ZA200209770B - 4,5-dihydro-thiazo-2-ylamine derivatives and their use as no-synthase inhibitors. - Google Patents
4,5-dihydro-thiazo-2-ylamine derivatives and their use as no-synthase inhibitors. Download PDFInfo
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- ZA200209770B ZA200209770B ZA200209770A ZA200209770A ZA200209770B ZA 200209770 B ZA200209770 B ZA 200209770B ZA 200209770 A ZA200209770 A ZA 200209770A ZA 200209770 A ZA200209770 A ZA 200209770A ZA 200209770 B ZA200209770 B ZA 200209770B
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- South Africa
- Prior art keywords
- formula
- compound
- dihydro
- pct
- thiazol
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Classifications
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- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0007396A FR2810036B1 (fr) | 2000-06-09 | 2000-06-09 | Derives de 4,5-dihydro-1,3-thiazol-2-ylamine, leur preparation et les compositions phamarceutiques les contenant |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200209770B true ZA200209770B (en) | 2004-03-02 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200209770A ZA200209770B (en) | 2000-06-09 | 2002-12-02 | 4,5-dihydro-thiazo-2-ylamine derivatives and their use as no-synthase inhibitors. |
Country Status (27)
| Country | Link |
|---|---|
| EP (1) | EP1299103B1 (es) |
| JP (1) | JP4171297B2 (es) |
| KR (1) | KR20030017990A (es) |
| CN (1) | CN1441673A (es) |
| AP (1) | AP2002002707A0 (es) |
| AT (1) | ATE305298T1 (es) |
| AU (2) | AU2001266123B2 (es) |
| BR (1) | BR0111543A (es) |
| CA (1) | CA2411572C (es) |
| DE (1) | DE60113686T2 (es) |
| DK (1) | DK1299103T3 (es) |
| DZ (1) | DZ3366A1 (es) |
| EA (1) | EA200300009A1 (es) |
| EC (1) | ECSP024374A (es) |
| ES (1) | ES2246327T3 (es) |
| FR (1) | FR2810036B1 (es) |
| HR (1) | HRP20020971A2 (es) |
| HU (1) | HUP0300996A3 (es) |
| IL (1) | IL153327A0 (es) |
| MA (1) | MA25815A1 (es) |
| MX (1) | MXPA02012072A (es) |
| NO (1) | NO20025885L (es) |
| NZ (1) | NZ522967A (es) |
| OA (1) | OA12285A (es) |
| PL (1) | PL360282A1 (es) |
| WO (1) | WO2001093867A1 (es) |
| ZA (1) | ZA200209770B (es) |
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| US8088935B2 (en) | 2003-12-23 | 2012-01-03 | Ironwood Pharmaceuticals, Inc. | Compounds and methods for the treatment of asthma |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1095710A (zh) * | 1992-11-27 | 1994-11-30 | 惠尔康基金会集团公司 | 酶抑制剂 |
| EP0724570B1 (en) * | 1993-10-21 | 1999-03-03 | G.D. Searle & Co. | Amidino derivatives useful as nitric oxide synthase inhibitors |
| AU4149696A (en) * | 1994-11-15 | 1996-06-06 | Merck & Co., Inc. | Substituted heterocycles as inhibitors of nitric oxide synthase |
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2000
- 2000-06-09 FR FR0007396A patent/FR2810036B1/fr not_active Expired - Fee Related
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2001
- 2001-06-07 AU AU2001266123A patent/AU2001266123B2/en not_active Ceased
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- 2001-06-07 CA CA002411572A patent/CA2411572C/fr not_active Expired - Fee Related
- 2001-06-07 DE DE60113686T patent/DE60113686T2/de not_active Expired - Lifetime
- 2001-06-07 OA OA1200200371A patent/OA12285A/fr unknown
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- 2001-06-07 EP EP01943579A patent/EP1299103B1/fr not_active Expired - Lifetime
- 2001-06-07 WO PCT/FR2001/001759 patent/WO2001093867A1/fr active IP Right Grant
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- 2001-06-07 DK DK01943579T patent/DK1299103T3/da active
- 2001-06-07 BR BR0111543-0A patent/BR0111543A/pt not_active Application Discontinuation
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2002
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- 2002-12-06 HR HR20020971A patent/HRP20020971A2/xx not_active Application Discontinuation
- 2002-12-09 MA MA26940A patent/MA25815A1/fr unknown
- 2002-12-09 EC EC2002004374A patent/ECSP024374A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1299103B1 (fr) | 2005-09-28 |
| ECSP024374A (es) | 2003-02-06 |
| BR0111543A (pt) | 2003-07-01 |
| NO20025885D0 (no) | 2002-12-06 |
| AP2002002707A0 (en) | 2002-12-31 |
| CN1441673A (zh) | 2003-09-10 |
| AU2001266123B2 (en) | 2007-01-25 |
| DE60113686D1 (de) | 2006-02-09 |
| DE60113686T2 (de) | 2006-07-13 |
| ATE305298T1 (de) | 2005-10-15 |
| NO20025885L (no) | 2003-01-29 |
| KR20030017990A (ko) | 2003-03-04 |
| WO2001093867A1 (fr) | 2001-12-13 |
| EP1299103A1 (fr) | 2003-04-09 |
| JP4171297B2 (ja) | 2008-10-22 |
| EA200300009A1 (ru) | 2003-04-24 |
| MA25815A1 (fr) | 2003-07-01 |
| FR2810036B1 (fr) | 2004-04-23 |
| IL153327A0 (en) | 2003-07-06 |
| AU6612301A (en) | 2001-12-17 |
| CA2411572A1 (fr) | 2001-12-13 |
| DK1299103T3 (da) | 2006-01-23 |
| FR2810036A1 (fr) | 2001-12-14 |
| HRP20020971A2 (en) | 2005-02-28 |
| ES2246327T3 (es) | 2006-02-16 |
| NZ522967A (en) | 2005-07-29 |
| HUP0300996A2 (hu) | 2003-08-28 |
| JP2003535135A (ja) | 2003-11-25 |
| PL360282A1 (en) | 2004-09-06 |
| MXPA02012072A (es) | 2004-08-19 |
| OA12285A (en) | 2006-05-12 |
| CA2411572C (fr) | 2009-11-10 |
| DZ3366A1 (fr) | 2001-12-13 |
| HUP0300996A3 (en) | 2006-02-28 |
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