ECSP066932A - Formas polimórficas de hidrobromuro acetato de metil(+)-(s)- alfa-(2-clorofenil)-6,7-dihidrotieno[3,2-c]piridina-5(4h), hidrobromuro de clopidogrel - Google Patents
Formas polimórficas de hidrobromuro acetato de metil(+)-(s)- alfa-(2-clorofenil)-6,7-dihidrotieno[3,2-c]piridina-5(4h), hidrobromuro de clopidogrelInfo
- Publication number
- ECSP066932A ECSP066932A EC2006006932A ECSP066932A ECSP066932A EC SP066932 A ECSP066932 A EC SP066932A EC 2006006932 A EC2006006932 A EC 2006006932A EC SP066932 A ECSP066932 A EC SP066932A EC SP066932 A ECSP066932 A EC SP066932A
- Authority
- EC
- Ecuador
- Prior art keywords
- hydrobromide
- chlorophenyl
- pyridine
- dihydrotiene
- alpha
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Abstract
La invención se refiere a las formas polimórficas B, C y D de acetato de hidrobromuro de metil(+)-(S)-a-(2-clorofenil)-6,7-dihidrotieno[3,2-C]piridina-5(4H), a las composiciones farmacéuticas que contienen el mismo y al método de utilización del mismo para inhibir la acumulación de plaquetas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US56379604P | 2004-04-20 | 2004-04-20 | |
PCT/US2005/013146 WO2005103058A1 (en) | 2004-04-20 | 2005-04-18 | Polymorphic forms of methyl (+) - (s) -alpha- (2-chlorophenyl) -6, 7-dihydrothieno `3,2-c!pyridine-584h) acetate hydrobromide, clopidrogel hydrobromide |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP066932A true ECSP066932A (es) | 2006-12-20 |
Family
ID=34966201
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2006006932A ECSP066932A (es) | 2004-04-20 | 2006-10-17 | Formas polimórficas de hidrobromuro acetato de metil(+)-(s)- alfa-(2-clorofenil)-6,7-dihidrotieno[3,2-c]piridina-5(4h), hidrobromuro de clopidogrel |
Country Status (20)
Country | Link |
---|---|
US (1) | US20070088049A1 (es) |
EP (1) | EP1756116A1 (es) |
JP (1) | JP2007533744A (es) |
KR (1) | KR20070012675A (es) |
CN (1) | CN1997648A (es) |
AU (1) | AU2005236034A1 (es) |
BR (1) | BRPI0509997A (es) |
CA (1) | CA2562507A1 (es) |
CR (1) | CR8678A (es) |
EA (1) | EA010831B1 (es) |
EC (1) | ECSP066932A (es) |
IL (1) | IL178680A0 (es) |
MA (1) | MA28588B1 (es) |
MX (1) | MXPA06012205A (es) |
NO (1) | NO20065233L (es) |
NZ (1) | NZ551371A (es) |
TN (1) | TNSN06331A1 (es) |
UA (1) | UA83919C2 (es) |
WO (1) | WO2005103058A1 (es) |
ZA (1) | ZA200608569B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0321256D0 (en) | 2003-09-11 | 2003-10-08 | Generics Uk Ltd | Novel crystalline compounds |
WO2006034451A2 (en) * | 2004-09-21 | 2006-03-30 | Teva Pharmaceutical Industries Ltd. | Crystalline clopidogrel hydrobromide and processes for preparation thereof |
SI22492A (sl) * | 2007-03-08 | 2008-10-31 | Krka, Tovarna Zdravil, D.D., Novo Mesto | Polimorfne oblike klopidogrel hidrobromida |
UY31531A1 (es) * | 2007-12-17 | 2009-08-03 | Sales derivadas de 8-oxoadenina composiciones farmacéuticas que las contienen y su uso en terapia como moduladores de receptor tipo toll (tlr) | |
ATE530172T1 (de) | 2008-02-26 | 2011-11-15 | Lesvi Laboratorios Sl | Pharmazeutische formulierungen mit clopidogrel |
HUP1400294A2 (hu) | 2014-06-13 | 2015-12-28 | Skillpharm Kft | Clopidogrel új alkalmazása |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2623810B2 (fr) * | 1987-02-17 | 1992-01-24 | Sanofi Sa | Sels de l'alpha-(tetrahydro-4,5,6,7 thieno(3,2-c) pyridyl-5) (chloro-2 phenyl) -acetate de methyle dextrogyre et compositions pharmaceutiques en contenant |
FR2779726B1 (fr) * | 1998-06-15 | 2001-05-18 | Sanofi Sa | Forme polymorphe de l'hydrogenosulfate de clopidogrel |
