ZA200301543B - Medicinal compositions. - Google Patents
Medicinal compositions. Download PDFInfo
- Publication number
- ZA200301543B ZA200301543B ZA200301543A ZA200301543A ZA200301543B ZA 200301543 B ZA200301543 B ZA 200301543B ZA 200301543 A ZA200301543 A ZA 200301543A ZA 200301543 A ZA200301543 A ZA 200301543A ZA 200301543 B ZA200301543 B ZA 200301543B
- Authority
- ZA
- South Africa
- Prior art keywords
- hmg
- coa reductase
- reductase inhibitor
- dimethylindolin
- octyl
- Prior art date
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- 239000000203 mixture Substances 0.000 title claims description 39
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- 229960002965 pravastatin Drugs 0.000 claims description 59
- TUZYXOIXSAXUGO-PZAWKZKUSA-N pravastatin Chemical compound C1=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(O)=O)[C@H]2[C@@H](OC(=O)[C@@H](C)CC)C[C@H](O)C=C21 TUZYXOIXSAXUGO-PZAWKZKUSA-N 0.000 claims description 59
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- XUKUURHRXDUEBC-KAYWLYCHSA-N Atorvastatin Chemical compound C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CC[C@@H](O)C[C@@H](O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-KAYWLYCHSA-N 0.000 claims description 55
- XUKUURHRXDUEBC-UHFFFAOYSA-N Atorvastatin Natural products C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CCC(O)CC(O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-UHFFFAOYSA-N 0.000 claims description 55
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-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Emergency Medicine (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000265082 | 2000-09-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200301543B true ZA200301543B (en) | 2004-06-09 |
Family
ID=18752403
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200301543A ZA200301543B (en) | 2000-09-01 | 2003-02-25 | Medicinal compositions. |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1314423A4 (no) |
| KR (1) | KR20030029871A (no) |
| CN (1) | CN1473042A (no) |
| AU (2) | AU8254101A (no) |
| BR (1) | BR0113523A (no) |
| CA (1) | CA2420951A1 (no) |
| CZ (1) | CZ2003593A3 (no) |
| HU (1) | HUP0301728A3 (no) |
| IL (1) | IL154414A0 (no) |
| MX (1) | MXPA03001857A (no) |
| NO (1) | NO20030946L (no) |
| NZ (1) | NZ524406A (no) |
| PL (1) | PL362244A1 (no) |
| RU (1) | RU2246302C2 (no) |
| SK (1) | SK2552003A3 (no) |
| WO (1) | WO2002020009A1 (no) |
| ZA (1) | ZA200301543B (no) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20030029871A (ko) * | 2000-09-01 | 2003-04-16 | 상꾜 가부시키가이샤 | 의약 조성물 |
| RU2358734C2 (ru) | 2003-08-29 | 2009-06-20 | Кова Ко., Лтд. | Способ стабилизации бляшки с высоким содержанием липидов и способ профилактики ее разрушения |
| TW200619204A (en) * | 2004-12-10 | 2006-06-16 | Kowa Co | Method for reduction, stabilization and prevention of rupture of lipid rich plaque |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3720395B2 (ja) * | 1994-09-20 | 2005-11-24 | 京都薬品工業株式会社 | 新規ヘテロ環誘導体、その製造方法およびその医薬用途 |
| DE69617731T2 (de) * | 1995-10-05 | 2002-08-08 | Kyoto Pharma Ind | Neue heterozyklische derivate und ihre medizinische anwendung |
| NZ319906A (en) * | 1995-11-02 | 2000-02-28 | Warner Lambert Co | Method of preparing a pharmaceutical composition for regulating lipid concentration comprising using an acyl-CoA cholesterol O-acyltransferase inhibitor and an HMG-CoA reductase inhibitor |
| YU23499A (sh) * | 1996-11-27 | 2001-07-10 | Pfizer Inc. | Inhibitorski amidi apo-b-sekrecije/mtp-a |
| CA2307553C (en) * | 1997-10-28 | 2003-06-17 | Korea Institute Of Science And Technology | Citrus peel extract as inhibitor of acyl coa-cholesterol-o-acyltransferase, inhibitor of macrophage-lipid complex accumulation on the arterial wall and preventive or treating agent for hepatic diseases |
| YU3501A (sh) * | 1998-07-21 | 2005-06-10 | Warner-Lambert Company | Zajedničko ordiniranje inhibitora acat i mmp za tretman oštećenja od ateroskleroze |
| AU7717500A (en) * | 1999-09-30 | 2001-04-30 | Merck & Co., Inc. | Anti-hypercholesterolemic drug combination |
| KR20030029871A (ko) * | 2000-09-01 | 2003-04-16 | 상꾜 가부시키가이샤 | 의약 조성물 |
-
2001
- 2001-08-29 KR KR10-2003-7002861A patent/KR20030029871A/ko not_active Application Discontinuation
- 2001-08-29 SK SK255-2003A patent/SK2552003A3/sk not_active Application Discontinuation
- 2001-08-29 CA CA002420951A patent/CA2420951A1/en not_active Abandoned
- 2001-08-29 PL PL01362244A patent/PL362244A1/xx unknown
- 2001-08-29 AU AU8254101A patent/AU8254101A/xx active Pending
- 2001-08-29 AU AU2001282541A patent/AU2001282541B2/en not_active Ceased
- 2001-08-29 CZ CZ2003593A patent/CZ2003593A3/cs unknown
- 2001-08-29 RU RU2003105835/15A patent/RU2246302C2/ru not_active IP Right Cessation
- 2001-08-29 EP EP01961177A patent/EP1314423A4/en not_active Withdrawn
- 2001-08-29 NZ NZ524406A patent/NZ524406A/en unknown
- 2001-08-29 MX MXPA03001857A patent/MXPA03001857A/es unknown
- 2001-08-29 HU HU0301728A patent/HUP0301728A3/hu unknown
- 2001-08-29 WO PCT/JP2001/007438 patent/WO2002020009A1/ja not_active Application Discontinuation
- 2001-08-29 IL IL15441401A patent/IL154414A0/xx unknown
- 2001-08-29 BR BR0113523-6A patent/BR0113523A/pt not_active IP Right Cessation
- 2001-08-29 CN CNA018184723A patent/CN1473042A/zh active Pending
-
2003
- 2003-02-25 ZA ZA200301543A patent/ZA200301543B/en unknown
- 2003-02-28 NO NO20030946A patent/NO20030946L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1473042A (zh) | 2004-02-04 |
| IL154414A0 (en) | 2003-09-17 |
| HUP0301728A3 (en) | 2004-05-28 |
| EP1314423A1 (en) | 2003-05-28 |
| EP1314423A4 (en) | 2004-05-19 |
| AU2001282541B2 (en) | 2004-06-24 |
| HUP0301728A2 (hu) | 2003-08-28 |
| NO20030946L (no) | 2003-04-08 |
| RU2246302C2 (ru) | 2005-02-20 |
| CA2420951A1 (en) | 2003-02-28 |
| PL362244A1 (en) | 2004-10-18 |
| CZ2003593A3 (cs) | 2003-05-14 |
| KR20030029871A (ko) | 2003-04-16 |
| AU8254101A (en) | 2002-03-22 |
| WO2002020009A1 (fr) | 2002-03-14 |
| SK2552003A3 (en) | 2003-08-05 |
| MXPA03001857A (es) | 2003-06-04 |
| BR0113523A (pt) | 2004-06-29 |
| NZ524406A (en) | 2004-06-25 |
| NO20030946D0 (no) | 2003-02-28 |
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