ZA845682B - Benzamidine derivatives having an antimicrobial activity process for their preparation and use as disinfectant drugs or preservatives - Google Patents

Benzamidine derivatives having an antimicrobial activity process for their preparation and use as disinfectant drugs or preservatives

Info

Publication number
ZA845682B
ZA845682B ZA845682A ZA845682A ZA845682B ZA 845682 B ZA845682 B ZA 845682B ZA 845682 A ZA845682 A ZA 845682A ZA 845682 A ZA845682 A ZA 845682A ZA 845682 B ZA845682 B ZA 845682B
Authority
ZA
South Africa
Prior art keywords
preservatives
preparation
antimicrobial activity
activity process
benzamidine derivatives
Prior art date
Application number
ZA845682A
Other languages
English (en)
Inventor
Madeleine Mosse
Henri Demarne
Robert Filhol
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of ZA845682B publication Critical patent/ZA845682B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C257/00—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
    • C07C257/10—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
    • C07C257/18—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having carbon atoms of amidino groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/13—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups
    • C07C205/19—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups bound to carbon atoms of six-membered aromatic rings and hydroxy groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/27—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups
    • C07C205/35—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/36—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system
    • C07C205/37—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/18—Monohydroxylic alcohols containing only six-membered aromatic rings as cyclic part
    • C07C33/20—Monohydroxylic alcohols containing only six-membered aromatic rings as cyclic part monocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/30—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing six-membered aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Cosmetics (AREA)
ZA845682A 1983-08-03 1984-07-23 Benzamidine derivatives having an antimicrobial activity process for their preparation and use as disinfectant drugs or preservatives ZA845682B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8312824A FR2550192B1 (fr) 1983-08-03 1983-08-03 Nouveaux derives de la benzamidine a activite antimicrobienne, leur procede de preparation, leur utilisation en tant que medicaments desinfectants ou conservateurs

Publications (1)

Publication Number Publication Date
ZA845682B true ZA845682B (en) 1985-02-27

Family

ID=9291379

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA845682A ZA845682B (en) 1983-08-03 1984-07-23 Benzamidine derivatives having an antimicrobial activity process for their preparation and use as disinfectant drugs or preservatives

Country Status (25)

Country Link
US (1) US4720581A (fi)
EP (1) EP0136195B1 (fi)
JP (1) JPS6054351A (fi)
KR (1) KR920000373B1 (fi)
AR (1) AR242556A1 (fi)
AT (1) ATE27952T1 (fi)
AU (1) AU563648B2 (fi)
CA (1) CA1238922A (fi)
CS (1) CS246088B2 (fi)
DD (1) DD220025A5 (fi)
DE (1) DE3464362D1 (fi)
DK (1) DK158662C (fi)
ES (1) ES534828A0 (fi)
FI (1) FI77020C (fi)
FR (1) FR2550192B1 (fi)
GR (1) GR82449B (fi)
HU (1) HU192567B (fi)
IL (1) IL72480A (fi)
MA (1) MA20180A1 (fi)
NO (1) NO157618C (fi)
NZ (1) NZ209092A (fi)
PT (1) PT79003B (fi)
SU (1) SU1319784A3 (fi)
YU (1) YU127684A (fi)
ZA (1) ZA845682B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2504361Y2 (ja) * 1990-12-14 1996-07-10 大和ハウス工業株式会社 建物の配管固定構造
DE4447361A1 (de) * 1994-12-21 1996-06-27 Schuelke & Mayr Gmbh Biozide Alkohole, ihre Herstellung und ihre Verwendung
EP2444393A1 (en) * 2003-02-19 2012-04-25 Eisai R&D Management Co., Ltd. Methods for producing cyclic benzamidine derivatives
EP1773794A4 (en) * 2004-07-05 2009-09-09 Dong Wha Pharm Ind Co Ltd IMPROVED METHOD FOR PREPARING N-HYDROXY-4 {5- [4- (5-ISOPROPYL-2-METHYL-1,3-THIAZOL-4-YL) -PHENOXY] -PENTOXY} -BENZAMIDINE
CN111362834B (zh) * 2020-02-26 2021-04-02 湖南大学 一种具有抗耐药性的抗菌脒类低聚物及其制作方法和用途
CN113754564B (zh) * 2021-08-02 2022-08-26 湖南大学 具有抗耐药性的抗菌脒类低聚物及其制作方法和用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2934438A (en) * 1958-03-20 1960-04-26 Michener Harold David Preservation process with alkyl guanidines
US3769427A (en) * 1970-10-01 1973-10-30 Armour Pharma Pharmaceutical compositions and methods of using same
IT1153988B (it) * 1981-10-05 1987-01-21 Medea Res Srl Composizioni ad attivita' antimicrobica

