ZA200503926B - Methods of using and compositions comprising (-)030(3,4-dimethoxy-phenyl)-3-(1-oxo 1,3-dihydro-isoindol-2-yl)-propionamide - Google Patents

Methods of using and compositions comprising (-)030(3,4-dimethoxy-phenyl)-3-(1-oxo 1,3-dihydro-isoindol-2-yl)-propionamide Download PDF

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Publication number
ZA200503926B
ZA200503926B ZA200503926A ZA200503926A ZA200503926B ZA 200503926 B ZA200503926 B ZA 200503926B ZA 200503926 A ZA200503926 A ZA 200503926A ZA 200503926 A ZA200503926 A ZA 200503926A ZA 200503926 B ZA200503926 B ZA 200503926B
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South Africa
Prior art keywords
enantiomerically pure
solvate
salt
disease
dihydro
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ZA200503926A
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English (en)
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George W Muller
Roger S Chen
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Celgene Corp
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/4035—Isoindoles, e.g. phthalimide
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
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ZA200503926A 2002-11-18 2005-05-16 Methods of using and compositions comprising (-)030(3,4-dimethoxy-phenyl)-3-(1-oxo 1,3-dihydro-isoindol-2-yl)-propionamide ZA200503926B (en)

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US42738002P 2002-11-18 2002-11-18

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ZA200503926B true ZA200503926B (en) 2006-08-30

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ZA200503926A ZA200503926B (en) 2002-11-18 2005-05-16 Methods of using and compositions comprising (-)030(3,4-dimethoxy-phenyl)-3-(1-oxo 1,3-dihydro-isoindol-2-yl)-propionamide

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US (1) US20040167199A1 (enExample)
EP (1) EP1569599A2 (enExample)
JP (1) JP2006515844A (enExample)
KR (1) KR20050086715A (enExample)
CN (1) CN1738614A (enExample)
AU (1) AU2003294312A1 (enExample)
BR (1) BR0316256A (enExample)
CA (1) CA2506442A1 (enExample)
MX (1) MXPA05005161A (enExample)
NZ (1) NZ540546A (enExample)
TW (1) TW200415143A (enExample)
WO (1) WO2004054501A2 (enExample)
ZA (1) ZA200503926B (enExample)

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