YU98003A - Supstituisana sulfonamidna jedinjenja, postupak za njihovu upotrebu kao leka za tretiranje poremećaja cns, gojaznosti i dijabetesa tipa ii - Google Patents

Supstituisana sulfonamidna jedinjenja, postupak za njihovu upotrebu kao leka za tretiranje poremećaja cns, gojaznosti i dijabetesa tipa ii

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Publication number
YU98003A
YU98003A YU98003A YUP98003A YU98003A YU 98003 A YU98003 A YU 98003A YU 98003 A YU98003 A YU 98003A YU P98003 A YUP98003 A YU P98003A YU 98003 A YU98003 A YU 98003A
Authority
YU
Yugoslavia
Prior art keywords
obesity
diabetes
treatment
type
medicament
Prior art date
Application number
YU98003A
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English (en)
Inventor
Katarina Beierlein
Ulf Bremberg
Patrizia Caldirola
Jensen Annika Jenmalm
Gary Johansson
Andrew Mott
Lars Tedenborg
Markus Thor
Original Assignee
Biovitrum Ab.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0102048A external-priority patent/SE0102048D0/xx
Priority claimed from SE0102386A external-priority patent/SE0102386D0/xx
Priority claimed from SE0103437A external-priority patent/SE0103437D0/xx
Application filed by Biovitrum Ab. filed Critical Biovitrum Ab.
Publication of YU98003A publication Critical patent/YU98003A/sh

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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
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  • Diabetes (AREA)
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  • Psychiatry (AREA)
  • Hematology (AREA)
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  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Addiction (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Quinoline Compounds (AREA)
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Abstract

Prikazani pronalazak se odnosi na jedinjenja supstituisanih sulfonamida opšte formule (I), gde P je sulfonamid ili amid-supstituisana sulfonska kiselina, a pomenuta jedinjenja su potencijalno korisna u profilaksi i lečenju medicinskih stanja koji su u vezi sa gojaznošću, dijabetisom tipa II i/ili poremećajima centralnog nervnog sistema.[The present invention relates to substituted sulfonamide compounds of the general formula (I), wherein P is sulfonamide or amide- substituted sulfonic acid, which compounds are potentially useful for the prophylaxis and treatment of medical conditions relating to obesity, type II diabetes and/or disorders of the central nervous system.
YU98003A 2001-06-11 2002-06-11 Supstituisana sulfonamidna jedinjenja, postupak za njihovu upotrebu kao leka za tretiranje poremećaja cns, gojaznosti i dijabetesa tipa ii YU98003A (sh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0102048A SE0102048D0 (sv) 2001-06-11 2001-06-11 New Compounds
SE0102386A SE0102386D0 (sv) 2001-07-03 2001-07-03 New compounds
SE0103437A SE0103437D0 (sv) 2001-10-16 2001-10-16 New compounds

Publications (1)

Publication Number Publication Date
YU98003A true YU98003A (sh) 2006-03-03

Family

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YU98003A YU98003A (sh) 2001-06-11 2002-06-11 Supstituisana sulfonamidna jedinjenja, postupak za njihovu upotrebu kao leka za tretiranje poremećaja cns, gojaznosti i dijabetesa tipa ii

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US (5) US7144883B2 (sh)
EP (1) EP1412325A1 (sh)
JP (2) JP4731114B2 (sh)
KR (3) KR100889718B1 (sh)
CN (2) CN100457726C (sh)
AU (1) AU2002309435B2 (sh)
BR (1) BR0210291A (sh)
CA (1) CA2445653A1 (sh)
EA (1) EA008476B1 (sh)
HK (1) HK1066790A1 (sh)
IL (1) IL158590A0 (sh)
MX (1) MXPA03011083A (sh)
NO (1) NO20035496D0 (sh)
NZ (1) NZ529032A (sh)
PL (1) PL367264A1 (sh)
WO (1) WO2002100822A1 (sh)
YU (1) YU98003A (sh)

Families Citing this family (78)

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Publication number Priority date Publication date Assignee Title
US7517884B2 (en) 1998-03-30 2009-04-14 Kalypsys Inc. Sulfonyl-substituted bicyclic compounds as modulators of PPAR
CN100457726C (zh) 2001-06-11 2009-02-04 比奥维特罗姆股份公开公司 取代的磺酰胺化合物、其制备方法及其作为治疗cns疾病、肥胖和ⅱ型糖尿病的药物的应用
CA2476173A1 (en) * 2002-02-22 2003-09-04 Ruth E. Tenbrink Arylsulfone derivatives
GB0204720D0 (en) * 2002-02-28 2002-04-17 Glaxo Group Ltd Novel use
EP1897881A3 (en) * 2002-06-20 2009-03-18 Biovitrum AB (publ) Compounds useful for the treatment of obesity, type II diabetes and CNS disorders
JP4754821B2 (ja) 2002-06-20 2011-08-24 プロキシマゲン・リミテッド 肥満症、ｉｉ型糖尿病およびｃｎｓ障害の治療に有用な新規化合物
NZ552283A (en) * 2002-06-20 2008-07-31 Biovitrum Ab Publ New compounds useful for the treatment of obesity, type II diabetes and CNS disorders
NZ538713A (en) 2002-08-12 2007-01-26 Takeda Chemical Industries Ltd Fused benzene derivative and use
SE0301446D0 (sv) * 2003-05-16 2003-05-16 Astrazeneca Ab New Compounds
ES2228268B1 (es) * 2003-07-30 2006-07-01 Laboratorios Del Dr. Esteve, S.A. Combinacion de sustancias activas conteniendo al menos un compuesto con afinidad por el receptor del neuropeptido y (npy) y al menos un compuesto con afinidad por el receptor 5-ht6.
ES2228267B1 (es) * 2003-07-30 2006-07-01 Laboratorios Del Dr. Esteve, S.A. Combinacion de sustancias activas conteniendo al menos un compuesto con afinidad por el receptor del neuropeptido y (npy) y al menos un compuesto con afinidad por el receptor 5-ht6.
GB0320320D0 (en) * 2003-08-29 2003-10-01 Glaxo Group Ltd Novel compounds
GB0321473D0 (en) 2003-09-12 2003-10-15 Glaxo Group Ltd Novel compounds
SE0302760D0 (sv) * 2003-10-20 2003-10-20 Biovitrum Ab New compounds
CA2545506A1 (en) * 2003-12-19 2005-06-30 Biovitrum Ab Novel benzofuran derivatives, which can be used in prophylaxis or treatment of 5-ht6 receptor-related disorder
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