ZA200502009B - 1-Pyridiin-4-yl-urea derivatives. - Google Patents
1-Pyridiin-4-yl-urea derivatives. Download PDFInfo
- Publication number
- ZA200502009B ZA200502009B ZA200502009A ZA200502009A ZA200502009B ZA 200502009 B ZA200502009 B ZA 200502009B ZA 200502009 A ZA200502009 A ZA 200502009A ZA 200502009 A ZA200502009 A ZA 200502009A ZA 200502009 B ZA200502009 B ZA 200502009B
- Authority
- ZA
- South Africa
- Prior art keywords
- pyrrolidin
- compounds
- urea
- methyl
- general formula
- Prior art date
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Landscapes
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
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| EP0210417 | 2002-09-17 |
Publications (1)
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| ZA200502009B true ZA200502009B (en) | 2005-11-01 |
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| Country | Link |
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| US (1) | US20060094716A1 (fr) |
| EP (1) | EP1554249A2 (fr) |
| JP (1) | JP2006505533A (fr) |
| KR (1) | KR20050043967A (fr) |
| CN (1) | CN1681789A (fr) |
| AU (1) | AU2003270186A1 (fr) |
| BR (1) | BR0314353A (fr) |
| CA (1) | CA2496624A1 (fr) |
| MX (1) | MXPA05002839A (fr) |
| NO (1) | NO20050932L (fr) |
| RU (1) | RU2005111589A (fr) |
| WO (1) | WO2004026836A2 (fr) |
| ZA (1) | ZA200502009B (fr) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
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| ATE555087T1 (de) * | 2002-11-27 | 2012-05-15 | Incyte Corp | 3-aminopyrrolidinderivate als modulatoren von chemokinrezeptoren |
| WO2004073634A2 (fr) | 2003-02-20 | 2004-09-02 | Encysive Pharmaceuticals Inc. | Antagonistes du recepteur de l'urotensine-ii de la phenylenediamine et antagonistes du ccr-9 |
| US7288538B2 (en) | 2003-02-20 | 2007-10-30 | Encysive Pharmaceuticals, Inc. | Phenylenediamine urotensin-II receptor antagonists and CCR-9 antagonists |
| US7320989B2 (en) | 2003-02-28 | 2008-01-22 | Encysive Pharmaceuticals, Inc. | Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-II receptor antagonists |
| AU2004218456A1 (en) | 2003-02-28 | 2004-09-16 | Encysive Pharmaceuticals Inc. | Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-II receptor antagonists. |
| JP2006519826A (ja) | 2003-03-06 | 2006-08-31 | グラクソ グループ リミテッド | 疼痛治療のための複素環式尿素誘導体 |
| EP1601665A2 (fr) * | 2003-03-07 | 2005-12-07 | Glaxo Group Limited | Derives d'uree |
| GB0305426D0 (en) * | 2003-03-08 | 2003-04-16 | Glaxo Group Ltd | Novel compounds |
| WO2004089296A2 (fr) | 2003-04-03 | 2004-10-21 | The Regents Of The University Of California | Inhibiteurs ameliores pour hydrolase epoxyde soluble |
| EP1670470B1 (fr) | 2003-09-26 | 2009-04-08 | Actelion Pharmaceuticals Ltd. | Derives de pyridine et leur utilisation comme antagonistes de l'urotensine ii |
| EP1765311A4 (fr) | 2004-03-16 | 2009-04-29 | Univ California | Reduction de la nephropathie au moyen d'inhibiteurs d'hydrolase d'epoxyde soluble et d'epoxyeicosanoides |
| MX2007004293A (es) * | 2004-10-12 | 2007-06-18 | Actelion Pharmaceuticals Ltd | 1[2-(4-bencil-4-hidroxi-piperidin-1-il)-etil]-3-(2-metil-quinolin -4-il)-urea como la sal de sulfato cristalina. |
| NZ554555A (en) | 2004-10-20 | 2011-09-30 | Univ California | Cyclohexyl-urea derivatives as improved inhibitors for the soluble epoxide hydrolase |
| NZ566023A (en) | 2005-09-21 | 2010-02-26 | Pfizer Ltd | Carboxamide derivatives as muscarinic receptor antagonists |
| TW200808723A (en) * | 2006-03-13 | 2008-02-16 | Univ California | Conformationally restricted urea inhibitors of soluble epoxide hydrolase |
| WO2008144268A1 (fr) * | 2007-05-15 | 2008-11-27 | Boehringer Ingelheim International Gmbh | Antagonistes de récepteur d'urotensine ii |
