ZA200209149B - 8ß-hydrocarbyl-substituted estratrienes for use as selective estrogens - Google Patents

8ß-hydrocarbyl-substituted estratrienes for use as selective estrogens Download PDF

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Publication number
ZA200209149B
ZA200209149B ZA200209149A ZA200209149A ZA200209149B ZA 200209149 B ZA200209149 B ZA 200209149B ZA 200209149 A ZA200209149 A ZA 200209149A ZA 200209149 A ZA200209149 A ZA 200209149A ZA 200209149 B ZA200209149 B ZA 200209149B
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group
hydrogen atom
radical
atom
estra
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ZA200209149A
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English (en)
Inventor
Peters Olaf
Thieme Ina
Hegele-Hartung Christa
Fritzemeier Karl-Heinrich
Hillisch Alexander
Elger Walter
Kollenkirchen Uwe
Patchev Vladimir
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Schering Ag
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Publication of ZA200209149B publication Critical patent/ZA200209149B/en

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    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
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    • C07J1/0059Estrane derivatives substituted in position 17 by a keto group
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    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
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    • A61P5/32Antioestrogens
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    • C07J1/0051Estrane derivatives
    • C07J1/0062Estrane derivatives substituted in position 17 alfa not substituted in position 17 beta
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    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
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    • C07J1/0051Estrane derivatives
    • C07J1/0066Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
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    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
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    • C07J1/0051Estrane derivatives
    • C07J1/0066Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
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    • C07J41/0072Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic

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ZA200209149A 2000-04-12 2002-11-11 8ß-hydrocarbyl-substituted estratrienes for use as selective estrogens ZA200209149B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10019167A DE10019167A1 (de) 2000-04-12 2000-04-12 Substituierte Estratriene als selektiv wirksame Estrogene

Publications (1)

Publication Number Publication Date
ZA200209149B true ZA200209149B (en) 2007-10-31

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ZA200209149A ZA200209149B (en) 2000-04-12 2002-11-11 8ß-hydrocarbyl-substituted estratrienes for use as selective estrogens

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JP (1) JP4860880B2 (sh)
KR (1) KR100825534B1 (sh)
AR (1) AR028329A1 (sh)
DE (2) DE10019167A1 (sh)
PE (1) PE20011215A1 (sh)
SI (1) SI1272504T1 (sh)
TW (1) TWI288138B (sh)
UA (1) UA79073C2 (sh)
UY (1) UY26665A1 (sh)
YU (1) YU77302A (sh)
ZA (1) ZA200209149B (sh)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0300335A2 (hu) * 2000-04-12 2003-07-28 Schering Ag. 8béta-hidrokarbil-szubsztituált ösztratriének mint szelektív hatású ösztrogének, alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények
DE10151114A1 (de) * 2001-10-15 2003-04-17 Schering Ag 8ß-Substituierte-11ß-aryl-estra-2,3,5(10)-trienderivate
PT1689410E (pt) * 2003-11-26 2008-08-18 Bayer Schering Pharma Ag Prevenção e tratamento de doenças cardíacas hipertensivas pelos estrogénios selectivos 8beta-vinil-estra-1,3,5(10)-trieno-3,17beta-diol e 17beta-fluoro-9alfa-vinil-estra-1,3,5(10)-trieno-3,16alfa-diol
WO2008064133A1 (en) * 2006-11-17 2008-05-29 Trustees Of Dartmouth College Synthesis and biological activities of new tricyclic-bis-enones (tbes)
EP2014672A1 (en) * 2007-07-12 2009-01-14 Bayer Schering Pharma Aktiengesellschaft 8-beta-substituted estratrienes as selectively active estrogens
JP2012509286A (ja) * 2008-11-21 2012-04-19 バイエル ファーマ アクチエンゲゼルシャフト 薬物送達システム

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3806546A (en) 1969-06-18 1974-04-23 American Cyanamid Co Steroid-like compounds and method of synthesis
US3681407A (en) 1969-06-18 1972-08-01 American Cyanamid Co 3-methoxy 8{62 -methylestra 1,3,5(10),9(11)-tetraene-17{62 -carboxylic acid lower alkyl ester and intermediates in the preparation thereof
US3736345A (en) 1971-05-18 1973-05-29 American Cyanamid Co Steroid-like compounds and method of synthesis

Also Published As

Publication number Publication date
UY26665A1 (es) 2001-11-30
DE10019167A1 (de) 2001-10-18
JP4860880B2 (ja) 2012-01-25
KR20030028734A (ko) 2003-04-10
KR100825534B1 (ko) 2008-04-25
JP2003534248A (ja) 2003-11-18
PE20011215A1 (es) 2001-11-29
SI1272504T1 (sl) 2007-10-31
UA79073C2 (en) 2007-05-25
YU77302A (sh) 2005-11-28
AR028329A1 (es) 2003-05-07
TWI288138B (en) 2007-10-11
DE50107204D1 (de) 2005-09-29

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