ZA200309095B - Oxazole/thiazol-derivatives activators of the hPPAR-alpha receptor. - Google Patents
Oxazole/thiazol-derivatives activators of the hPPAR-alpha receptor. Download PDFInfo
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- ZA200309095B ZA200309095B ZA200309095A ZA200309095A ZA200309095B ZA 200309095 B ZA200309095 B ZA 200309095B ZA 200309095 A ZA200309095 A ZA 200309095A ZA 200309095 A ZA200309095 A ZA 200309095A ZA 200309095 B ZA200309095 B ZA 200309095B
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- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Landscapes
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- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Biomedical Technology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0113231.5A GB0113231D0 (en) | 2001-05-31 | 2001-05-31 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200309095B true ZA200309095B (en) | 2005-02-21 |
Family
ID=9915636
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200309095A ZA200309095B (en) | 2001-05-31 | 2003-11-21 | Oxazole/thiazol-derivatives activators of the hPPAR-alpha receptor. |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US7157479B2 (de) |
| EP (1) | EP1399430B1 (de) |
| JP (1) | JP2004532267A (de) |
| KR (1) | KR100859591B1 (de) |
| CN (1) | CN1307166C (de) |
| AR (1) | AR034051A1 (de) |
| AU (1) | AU2002317765B2 (de) |
| BR (1) | BR0209785A (de) |
| CA (1) | CA2448205A1 (de) |
| CO (1) | CO5540297A2 (de) |
| CY (1) | CY1107206T1 (de) |
| CZ (1) | CZ20033252A3 (de) |
| DE (1) | DE60223805T2 (de) |
| DK (1) | DK1399430T3 (de) |
| ES (1) | ES2296965T3 (de) |
| GB (1) | GB0113231D0 (de) |
| HK (1) | HK1064367A1 (de) |
| HU (1) | HUP0400043A3 (de) |
| IL (1) | IL158929A0 (de) |
| MX (1) | MXPA03011032A (de) |
| MY (1) | MY132656A (de) |
| NO (1) | NO20035209L (de) |
| NZ (1) | NZ529754A (de) |
| PL (1) | PL367248A1 (de) |
| PT (1) | PT1399430E (de) |
| SI (1) | SI1399430T1 (de) |
| TW (1) | TWI245760B (de) |
| WO (1) | WO2002096895A1 (de) |
| ZA (1) | ZA200309095B (de) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002335231B2 (en) * | 2001-10-12 | 2008-05-08 | Nippon Chemiphar Co., Ltd. | Activator for peroxisome proliferator-activated receptor delta |
| AU2003261935A1 (en) | 2002-09-06 | 2004-03-29 | Takeda Pharmaceutical Company Limited | Furan or thiophene derivative and medicinal use thereof |
| GB0314370D0 (en) * | 2003-06-19 | 2003-07-23 | Glaxo Group Ltd | Chemical compounds |
| GB0323702D0 (en) * | 2003-10-09 | 2003-11-12 | Smithkline Beecham Corp | Chemical compound |
| MXPA06004641A (es) | 2003-11-05 | 2006-06-27 | Hoffmann La Roche | Derivados de fenilo como agonistas para. |
| FR2882359A1 (fr) * | 2005-02-24 | 2006-08-25 | Negma Lerads Soc Par Actions S | Derives activateurs de ppar, procede de preparation et application en therapeutique |
| CN101007790B (zh) * | 2006-01-27 | 2011-03-30 | 北京摩力克科技有限公司 | 草氨酸衍生物、其制备方法和医药用途 |
| FR2901792A1 (fr) * | 2006-06-06 | 2007-12-07 | Negma Lerads Soc Par Actions S | DERIVES ACTIVATEURS DE PPARs, PROCEDE DE PREPARATION ET APPLICATION EN THERAPEUTIQUE |
| EP2380884B1 (de) | 2008-12-01 | 2014-02-12 | Mitsubishi Tanabe Pharma Corporation | Carbonsäurederivat mit thiazolring und dessen pharmazeutische verwendung |
