AP2326A - Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors. - Google Patents

Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors.

Info

Publication number
AP2326A
AP2326A AP2007003905A AP2007003905A AP2326A AP 2326 A AP2326 A AP 2326A AP 2007003905 A AP2007003905 A AP 2007003905A AP 2007003905 A AP2007003905 A AP 2007003905A AP 2326 A AP2326 A AP 2326A
Authority
AP
ARIPO
Prior art keywords
kinase inhibitors
map kinase
triazolopyridinylsulfanyl
derivatives
triazolopyridinylsulfanyl derivatives
Prior art date
Application number
AP2007003905A
Other languages
English (en)
Other versions
AP2007003905A0 (en
Inventor
Russell Andrew Lewthwaite
John Paul Mathias
David Simon Millan
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0418015A external-priority patent/GB0418015D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of AP2007003905A0 publication Critical patent/AP2007003905A0/xx
Application granted granted Critical
Publication of AP2326A publication Critical patent/AP2326A/xx

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
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  • Virology (AREA)
  • Neurology (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
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  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
AP2007003905A 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors. AP2326A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0418015A GB0418015D0 (en) 2004-08-12 2004-08-12 New compounds
US69155905P 2005-06-17 2005-06-17
PCT/IB2005/002574 WO2006018718A2 (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors

Publications (2)

Publication Number Publication Date
AP2007003905A0 AP2007003905A0 (en) 2007-02-28
AP2326A true AP2326A (en) 2011-11-24

Family

ID=35783420

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2007003905A AP2326A (en) 2004-08-12 2005-08-09 Triazolopyridinylsulfanyl derivatives as p38 map kinase inhibitors.

Country Status (34)

Country Link
US (2) US7511057B2 (de)
EP (1) EP1778686B9 (de)
JP (1) JP4084836B2 (de)
AP (1) AP2326A (de)
AR (1) AR050692A1 (de)
AT (1) ATE412652T1 (de)
AU (1) AU2005273612B2 (de)
BR (1) BRPI0514255A (de)
CA (1) CA2576297C (de)
CR (1) CR8918A (de)
CU (1) CU23497A3 (de)
CY (1) CY1108788T1 (de)
DE (1) DE602005010714D1 (de)
DK (1) DK1778686T3 (de)
EA (1) EA012119B1 (de)
EC (1) ECSP077232A (de)
ES (1) ES2314690T3 (de)
GE (1) GEP20104973B (de)
GT (1) GT200500218A (de)
HN (1) HN2005000418A (de)
HR (1) HRP20080608T3 (de)
IL (1) IL181047A (de)
MA (1) MA28798B1 (de)
MX (1) MX2007001759A (de)
MY (1) MY140021A (de)
NL (1) NL1029726C2 (de)
NO (1) NO339320B1 (de)
NZ (1) NZ552868A (de)
PL (1) PL1778686T3 (de)
PT (1) PT1778686E (de)
SI (1) SI1778686T1 (de)
SV (1) SV2006002193A (de)
TN (1) TNSN07050A1 (de)
WO (1) WO2006018718A2 (de)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7572807B2 (en) * 2005-06-09 2009-08-11 Bristol-Myers Squibb Company Heteroaryl 11-beta-hydroxysteroid dehydrogenase type I inhibitors
US7579360B2 (en) * 2005-06-09 2009-08-25 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
EP1984363A1 (de) * 2006-02-09 2008-10-29 Pfizer Limited Triazolopyridinverbindungen
JP5244369B2 (ja) * 2006-11-10 2013-07-24 富士フイルム株式会社 ５−アミノピラゾール誘導体の製造方法、アゾ色素
EP1992344A1 (de) 2007-05-18 2008-11-19 Institut Curie P38 Alpha als therapeutisches Target für Erkrankungen, die mit einer FGFR3- Mutation assoziiert sind
US8119658B2 (en) * 2007-10-01 2012-02-21 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
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