ZA200601898B - Process for preparing water soluble diterpenes and their applications - Google Patents

Process for preparing water soluble diterpenes and their applications

Info

Publication number
ZA200601898B
ZA200601898B ZA200601898A ZA200601898A ZA200601898B ZA 200601898 B ZA200601898 B ZA 200601898B ZA 200601898 A ZA200601898 A ZA 200601898A ZA 200601898 A ZA200601898 A ZA 200601898A ZA 200601898 B ZA200601898 B ZA 200601898B
Authority
ZA
South Africa
Prior art keywords
applications
water soluble
preparing water
diterpenes
soluble diterpenes
Prior art date
Application number
ZA200601898A
Other languages
English (en)
Inventor
Majeed Muhammed
Kumar Arvind
Nagabhushanam Kalyanam
Prakash Subbalakshmi
Original Assignee
Majeed Muhammed
Kumar Arvind
Nagabhushanam Kalyanam
Prakash Subbalakshmi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Majeed Muhammed, Kumar Arvind, Nagabhushanam Kalyanam, Prakash Subbalakshmi filed Critical Majeed Muhammed
Publication of ZA200601898B publication Critical patent/ZA200601898B/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23L—FOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/10—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
    • A23L33/105—Plant extracts, their artificial duplicates or their derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40—Cyclodextrins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/04—Artificial tears; Irrigation solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A61P39/06—Free radical scavengers or antioxidants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/92—Naphthopyrans; Hydrogenated naphthopyrans
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23V—INDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2002/00—Food compositions, function of food ingredients or processes for food or foodstuffs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Food Science & Technology (AREA)
  • Botany (AREA)
  • Inorganic Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Nutrition Science (AREA)
  • Mycology (AREA)
  • Toxicology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Transplantation (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)
  • Pyrane Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
ZA200601898A 2003-09-08 2006-03-06 Process for preparing water soluble diterpenes and their applications ZA200601898B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10/605,086 US6960300B2 (en) 2003-09-08 2003-09-08 Process for preparing water soluble diterpenes and their applications

Publications (1)

Publication Number Publication Date
ZA200601898B true ZA200601898B (en) 2008-09-25

Family

ID=34225859

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200601898A ZA200601898B (en) 2003-09-08 2006-03-06 Process for preparing water soluble diterpenes and their applications

Country Status (14)

Country Link
US (2) US6960300B2 (zh)
EP (1) EP1718568B1 (zh)
JP (1) JP5021305B2 (zh)
CN (1) CN1882508B (zh)
AU (1) AU2004272005B2 (zh)
BR (1) BRPI0413957A (zh)
CA (1) CA2537820C (zh)
EA (1) EA012836B1 (zh)
HK (1) HK1098450A1 (zh)
MX (1) MXPA06002684A (zh)
NZ (1) NZ545765A (zh)
RS (1) RS20060169A (zh)
WO (1) WO2005025500A2 (zh)
ZA (1) ZA200601898B (zh)

