WO2021010814A3 - Composiciones de recubrimientos en película para tabletas con brillantez incrementada, procedimiento de preparación y aplicación - Google Patents

Composiciones de recubrimientos en película para tabletas con brillantez incrementada, procedimiento de preparación y aplicación Download PDF

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Publication number
WO2021010814A3
WO2021010814A3 PCT/MX2020/050017 MX2020050017W WO2021010814A3 WO 2021010814 A3 WO2021010814 A3 WO 2021010814A3 MX 2020050017 W MX2020050017 W MX 2020050017W WO 2021010814 A3 WO2021010814 A3 WO 2021010814A3
Authority
WO
WIPO (PCT)
Prior art keywords
compositions
film coatings
film
coatings
glucopyranosyl
Prior art date
Application number
PCT/MX2020/050017
Other languages
English (en)
French (fr)
Other versions
WO2021010814A2 (es
Inventor
Francisco ESCORCIA RODRÍGUEZ
Maria de Lourdes GARCIA MONDRAGON
Ana Karen FLORES NAVARRETE
José Luis ESPITIA RODRIGUEZ
Original Assignee
Dva Farma Mexicana S.A. De C.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dva Farma Mexicana S.A. De C.V. filed Critical Dva Farma Mexicana S.A. De C.V.
Priority to BR112021015768A priority Critical patent/BR112021015768A2/pt
Priority to EP20839714.1A priority patent/EP4000605A4/en
Priority to US17/616,438 priority patent/US20220233450A1/en
Priority to PE2021002054A priority patent/PE20220805A1/es
Publication of WO2021010814A2 publication Critical patent/WO2021010814A2/es
Publication of WO2021010814A3 publication Critical patent/WO2021010814A3/es
Priority to CONC2022/0001370A priority patent/CO2022001370A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/2853—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2813—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/282—Organic compounds, e.g. fats
    • A61K9/2826—Sugars or sugar alcohols, e.g. sucrose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846—Poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)

Abstract

El presente documento describe composiciones y procedimientos de aplicación de recubrimiento de tabletas farmacéuticas, reconocidos como recubrimientos de película en donde se logra obtener producto final recubierto con brillantez superior a la alcanzable con composiciones típicas. La diferencia principal en la composición, está en la inclusión del producto derivado de isomaltulosa, el cual es una mezcla de 6-O-α-D-glucopiranosil-D-manitol dihidratado con 6-O-α-D-glucopiranosil-D-sorbitol, conocido como Isomalt, combinado con una variedad de polímeros filmógenos como copolímero de etilenglicol y alcohol polivinílico, copovidona, alcohol polivinílico, y derivados celulósicos, en donde las condiciones de proceso son ventajosas al ser posible manejar altas concentraciones de sólidos en su preparación y rangos temperaturas de aplicación más amplias que las normalmente recomendadas para recubrimientos de película.
PCT/MX2020/050017 2019-07-15 2020-07-13 Composiciones de recubrimientos en película para tabletas con brillantez incrementada, procedimiento de preparación y aplicación WO2021010814A2 (es)

Priority Applications (5)

Application Number Priority Date Filing Date Title
BR112021015768A BR112021015768A2 (pt) 2019-07-15 2020-07-13 Composições de revestimentos de película para comprimidos com brilho aumentado, preparação e aplicação do procedimento
EP20839714.1A EP4000605A4 (en) 2019-07-15 2020-07-13 COMPOSITIONS OF FILM COATINGS FOR TABLETS WITH INCREASED GLOSS, PROCESS FOR THEIR PREPARATION AND THEIR USE
US17/616,438 US20220233450A1 (en) 2019-07-15 2020-07-13 Compositions of film coatings for tablets with increased gloss, method for production thereof and application of same
PE2021002054A PE20220805A1 (es) 2019-07-15 2020-07-13 Composiciones de recubrimientos en pelicula para tabletas con brillantez incrementada, procedimiento de preparacion y aplicacion
CONC2022/0001370A CO2022001370A2 (es) 2019-07-15 2022-02-10 Composiciones de recubrimientos en película para tabletas con brillantez incrementada, procedimiento de preparación y aplicación

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
MX2019008440A MX2019008440A (es) 2019-07-15 2019-07-15 Composiciones de recubrimientos en pelicula para tabletas con brillantez incrementada, procedimiento de preparacion y aplicacion.
MXMX/A/2019/008440 2019-07-15