AU1816901A (en) * | 1999-12-06 | 2001-06-12 | Euro-Celtique S.A. | Benzimidazole compounds having nociceptin receptor affinity |
CA2470479A1 (en) * | 2001-12-18 | 2003-06-26 | Teva Pharmaceutical Industries Ltd. | Polymorphs of clopidogrel hydrogensulfate |
US7074928B2 (en) * | 2002-01-11 | 2006-07-11 | Teva Pharmaceutical Industries, Ltd. | Polymorphs of clopidogrel hydrogensulfate |
HUP0200438A3 (en) * | 2002-02-06 | 2003-10-28 | Egis Gyogyszergyar Nyilvanosan | Novel clopidogrel hydrochloride polymorphs, process for the preparation thereof, their use and pharmaceutical compositions containing them |
CZ297472B6 (cs) * | 2002-08-27 | 2006-12-13 | Zentiva, A.S. | Zpusob výroby clopidogrelu hydrogensulfátu krystalické formy I |
DE10305984A1 (de) * | 2003-02-13 | 2004-09-02 | Helm Ag | Salze organischer Säuren mit Clopidogrel und deren Verwendung zur Herstellung phamazeutischer Formulierungen |
GB0321256D0 (en) * | 2003-09-11 | 2003-10-08 | Generics Uk Ltd | Novel crystalline compounds |
GB0325603D0 (en) * | 2003-11-03 | 2003-12-10 | Sandoz Ag | Organic compounds |
EA008972B1 (ru) * | 2004-01-13 | 2007-10-26 | Зентива А.С. | Новые кристаллические формы гидробромида клопидогреля и способы их получения |
RU2006133842A (ru) * | 2004-02-24 | 2008-03-27 | Зигфрид Дженерикс Интерэшнл Аг (Ch) | Фармакологически приемлемые соли клопидогрела |
-
2005
- 2005-04-18 KR KR1020067021700A patent/KR20070012675A/ko not_active Application Discontinuation
- 2005-04-18 CA CA002562507A patent/CA2562507A1/en not_active Abandoned
- 2005-04-18 ZA ZA200608569A patent/ZA200608569B/xx unknown
- 2005-04-18 WO PCT/US2005/013146 patent/WO2005103058A1/en active Application Filing
- 2005-04-18 JP JP2007509543A patent/JP2007533744A/ja active Pending
- 2005-04-18 NZ NZ551371A patent/NZ551371A/en unknown
- 2005-04-18 AU AU2005236034A patent/AU2005236034A1/en not_active Abandoned
- 2005-04-18 MX MXPA06012205A patent/MXPA06012205A/es not_active Application Discontinuation
- 2005-04-18 UA UAA200612105A patent/UA83919C2/ru unknown
- 2005-04-18 BR BRPI0509997-8A patent/BRPI0509997A/pt not_active IP Right Cessation
- 2005-04-18 CN CNA2005800118591A patent/CN1997648A/zh active Pending
- 2005-04-18 EA EA200601921A patent/EA010831B1/ru not_active IP Right Cessation
- 2005-04-18 EP EP05736220A patent/EP1756116A1/en not_active Withdrawn
-
2006
- 2006-10-09 CR CR8678A patent/CR8678A/es not_active Application Discontinuation
- 2006-10-13 TN TNP2006000331A patent/TNSN06331A1/en unknown
- 2006-10-17 EC EC2006006932A patent/ECSP066932A/es unknown
- 2006-10-17 IL IL178680A patent/IL178680A0/en unknown
- 2006-10-19 US US11/550,891 patent/US20070088049A1/en not_active Abandoned
- 2006-11-14 NO NO20065233A patent/NO20065233L/no not_active Application Discontinuation
- 2006-11-20 MA MA29464A patent/MA28588B1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
KR20070012675A (ko) | 2007-01-26 |
BRPI0509997A (pt) | 2007-10-16 |
NZ551371A (en) | 2010-07-30 |
EA010831B1 (ru) | 2008-12-30 |
WO2005103058A1 (en) | 2005-11-03 |
CR8678A (es) | 2007-08-28 |
MXPA06012205A (es) | 2007-01-31 |
CA2562507A1 (en) | 2005-11-03 |
NO20065233L (no) | 2006-11-14 |
TNSN06331A1 (en) | 2008-02-22 |
IL178680A0 (en) | 2007-02-11 |
JP2007533744A (ja) | 2007-11-22 |
UA83919C2 (en) | 2008-08-26 |
EA200601921A1 (ru) | 2007-02-27 |
US20070088049A1 (en) | 2007-04-19 |
ZA200608569B (en) | 2007-12-27 |
MA28588B1 (fr) | 2007-05-02 |
CN1997648A (zh) | 2007-07-11 |
AU2005236034A1 (en) | 2005-11-03 |
EP1756116A1 (en) | 2007-02-28 |
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