ZA200408618B - A combination product comprising an anti-coagulant and anti-arrhythmic oxabispidenes - Google Patents
A combination product comprising an anti-coagulant and anti-arrhythmic oxabispidenes Download PDFInfo
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- ZA200408618B ZA200408618B ZA200408618A ZA200408618A ZA200408618B ZA 200408618 B ZA200408618 B ZA 200408618B ZA 200408618 A ZA200408618 A ZA 200408618A ZA 200408618 A ZA200408618 A ZA 200408618A ZA 200408618 B ZA200408618 B ZA 200408618B
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- GXTOJJVRHWFNPK-UHFFFAOYSA-N tert-butyl n-[2-[7-[3-(4-cyanophenoxy)propyl]-9-oxa-3,7-diazabicyclo[3.3.1]nonan-3-yl]ethyl]carbamate Chemical compound C1C(O2)CN(CCNC(=O)OC(C)(C)C)CC2CN1CCCOC1=CC=C(C#N)C=C1 GXTOJJVRHWFNPK-UHFFFAOYSA-N 0.000 description 1
- CIJQTPFWFXOSEO-NDMITSJXSA-J tetrasodium;(2r,3r,4s)-2-[(2r,3s,4r,5r,6s)-5-acetamido-6-[(1r,2r,3r,4r)-4-[(2r,3s,4r,5r,6r)-5-acetamido-6-[(4r,5r,6r)-2-carboxylato-4,5-dihydroxy-6-[[(1r,3r,4r,5r)-3-hydroxy-4-(sulfonatoamino)-6,8-dioxabicyclo[3.2.1]octan-2-yl]oxy]oxan-3-yl]oxy-2-(hydroxy Chemical compound [Na+].[Na+].[Na+].[Na+].O([C@@H]1[C@@H](COS(O)(=O)=O)O[C@@H]([C@@H]([C@H]1O)NC(C)=O)O[C@@H]1C(C[C@H]([C@@H]([C@H]1O)O)O[C@@H]1[C@@H](CO)O[C@H](OC2C(O[C@@H](OC3[C@@H]([C@@H](NS([O-])(=O)=O)[C@@H]4OC[C@H]3O4)O)[C@H](O)[C@H]2O)C([O-])=O)[C@H](NC(C)=O)[C@H]1C)C([O-])=O)[C@@H]1OC(C([O-])=O)=C[C@H](O)[C@H]1O CIJQTPFWFXOSEO-NDMITSJXSA-J 0.000 description 1
- 229960005001 ticlopidine Drugs 0.000 description 1
- PHWBOXQYWZNQIN-UHFFFAOYSA-N ticlopidine Chemical compound ClC1=CC=CC=C1CN1CC(C=CS2)=C2CC1 PHWBOXQYWZNQIN-UHFFFAOYSA-N 0.000 description 1
- 229950005830 tifacogin Drugs 0.000 description 1
- 210000001519 tissue Anatomy 0.000 description 1
- 230000009261 transgenic effect Effects 0.000 description 1
- 238000012384 transportation and delivery Methods 0.000 description 1
- 229960005356 urokinase Drugs 0.000 description 1
- 235000019168 vitamin K Nutrition 0.000 description 1
- 239000011712 vitamin K Substances 0.000 description 1
- 150000003721 vitamin K derivatives Chemical class 0.000 description 1
- 229940046010 vitamin k Drugs 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines having two or more nitrogen atoms in the same ring, e.g. oxadiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/06—Tripeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Gastroenterology & Hepatology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0201374A SE0201374D0 (sv) | 2002-05-06 | 2002-05-06 | Pharmaceutical combination |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200408618B true ZA200408618B (en) | 2006-06-28 |
Family
ID=20287789
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200408618A ZA200408618B (en) | 2002-05-06 | 2004-10-25 | A combination product comprising an anti-coagulant and anti-arrhythmic oxabispidenes |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20050119259A1 (es) |
| EP (1) | EP1503783A1 (es) |
| JP (1) | JP2005529140A (es) |
| KR (1) | KR20040104692A (es) |
| CN (1) | CN1652812A (es) |
| AR (1) | AR039883A1 (es) |
| AU (1) | AU2003230517A1 (es) |
| BR (1) | BR0309336A (es) |
