ZA957794B - [1.2.4]triazolo[4,3-a]quinoxalinone derivatives their preparation and use - Google Patents

[1.2.4]triazolo[4,3-a]quinoxalinone derivatives their preparation and use

Info

Publication number
ZA957794B
ZA957794B ZA957794A ZA957794A ZA957794B ZA 957794 B ZA957794 B ZA 957794B ZA 957794 A ZA957794 A ZA 957794A ZA 957794 A ZA957794 A ZA 957794A ZA 957794 B ZA957794 B ZA 957794B
Authority
ZA
South Africa
Prior art keywords
alkyl
triazolo
independently
preparation
pox
Prior art date
Application number
ZA957794A
Other languages
English (en)
Inventor
Flemming Elmelund Nielsen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of ZA957794B publication Critical patent/ZA957794B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Otolaryngology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ZA957794A 1994-09-16 1995-09-15 [1.2.4]triazolo[4,3-a]quinoxalinone derivatives their preparation and use ZA957794B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK106694 1994-09-16

Publications (1)

Publication Number Publication Date
ZA957794B true ZA957794B (en) 1996-05-14

Family

ID=8100607

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA957794A ZA957794B (en) 1994-09-16 1995-09-15 [1.2.4]triazolo[4,3-a]quinoxalinone derivatives their preparation and use

Country Status (22)

Country Link
EP (1) EP0781282B1 (cs)
JP (1) JPH10506620A (cs)
KR (1) KR970706285A (cs)
CN (1) CN1193973A (cs)
AT (1) ATE183186T1 (cs)
AU (1) AU694554B2 (cs)
CA (1) CA2200056A1 (cs)
CZ (1) CZ284930B6 (cs)
DE (1) DE69511420T2 (cs)
DK (1) DK0781282T3 (cs)
ES (1) ES2138233T3 (cs)
FI (1) FI971076L (cs)
GR (1) GR3031788T3 (cs)
HU (1) HUT76802A (cs)
IL (1) IL115299A0 (cs)
NO (1) NO308797B1 (cs)
NZ (1) NZ292108A (cs)
PL (1) PL319175A1 (cs)
SK (1) SK282457B6 (cs)
TW (1) TW397835B (cs)
WO (1) WO1996008493A1 (cs)
ZA (1) ZA957794B (cs)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL125950A0 (en) * 1997-09-05 1999-04-11 Pfizer Prod Inc Methods of administering ampa receptor antagonists to treat dyskinesias associated with dopamine agonist therapy
TR200001728T2 (tr) 1997-11-11 2000-09-21 Ono Pharmaceutical Co., Ltd. Birleşik pirazin türevleri
CA2754457A1 (en) 2009-03-05 2010-09-10 Astellas Pharma Inc. Quinoxaline compounds
KR20130097178A (ko) 2010-09-07 2013-09-02 아스텔라스세이야쿠 가부시키가이샤 퀴녹살린 화합물

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4354027A (en) * 1980-05-19 1982-10-12 Usv Pharmaceutical Corporation Triazoloquinoxalin-4-ones
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof
DK162491D0 (da) * 1991-09-20 1991-09-20 Novo Nordisk As Heterocycliske forbindelser, deres fremstilling og farmaceutiske praeparater indeholdende forbindelserne
AU3767793A (en) * 1992-04-03 1993-11-08 Yamanouchi Pharmaceutical Co., Ltd. Fused quinoxalinone derivative and pharmaceutical composition containing the same
DK31093D0 (cs) * 1993-03-19 1993-03-19 Novo Nordisk As
EP0698024B1 (en) * 1993-05-06 1997-01-22 Novo Nordisk A/S [1,2,4]TRIAZOLO [4,3-a]QUINOXALINE COMPOUNDS, THEIR PREPARATION AND USE

Also Published As

Publication number Publication date
DE69511420D1 (de) 1999-09-16
IL115299A0 (en) 1995-12-31
EP0781282A1 (en) 1997-07-02
JPH10506620A (ja) 1998-06-30
CN1193973A (zh) 1998-09-23
KR970706285A (ko) 1997-11-03
NO971187D0 (no) 1997-03-14
AU694554B2 (en) 1998-07-23
FI971076A7 (fi) 1997-05-13
WO1996008493A1 (en) 1996-03-21
ES2138233T3 (es) 2000-01-01
TW397835B (en) 2000-07-11
SK282457B6 (sk) 2002-02-05
DK0781282T3 (da) 2000-02-28
SK33497A3 (en) 1998-02-04
NZ292108A (en) 1999-02-25
HUT76802A (en) 1997-11-28
DE69511420T2 (de) 2000-03-30
GR3031788T3 (en) 2000-02-29
NO308797B1 (no) 2000-10-30
NO971187L (no) 1997-05-15
FI971076A0 (fi) 1997-03-14
AU3380895A (en) 1996-03-29
CA2200056A1 (en) 1996-03-21
CZ284930B6 (cs) 1999-04-14
FI971076L (fi) 1997-05-13
PL319175A1 (en) 1997-08-04
ATE183186T1 (de) 1999-08-15
EP0781282B1 (en) 1999-08-11
CZ75397A3 (en) 1997-08-13

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