Publications (2)

Publication Number Publication Date
WO2021010814A2 WO2021010814A2 (es) 2021-01-21
WO2021010814A3 true WO2021010814A3 (es) 2021-04-15

Family

ID=74211167

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/MX2020/050017 WO2021010814A2 (es) 2019-07-15 2020-07-13 Composiciones de recubrimientos en película para tabletas con brillantez incrementada, procedimiento de preparación y aplicación

Country Status (8)

Country Link
US (1) US20220233450A1 (es)
EP (1) EP4000605A4 (es)
AR (1) AR119406A1 (es)
BR (1) BR112021015768A2 (es)
CO (1) CO2022001370A2 (es)
MX (1) MX2019008440A (es)
PE (1) PE20220805A1 (es)
WO (1) WO2021010814A2 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4324465A1 (en) * 2022-08-15 2024-02-21 Gedea Biotech AB Compounds for use in the treatment of a microbial infection in the urogenital system

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1989003678A1 (en) * 1987-10-30 1989-05-05 Stolle Research & Development Corporation Low residual solvent microspheres and microencapsulation process
US5665406A (en) * 1992-03-23 1997-09-09 Wm. Wrigley Jr. Company Polyol coated chewing gum having improved shelf life and method of making
US20040022755A1 (en) * 2002-08-02 2004-02-05 Satish Kamath Polyacrylic film forming compositions
US20170281553A1 (en) * 2010-05-11 2017-10-05 Sensient Colors Llc Film coating composition and methods of making and using the same

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10207427A1 (de) * 2002-02-21 2003-09-04 Basf Ag Schnelllöslicher Filmüberzug basierend auf Polyvinylalkohol-Polyether-Pfropfcopolymeren in Kombination mit Hydroxy-, Amid-, oder Esterfunktionen enthaltenden Komponenten
CA2566771A1 (en) * 2004-06-07 2005-12-22 Wyeth Sugar coatings and methods therefor
FR2921835B1 (fr) * 2007-10-05 2012-05-04 Soc Dexploitation De Produits Pour Les Industries Chimiques Seppic Composition d'enrobage comprenant du polydextrose, procede pour sa preparation et utilisation pour enrober les formes solides ingerables
CN101903017B (zh) 2008-01-10 2014-12-24 赢创罗姆有限公司 具有增强的脉冲活性物质释放的包衣的药物或营养制剂
US20090214699A1 (en) * 2008-02-25 2009-08-27 Bernd Hasslinger Coated comestibles and processes for their preparation
WO2010052727A1 (en) 2008-11-04 2010-05-14 Ideal Cures Private Limited High performance film coating compositions
EP2393360B1 (en) 2009-02-05 2015-11-04 Takeda Pharmaceutical Company Limited Pyridazinone compounds
BE1020860A3 (nl) 2012-08-09 2014-06-03 Ecover Co Ordination Ct Nv Tablet coating.
ES2953728T3 (es) * 2014-02-28 2023-11-15 Intercontinental Great Brands Llc Método para recubrir núcleos comestibles y el uso de un método para limitar la adherencia de los núcleos comestibles a la pared interior del tambor

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1989003678A1 (en) * 1987-10-30 1989-05-05 Stolle Research & Development Corporation Low residual solvent microspheres and microencapsulation process
US5665406A (en) * 1992-03-23 1997-09-09 Wm. Wrigley Jr. Company Polyol coated chewing gum having improved shelf life and method of making
US20040022755A1 (en) * 2002-08-02 2004-02-05 Satish Kamath Polyacrylic film forming compositions
US20170281553A1 (en) * 2010-05-11 2017-10-05 Sensient Colors Llc Film coating composition and methods of making and using the same

Also Published As

Publication number Publication date
EP4000605A4 (en) 2022-08-24
US20220233450A1 (en) 2022-07-28
WO2021010814A2 (es) 2021-01-21
MX2019008440A (es) 2021-01-18
EP4000605A2 (en) 2022-05-25
CO2022001370A2 (es) 2022-03-18
BR112021015768A2 (pt) 2022-02-08
AR119406A1 (es) 2021-12-15
PE20220805A1 (es) 2022-05-20

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