i lepkosprężystych właściwości powierzchni biologicznych tkanek miękkich | |
IL236637A0 (en) | Difluorolactam compounds as selective ep4 receptor agonists for use in the treatment of ep4-mediated conditions and diseases | |
PL2538918T3 (pl) | Cytocholina do leczenia jaskry | |
IL250077A0 (en) | Lactam compounds as selective agonists for the ep4 receptor for use in the treatment of ep4-mediated diseases and conditions | |
IL230959B (en) | A device for the treatment of eye disease | |
EP2734188A4 (fr) | Compositions et procédés pour le traitement d'allergies de la surface oculaire | |
IL205774A0 (en) | Novel compounds for the treatment of glaucoma and ocular hypertension | |
PL2456445T3 (pl) | Środek do leczenia chorób skóry | |
IL221469A0 (en) | A3ar agonists for the treatment of uveitis | |
AU2012901278A0 (en) | Methods and compositions for reducing ocular discomfort | |
IL223055A0 (en) | Compositions for the treatment of gynaecological disorders | |
GB0911577D0 (en) | Compositions for the treatment of dry eye | |
GB0901727D0 (en) | The treatment of ophthalmic diseases |