| CA (1) | CA2485086A1 (es) |
| IL (1) | IL164939A0 (es) |
| IS (1) | IS7536A (es) |
| MX (1) | MXPA04010717A (es) |
| NO (1) | NO20044555L (es) |
| PL (1) | PL372526A1 (es) |
| RU (1) | RU2004129729A (es) |
| SE (1) | SE0201374D0 (es) |
| TW (1) | TW200307549A (es) |
| WO (1) | WO2003092720A1 (es) |
| ZA (1) | ZA200408618B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ITMI20042068A1 (it) * | 2004-10-29 | 2005-01-29 | Opocrin Spa | Nuovo uso di eparine a bassissimo peso molecolare |
| WO2006137772A1 (en) * | 2005-06-20 | 2006-12-28 | Astrazeneca Ab | New physical form of n,n´- disubstituted oxabispidines |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU178398B (en) * | 1979-06-12 | 1982-04-28 | Gyogyszerkutato Intezet | Process for producing new agmatine derivatives of activity against haemagglutination |
| SE9903759D0 (sv) * | 1999-10-18 | 1999-10-18 | Astra Ab | Pharmaceutically active compounds |
| US6462021B1 (en) * | 2000-11-06 | 2002-10-08 | Astrazeneca Ab | Use of low molecular weight thrombin inhibitor |
-
2002
- 2002-05-06 SE SE0201374A patent/SE0201374D0/xx unknown
-
2003
- 2003-04-24 TW TW092109612A patent/TW200307549A/zh unknown
- 2003-05-05 BR BR0309336-0A patent/BR0309336A/pt not_active IP Right Cessation
- 2003-05-05 AU AU2003230517A patent/AU2003230517A1/en not_active Abandoned
- 2003-05-05 US US10/513,190 patent/US20050119259A1/en not_active Abandoned
- 2003-05-05 CN CNA038103273A patent/CN1652812A/zh active Pending
- 2003-05-05 EP EP03723588A patent/EP1503783A1/en not_active Withdrawn
- 2003-05-05 KR KR10-2004-7017642A patent/KR20040104692A/ko not_active Application Discontinuation
- 2003-05-05 CA CA002485086A patent/CA2485086A1/en not_active Abandoned
- 2003-05-05 RU RU2004129729/15A patent/RU2004129729A/ru not_active Application Discontinuation
- 2003-05-05 PL PL03372526A patent/PL372526A1/xx not_active Application Discontinuation
- 2003-05-05 MX MXPA04010717A patent/MXPA04010717A/es unknown
- 2003-05-05 WO PCT/SE2003/000719 patent/WO2003092720A1/en active Application Filing
- 2003-05-05 JP JP2004500903A patent/JP2005529140A/ja active Pending
- 2003-05-06 AR ARP030101592A patent/AR039883A1/es not_active Application Discontinuation
-
2004
- 2004-10-22 NO NO20044555A patent/NO20044555L/no unknown
- 2004-10-25 ZA ZA200408618A patent/ZA200408618B/en unknown
- 2004-10-31 IL IL16493904A patent/IL164939A0/xx unknown
- 2004-11-18 IS IS7536A patent/IS7536A/is unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2004129729A (ru) | 2005-07-10 |
| BR0309336A (pt) | 2005-03-08 |
| SE0201374D0 (sv) | 2002-05-06 |
| WO2003092720A8 (en) | 2005-03-10 |
| AR039883A1 (es) | 2005-03-09 |
| MXPA04010717A (es) | 2005-03-07 |
| WO2003092720A1 (en) | 2003-11-13 |
| IL164939A0 (en) | 2005-12-18 |
| JP2005529140A (ja) | 2005-09-29 |
| NO20044555L (no) | 2004-11-16 |
| KR20040104692A (ko) | 2004-12-10 |
| PL372526A1 (en) | 2005-07-25 |
| CN1652812A (zh) | 2005-08-10 |
| EP1503783A1 (en) | 2005-02-09 |
| AU2003230517A1 (en) | 2003-11-17 |
| TW200307549A (en) | 2003-12-16 |
| US20050119259A1 (en) | 2005-06-02 |
| IS7536A (is) | 2004-11-18 |
| CA2485086A1 (en) | 2003-11-13 |
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