| EP2297107B1 (fr) * | 2008-06-03 | 2013-11-13 | Actelion Pharmaceuticals Ltd. | Dérivés de [4-(1-amino-éthyl)-cyclohexyl]-méthyl-amine et de [6-(1-amino-ethyl)-tétrahydro-pyran-3-yl]-méthyl-amine comme antibacteriels |
| US9296693B2 (en) | 2010-01-29 | 2016-03-29 | The Regents Of The University Of California | Acyl piperidine inhibitors of soluble epoxide hydrolase |
| WO2011121555A1 (fr) * | 2010-03-31 | 2011-10-06 | Actelion Pharmaceuticals Ltd | Dérivés d'isoquinoléin-3-ylurée antibactériens |
| JP2014512337A (ja) * | 2011-01-28 | 2014-05-22 | ユニバーシティ オブ ケンタッキー リサーチ ファウンデーション | スチルベン類似体およびがんを処置する方法 |
| WO2016116900A1 (fr) * | 2015-01-23 | 2016-07-28 | Gvk Biosciences Private Limited | Inhibiteurs de trka kinase |
| CN107056673B (zh) * | 2016-09-09 | 2019-10-29 | 南京工业大学 | 一种3,4-二芳基马来酰亚胺衍生物及其制备方法与应用 |
| CN106432039B (zh) * | 2016-09-27 | 2019-02-22 | 南京工业大学 | 3,4-二芳基马来酰亚胺衍生物及其制备方法与应用 |
| WO2020042972A1 (fr) * | 2018-08-27 | 2020-03-05 | 北京赛特明强医药科技有限公司 | Composé de dioxane et de quinazoline ou de quinoléine lié à un cycle aromatique substitué par urée, composition et utilisation associée |
| FI4097099T3 (fi) | 2020-02-07 | 2024-07-30 | Gasherbrum Bio Inc | Heterosyklisiä glp-1-agonisteja |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR016817A1 (es) * | 1997-08-14 | 2001-08-01 | Smithkline Beecham Plc | Derivados de fenilurea o feniltiourea, procedimiento para su preparacion, coleccion de compuestos, compuestos intermediarios, composicion farmaceutica,metodo de tratamiento y uso de dichos compuestos para la manufactura de un medicamento |
| AUPP003197A0 (en) * | 1997-09-03 | 1997-11-20 | Fujisawa Pharmaceutical Co., Ltd. | New heterocyclic compounds |
| WO2000047577A1 (fr) * | 1999-02-12 | 2000-08-17 | Smithkline Beecham Plc | Derives de phenyluree et de phenylthiouree utilises comme antagonistes des recepteurs de l'orexine |
| NZ527276A (en) * | 2001-03-27 | 2004-11-26 | Actelion Pharmaceuticals Ltd | 1,2,3,4-tetrahydroisoquinoline derivatives as urotensin II receptor antagonists |
| CA2473892C (fr) * | 2001-12-04 | 2010-09-21 | Actelion Pharmaceuticals Ltd | Nouveaux derives de quinoleines |
-
2003
- 2003-09-12 AU AU2003270186A patent/AU2003270186A1/en not_active Abandoned
- 2003-09-12 MX MXPA05002839A patent/MXPA05002839A/es unknown
- 2003-09-12 US US10/528,043 patent/US20060094716A1/en not_active Abandoned
- 2003-09-12 CA CA002496624A patent/CA2496624A1/fr not_active Abandoned
- 2003-09-12 CN CNA038219646A patent/CN1681789A/zh active Pending
- 2003-09-12 EP EP03750534A patent/EP1554249A2/fr not_active Withdrawn
- 2003-09-12 KR KR1020057004455A patent/KR20050043967A/ko not_active Application Discontinuation
- 2003-09-12 RU RU2005111589/04A patent/RU2005111589A/ru not_active Application Discontinuation
- 2003-09-12 WO PCT/EP2003/010154 patent/WO2004026836A2/fr not_active Application Discontinuation
- 2003-09-12 BR BR0314353-8A patent/BR0314353A/pt not_active IP Right Cessation
- 2003-09-12 JP JP2004537065A patent/JP2006505533A/ja not_active Abandoned
-
2005
- 2005-02-21 NO NO20050932A patent/NO20050932L/no not_active Application Discontinuation
- 2005-03-09 ZA ZA200502009A patent/ZA200502009B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004026836A3 (fr) | 2005-01-20 |
| CA2496624A1 (fr) | 2004-04-01 |
| KR20050043967A (ko) | 2005-05-11 |
| WO2004026836A8 (fr) | 2005-05-12 |
| AU2003270186A1 (en) | 2004-04-08 |
| NO20050932L (no) | 2005-04-15 |
| WO2004026836A2 (fr) | 2004-04-01 |
| RU2005111589A (ru) | 2006-01-20 |
| BR0314353A (pt) | 2005-07-19 |
| EP1554249A2 (fr) | 2005-07-20 |
| CN1681789A (zh) | 2005-10-12 |
| JP2006505533A (ja) | 2006-02-16 |
| US20060094716A1 (en) | 2006-05-04 |
| MXPA05002839A (es) | 2005-05-27 |
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