Also Published As

Publication number Publication date
JPS6054351A (ja) 1985-03-28
SU1319784A3 (ru) 1987-06-23
NO157618B (no) 1988-01-11
CS246088B2 (en) 1986-10-16
YU127684A (en) 1986-12-31
FR2550192B1 (fr) 1986-04-04
FI843061A0 (fi) 1984-08-02
NZ209092A (en) 1987-03-06
DE3464362D1 (en) 1987-07-30
ES8504112A1 (es) 1985-04-16
AU3079084A (en) 1985-02-07
CS584184A2 (en) 1985-12-16
ATE27952T1 (de) 1987-07-15
EP0136195A1 (fr) 1985-04-03
GR82449B (fi) 1984-12-13
AR242556A1 (es) 1993-04-30
DK158662C (da) 1990-12-10
NO157618C (no) 1988-04-20
CA1238922A (en) 1988-07-05
DD220025A5 (de) 1985-03-20
FI77020B (fi) 1988-09-30
FI77020C (fi) 1989-01-10
NO843114L (no) 1985-02-04
KR920000373B1 (ko) 1992-01-13
IL72480A0 (en) 1984-11-30
DK362384A (da) 1985-02-04
MA20180A1 (fr) 1985-04-01
US4720581A (en) 1988-01-19
HU192567B (en) 1987-06-29
AU563648B2 (en) 1987-07-16
EP0136195B1 (fr) 1987-06-24
FI843061A (fi) 1985-02-04
PT79003B (fr) 1986-06-18
ES534828A0 (es) 1985-04-16
PT79003A (fr) 1984-08-01
DK362384D0 (da) 1984-07-24
KR850001730A (ko) 1985-04-01
IL72480A (en) 1987-10-30
DK158662B (da) 1990-07-02
HUT34724A (en) 1985-04-28
FR2550192A1 (fr) 1985-02-08

Similar Documents

Publication Publication Date Title
HK128797A (en) 7-piperazinyl-or 7-morpholino-4-oxo-quinoline-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents
IT8467767A0 (it) Preparati farmaceutici ad attivita antimicrobica e procedimento per laloro preparazione
IL87866A0 (en) 2-anilinopyrimidine derivatives,their preparation and their use as pesticides
HUT45850A (en) Insecticides comprising azolinone derivatives as active ingredient and process for producing the active ingredients
HUT48605A (en) Fungicides comprising hydroxyalkylazolyl derivatives as active ingredient and process for producing the active ingredient
AU2302288A (en) 4-quinoline-3-carboxylic acid derivatives and their use as antibacterial agents
EP0238060A3 (en) Cephalosporin derivatives, processes for their preparation and antibacterial agents
AU591046B2 (en) Physiologically active agent for agricultural use
HUT47233A (en) Process for producing pharmaceutical comprising phenol derivatives as active ingredient and for producing the active ingredients
PT78049A (en) Biologically active ketone derivative preparation and use
ZA845682B (en) Benzamidine derivatives having an antimicrobial activity process for their preparation and use as disinfectant drugs or preservatives
IL81990A0 (en) Compounds and pharmaceutical preparations having calcium regulatory activity
AU5668286A (en) Carbohydrate derivatives and compositions thereof for therapeutic or diagnostic use, and methods for their use
EP0287471A3 (en) Carboxystyrene derivatives and drugs containing them as effective ingredients
HU9201358D0 (en) 2-amino-pirimidine-4-carboxamide derivatives, process for their production and for the production of medical preparations containing them as active agents
HUT43318A (en) Fungicides comprising 2-cyano-benzimidazole derivatives as active substance and process for preparing the active substances
GB2105329B (en) Penem-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents
IL88393A0 (en) Imidiates,their preparation and their use as insecticides
HUT48606A (en) Fungicides comprising hydroxyalkyltriazolyl derivatives as active ingredient and process for producing the active ingredients
ZA885329B (en) Hydroxyethylazole derivatives and their use as fungicides
ZW15489A1 (en) New antimicrobial phenazine derivatives,method for their preparation,compositions containing them,and their use in therapy
HUT46641A (en) Fungicides comprising propargyl-oxy-benzene derivatives as active ingredient and process for producing the active ingredients
IL70758A (en) 3-acyl-2-nitromethylenetetrahydro-2h-1,3-thiazine derivatives,their preparation and their use as insecticides
ZA849442B (en) Sphingosine derivatives,their preparation and pharmaceutical formulation
HUT44240A (en) Pesticide comprising pyrazolin-5-one derivatives as active substance and process for preparing the pyrazolin-5-one derivatives