ZA911728B - Benzisothiazolinone-1-dioxide derivatives as elastase inhibitors - Google Patents

Benzisothiazolinone-1-dioxide derivatives as elastase inhibitors

Info

Publication number
ZA911728B
ZA911728B ZA911728A ZA911728A ZA911728B ZA 911728 B ZA911728 B ZA 911728B ZA 911728 A ZA911728 A ZA 911728A ZA 911728 A ZA911728 A ZA 911728A ZA 911728 B ZA911728 B ZA 911728B
Authority
ZA
South Africa
Prior art keywords
benzisothiazolinone
compositions
elastase inhibitors
chem
dioxide derivatives
Prior art date
Application number
ZA911728A
Other languages
English (en)
Inventor
Ladislas Robert
Robert Ladislas
Elemer Moczar
Moczar Elemer
William Georges Homebeck
Georges Homebeck William
Christiane Marie-Pierr Kerneur
Marie-Pierre Kerneu Christiane
Original Assignee
Unilever Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Unilever Plc filed Critical Unilever Plc
Publication of ZA911728B publication Critical patent/ZA911728B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/08Anti-ageing preparations
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/74Biological properties of particular ingredients
    • A61K2800/78Enzyme modulators, e.g. Enzyme agonists
    • A61K2800/782Enzyme inhibitors; Enzyme antagonists
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00Preparations for care of the hair

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Gerontology & Geriatric Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
ZA911728A 1990-03-08 1991-03-08 Benzisothiazolinone-1-dioxide derivatives as elastase inhibitors ZA911728B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9002951A FR2659327A1 (fr) 1990-03-08 1990-03-08 Derives du benzisothiazolinone-1-dioxyde, utilisables comme inhibiteurs des elastases.

Publications (1)

Publication Number Publication Date
ZA911728B true ZA911728B (en) 1992-11-25

Family

ID=9394523

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA911728A ZA911728B (en) 1990-03-08 1991-03-08 Benzisothiazolinone-1-dioxide derivatives as elastase inhibitors

Country Status (16)

Country Link
US (2) US5338747A (ko)
EP (1) EP0446047B1 (ko)
JP (1) JPH04234863A (ko)
KR (1) KR960014782B1 (ko)
AT (1) ATE154347T1 (ko)
AU (1) AU636013B2 (ko)
BR (1) BR9100938A (ko)
CA (1) CA2037665A1 (ko)
DE (1) DE69126460T2 (ko)
ES (1) ES2102994T3 (ko)
FR (1) FR2659327A1 (ko)
ID (1) ID820B (ko)
IN (1) IN172035B (ko)
MY (1) MY106067A (ko)
TW (1) TW200472B (ko)
ZA (1) ZA911728B (ko)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5306818A (en) * 1990-11-01 1994-04-26 Sterling Winthrop Inc. Tetrahydro 2-saccharinylmerthyl aryl carboxylates
US5512589A (en) * 1990-11-01 1996-04-30 Sterling Winthrop Inc. 2-saccharinylmethyl aryl carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof
US5250696A (en) * 1990-11-01 1993-10-05 Sterling Winthrop Inc. 2-saccharinylmethyl aryl carboxylate
TW226016B (ko) * 1991-12-30 1994-07-01 Sterling Winthrop Inc
AU653279B2 (en) * 1991-12-30 1994-09-22 Sanofi Novel 2-saccharinylmethyl heterocyclic carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof
US6375948B1 (en) 1999-07-12 2002-04-23 Kao Corporation Treating method for suppressing hair growth
GB0129987D0 (en) * 2001-12-14 2002-02-06 Zylepsis Ltd Skin compositions
US7169933B2 (en) * 2003-11-14 2007-01-30 3M Innovative Properties Company N-sulfonylaminocarbonyl containing compounds
US7361767B2 (en) 2003-11-14 2008-04-22 3M Innovative Properties Company N-sulfonyldicarboximide containing tethering compounds
WO2005049590A2 (en) * 2003-11-14 2005-06-02 3M Innovative Properties Company N-sulfonylaminocarbonyl containing compounds
US7423155B2 (en) 2003-11-14 2008-09-09 3M Innovative Properties Company N-sulfonyldicarboximide containing tethering compounds
US7943388B2 (en) 2003-11-14 2011-05-17 3M Innovative Properties Company Acoustic sensors and methods
US7402678B2 (en) 2004-12-17 2008-07-22 3M Innovative Properties Company Multifunctional amine capture agents
US7342082B2 (en) 2004-12-17 2008-03-11 3M Innovative Properties Company Soluble polymers as amine capture agents and methods
WO2005066121A2 (en) * 2003-12-30 2005-07-21 3M Innovative Properties Company Multifunctional amine capture agents
US7544756B2 (en) 2005-09-30 2009-06-09 3M Innovative Properties Company Crosslinked polymers with amine binding groups
US7544755B2 (en) 2005-09-30 2009-06-09 3M Innovative Properties Company Crosslinked polymers with amine binding groups
US7544754B2 (en) * 2005-09-30 2009-06-09 3M Innovative Properties Company Crosslinked polymers with amine binding groups
US8034448B2 (en) * 2008-08-19 2011-10-11 Los Alamos National Security, Llc Fibrous composites comprising carbon nanotubes and silica
AR079232A1 (es) 2009-12-01 2012-01-04 Lubrizol Advanced Mat Inc Polimeros multiproposito estables hidroliticamente
WO2018049324A1 (en) * 2016-09-12 2018-03-15 Numerate, Inc. Monocyclic compounds useful as gpr120 modulators
US10865201B2 (en) 2016-09-12 2020-12-15 Valo Health, Inc. Bicyclic compounds useful as GPR120 modulators

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4195023A (en) * 1975-08-20 1980-03-25 Merck & Co., Inc. 2-(2-Furoyl)1,2-benzisothiazole-3-one, 2-(2-furoyl) saccharin, and 2-(2-thenoyl) saccharin
US4276298A (en) * 1978-03-24 1981-06-30 Merck & Co., Inc. 2-Aryl-1,2-benzisothiazolinone-1,1-dioxides and their use as selective protease inhibitors
FR2546164B1 (fr) * 1983-05-16 1987-07-17 Centre Nat Rech Scient Nouveaux derives de peptides, leur preparation et leur application comme inhibiteurs de l'elastase

Also Published As

Publication number Publication date
KR910016330A (ko) 1991-11-05
MY106067A (en) 1995-03-31
IN172035B (ko) 1993-03-20
DE69126460D1 (de) 1997-07-17
FR2659327A1 (fr) 1991-09-13
EP0446047A1 (en) 1991-09-11
AU7263591A (en) 1991-09-12
US5411978A (en) 1995-05-02
KR960014782B1 (en) 1996-10-19
ATE154347T1 (de) 1997-06-15
ID820B (id) 1996-07-22
DE69126460T2 (de) 1997-12-04
BR9100938A (pt) 1991-11-05
JPH04234863A (ja) 1992-08-24
ES2102994T3 (es) 1997-08-16
TW200472B (ko) 1993-02-21
EP0446047B1 (en) 1997-06-11
US5338747A (en) 1994-08-16
AU636013B2 (en) 1993-04-08
CA2037665A1 (en) 1991-09-09

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