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US20060122261A1 (en) * 2003-11-20 2006-06-08 Muhammed Majeed [method of preparing labdane diterpene composition, preferably isoforskolin and deacetylforskolin from forskolin extract and their use for promoting lean body mass and other applications]
US20110077292A1 (en) * 2004-07-01 2011-03-31 Biotest Laboratories, Llc. Forskolin carbonates and uses thereof
JP2007210988A (ja) * 2006-02-07 2007-08-23 Sabinsa Corp ジテルペンフォルスコリン及びその誘導体で男性ホルモン及び女性ホルモンを生理学的に増大するための組成物
WO2007108727A1 (en) * 2006-03-22 2007-09-27 Leangene Ab Method for monitoring the effect of compounds on foxc2 expression
US20080226571A1 (en) * 2007-03-16 2008-09-18 Muhammed Majeed Compositions and methods to effect enhanced photoprotection against UV A and UV B induced damage of human skin
US20080241285A1 (en) * 2007-04-01 2008-10-02 Muhammed Majeed Compositions and Methods to Treat Alopecia
WO2009110009A2 (en) * 2008-03-07 2009-09-11 Sun Pharma Advanced Research Company Ltd., Opthalmic composition
US20100076069A1 (en) * 2008-09-22 2010-03-25 Muhammed Majeed Forskolin dosing regimen in open angle glaucoma and patient compliance methods thereof
US8975241B2 (en) * 2009-10-08 2015-03-10 Song Ho Biomed Co., Ltd. Composition for treating and preventing obesity including high water-soluble 2-hydroxypropyl-betacyclodextrin as effective component
EP2496080A4 (en) * 2009-11-02 2013-05-15 Nupathe Inc METHOD FOR THE TREATMENT OF MORBUS PARKINSON
AU2011340203B2 (en) * 2010-12-09 2015-11-26 Indus Biotech Private Limited A complex of Garcinol, Cyclodextrin and method thereof
CN103588745B (zh) * 2013-11-26 2015-10-28 陕西嘉禾植物化工有限责任公司 一种从毛喉鞘蕊花中提取和分离弗斯可林的方法
WO2017103840A1 (en) * 2015-12-16 2017-06-22 MOHAMED ABDULLA ANZAR, Cheppattu A water soluble 10% w/w forskolin composition and a method of synthesizing the same
US11045444B2 (en) 2016-06-30 2021-06-29 Plume Cosmetics Inc. Composition and method for promoting eyelash and eyebrow growth exclusively containing naturally sourced ingredients
RS61915B1 (sr) * 2017-01-09 2021-06-30 Scipharm S A R L Novi postupak za pripremu forskolina rastvorljivog u vodi
WO2018235939A1 (ja) * 2017-06-23 2018-12-27 Ｔｋヘルスリサーチ株式会社 包接化された抗酸化物質を含む眼科用組成物ならびにその使用
JP7004968B2 (ja) 2017-10-06 2022-01-21 青葉化成株式会社 食用の徐放性機能材の製造方法
CN108651819A (zh) * 2018-05-18 2018-10-16 南昌大学 一种稳定态全谷物超微粉速食粉的制备方法
JP7130110B2 (ja) * 2019-03-01 2022-09-02 長谷川香料株式会社 セスキテルペン酸素付加体の製造方法、化合物および組成物
WO2020186235A1 (en) 2019-03-14 2020-09-17 The Broad Institute, Inc. Compositions and methods for modulating cgrp signaling to regulate intestinal innate lymphoid cells
JP2023511432A (ja) 2020-01-23 2023-03-17 サイファーム ソシエテ ア レスポンサビリテ リミテ ７－デアセチル－フォルスコリンとｐｖｐの複合体
KR20220149987A (ko) * 2021-05-03 2022-11-10 연세대학교 산학협력단 안구건조증 또는 안구건조증 연관 안과 질환의 예방, 개선 또는 치료용 조성물
CN117586217B (zh) * 2024-01-17 2024-03-19 云南省药物研究所 一种基于国产毛喉鞘蕊花的佛司可林制备方法

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HU181703B (en) * 1980-05-09 1983-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing aqueus solutuins of water insoluble or hardly soluble vitamines, steroides, localanesthetics, prostanoides and non-steroid and antiphlogistic agents
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Also Published As

Publication number Publication date
CA2537820C (en) 2013-03-26
NZ545765A (en) 2009-11-27
CN1882508A (zh) 2006-12-20
RS20060169A (en) 2008-08-07
JP5021305B2 (ja) 2012-09-05
AU2004272005A1 (en) 2005-03-24
US6960300B2 (en) 2005-11-01
EP1718568A2 (en) 2006-11-08
WO2005025500A2 (en) 2005-03-24
MXPA06002684A (es) 2007-03-15
BRPI0413957A (pt) 2006-10-31
CN1882508B (zh) 2010-07-14
CA2537820A1 (en) 2005-03-24
JP2007505040A (ja) 2007-03-08
US20050051483A1 (en) 2005-03-10
EA012836B1 (ru) 2009-12-30
HK1098450A1 (en) 2007-07-20
WO2005025500A3 (en) 2005-06-09
US20050284812A1 (en) 2005-12-29
EA200600528A1 (ru) 2006-08-25
EP1718568B1 (en) 2012-12-26
AU2004272005B2 (en) 2011-03-10
EP1718568A4 (en) 2009-01-07

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