| CN110803996B (zh) * | 2019-11-13 | 2022-01-11 | 台州市创源工业技术有限公司 | 一种羟基苄胺的合成方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998007699A1 (fr) | 1996-08-19 | 1998-02-26 | Japan Tobacco Inc. | Derives d'acide propionique et applications de ces derives |
| DE69941777D1 (de) | 1998-03-10 | 2010-01-21 | Ono Pharmaceutical Co | Carbonsäurederivate und medikamente die diese als aktiven wirkstoff enthalten |
| ES2261202T3 (es) * | 1999-04-28 | 2006-11-16 | Sanofi-Aventis Deutschland Gmbh | Derivados de acido de triarilo como ligandos para el receptor ppar. |
| GB9914977D0 (en) | 1999-06-25 | 1999-08-25 | Glaxo Group Ltd | Chemical compounds |
| CA2382966A1 (en) * | 1999-08-27 | 2001-03-08 | Eli Lilly And Company | Biaryl-oxa(thia)zole derivatives and their use as ppars modulators |
| PE20011010A1 (es) * | 1999-12-02 | 2001-10-18 | Glaxo Group Ltd | Oxazoles y tiazoles sustituidos como agonista del receptor activado por el proliferador de peroxisomas humano |
| GB0113233D0 (en) * | 2001-05-31 | 2001-07-25 | Glaxo Group Ltd | Chemical compounds |
-
2001
- 2001-05-31 GB GBGB0113231.5A patent/GB0113231D0/en not_active Ceased
-
2002
- 2002-05-29 SI SI200230654T patent/SI1399430T1/sl unknown
- 2002-05-29 ES ES02747331T patent/ES2296965T3/es not_active Expired - Lifetime
- 2002-05-29 AU AU2002317765A patent/AU2002317765B2/en not_active Ceased
- 2002-05-29 MY MYPI20021973A patent/MY132656A/en unknown
- 2002-05-29 US US10/478,936 patent/US7157479B2/en not_active Expired - Fee Related
- 2002-05-29 CN CNB028149424A patent/CN1307166C/zh not_active Expired - Fee Related
- 2002-05-29 IL IL15892902A patent/IL158929A0/xx unknown
- 2002-05-29 JP JP2003500074A patent/JP2004532267A/ja active Pending
- 2002-05-29 NZ NZ529754A patent/NZ529754A/en unknown
- 2002-05-29 CZ CZ20033252A patent/CZ20033252A3/cs unknown
- 2002-05-29 DE DE60223805T patent/DE60223805T2/de not_active Expired - Fee Related
- 2002-05-29 BR BR0209785-0A patent/BR0209785A/pt not_active IP Right Cessation
- 2002-05-29 WO PCT/EP2002/005886 patent/WO2002096895A1/en active IP Right Grant
- 2002-05-29 PL PL02367248A patent/PL367248A1/xx not_active Application Discontinuation
- 2002-05-29 PT PT02747331T patent/PT1399430E/pt unknown
- 2002-05-29 EP EP02747331A patent/EP1399430B1/de not_active Expired - Lifetime
- 2002-05-29 DK DK02747331T patent/DK1399430T3/da active
- 2002-05-29 CA CA002448205A patent/CA2448205A1/en not_active Abandoned
- 2002-05-29 MX MXPA03011032A patent/MXPA03011032A/es active IP Right Grant
- 2002-05-29 AR ARP020101999A patent/AR034051A1/es unknown
- 2002-05-29 HU HU0400043A patent/HUP0400043A3/hu unknown
- 2002-05-29 TW TW091111392A patent/TWI245760B/zh not_active IP Right Cessation
- 2002-05-29 KR KR1020037015678A patent/KR100859591B1/ko not_active IP Right Cessation
-
2003
- 2003-11-21 ZA ZA200309095A patent/ZA200309095B/en unknown
- 2003-11-24 NO NO20035209A patent/NO20035209L/no not_active Application Discontinuation
- 2003-12-03 CO CO03106490A patent/CO5540297A2/es not_active Application Discontinuation
-
2004
- 2004-09-13 HK HK04106944A patent/HK1064367A1/xx not_active IP Right Cessation
-
2008
- 2008-02-19 CY CY20081100202T patent/CY1107206T1/el unknown
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