ZA200308859B - Pyrimidine, triazine and pyrazine derivatives as glutamate receptors. - Google Patents

Pyrimidine, triazine and pyrazine derivatives as glutamate receptors. Download PDF

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Publication number
ZA200308859B
ZA200308859B ZA200308859A ZA200308859A ZA200308859B ZA 200308859 B ZA200308859 B ZA 200308859B ZA 200308859 A ZA200308859 A ZA 200308859A ZA 200308859 A ZA200308859 A ZA 200308859A ZA 200308859 B ZA200308859 B ZA 200308859B
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South Africa
Prior art keywords
phenyl
carbonitrile
pyrimidine
formula
fluoro
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ZA200308859A
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English (en)
Inventor
Alfred Binggeli
Thierry Masquelin
Maurice Wilhelm
Hans-Peter Maerki
Vincent Mutel
Wolfgang Wostl
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Hoffmann La Roche
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Publication of ZA200308859B publication Critical patent/ZA200308859B/en

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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
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    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

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ZA200308859A 2001-06-01 2003-11-13 Pyrimidine, triazine and pyrazine derivatives as glutamate receptors. ZA200308859B (en)

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Application Number Priority Date Filing Date Title
EP01113379 2001-06-01

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ZA200308859B true ZA200308859B (en) 2005-02-14

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ZA200308859A ZA200308859B (en) 2001-06-01 2003-11-13 Pyrimidine, triazine and pyrazine derivatives as glutamate receptors.

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US (1) US6673795B2 (https=)
EP (1) EP1397351B1 (https=)
JP (1) JP4049742B2 (https=)
KR (1) KR100602927B1 (https=)
CN (1) CN1245391C (https=)
AR (1) AR036075A1 (https=)
AT (1) ATE448210T1 (https=)
AU (1) AU2002319183B2 (https=)
BR (1) BR0210102A (https=)
CA (1) CA2448602C (https=)
DE (1) DE60234338D1 (https=)
DK (1) DK1397351T3 (https=)
ES (1) ES2332505T3 (https=)
MX (1) MXPA03010822A (https=)
PT (1) PT1397351E (https=)
WO (1) WO2002098864A1 (https=)
ZA (1) ZA200308859B (https=)

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ES2987794T3 (es) 2018-06-06 2024-11-18 Arena Pharm Inc Procedimientos de tratamiento de afecciones relacionadas con el receptor S1P1

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US6673795B2 (en) 2004-01-06
MXPA03010822A (es) 2004-02-17
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AR036075A1 (es) 2004-08-11
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